BE824742A - Nouveaux composes d'indole substitues en positions 1 et 2, leur procede de preparation et les preparations pharmaceutiques les contenant - Google Patents

Nouveaux composes d'indole substitues en positions 1 et 2, leur procede de preparation et les preparations pharmaceutiques les contenant

Info

Publication number
BE824742A
BE824742A BE152675A BE152675A BE824742A BE 824742 A BE824742 A BE 824742A BE 152675 A BE152675 A BE 152675A BE 152675 A BE152675 A BE 152675A BE 824742 A BE824742 A BE 824742A
Authority
BE
Belgium
Prior art keywords
positions
preparation process
pharmaceutical preparations
preparations containing
compounds substituted
Prior art date
Application number
BE152675A
Other languages
English (en)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of BE824742A publication Critical patent/BE824742A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BE152675A 1974-01-25 1975-01-24 Nouveaux composes d'indole substitues en positions 1 et 2, leur procede de preparation et les preparations pharmaceutiques les contenant BE824742A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH104774 1974-01-25

Publications (1)

Publication Number Publication Date
BE824742A true BE824742A (fr) 1975-07-24

Family

ID=4201215

Family Applications (1)

Application Number Title Priority Date Filing Date
BE152675A BE824742A (fr) 1974-01-25 1975-01-24 Nouveaux composes d'indole substitues en positions 1 et 2, leur procede de preparation et les preparations pharmaceutiques les contenant

Country Status (14)

Country Link
JP (1) JPS50106969A (fr)
AT (1) ATA53175A (fr)
AU (1) AU7756375A (fr)
BE (1) BE824742A (fr)
DE (1) DE2501468A1 (fr)
DK (1) DK3375A (fr)
ES (1) ES434079A1 (fr)
FR (1) FR2258853B1 (fr)
GB (1) GB1472342A (fr)
IE (1) IE40368B1 (fr)
IL (1) IL46505A0 (fr)
NL (1) NL7500535A (fr)
SE (1) SE7500262L (fr)
ZA (1) ZA75522B (fr)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4999186A (en) * 1986-06-27 1991-03-12 The Procter & Gamble Company Novel sunscreen agents, sunscreen compositions and methods for preventing sunburn
KR20030024661A (ko) * 2000-04-28 2003-03-26 박스터 헬쓰케어 에스.에이. 2-아실 인돌 유도체 및 항종양제로서의 이의 용도
DE10152306A1 (de) * 2001-10-26 2003-07-24 Asta Medica Ag 2-Acylindolderivate mit neuen therapeutisch wertvollen Eigenschaften
US20100298343A1 (en) * 2007-10-05 2010-11-25 John Howard Hutchinson 5-lipoxygenase-activating protein (flap) inhibitors
CN104945420A (zh) 2009-06-29 2015-09-30 因塞特公司 作为pi3k抑制剂的嘧啶酮类
US8759359B2 (en) 2009-12-18 2014-06-24 Incyte Corporation Substituted heteroaryl fused derivatives as PI3K inhibitors
TW201130842A (en) 2009-12-18 2011-09-16 Incyte Corp Substituted fused aryl and heteroaryl derivatives as PI3K inhibitors
JP5816678B2 (ja) 2010-04-14 2015-11-18 インサイト・コーポレイションIncyte Corporation PI3Kδ阻害剤としての縮合誘導体
US9062055B2 (en) 2010-06-21 2015-06-23 Incyte Corporation Fused pyrrole derivatives as PI3K inhibitors
AR084366A1 (es) 2010-12-20 2013-05-08 Incyte Corp N-(1-(fenil sustituido)etil)-9h-purin-6-aminas como inhibidores de pi3k
WO2012125629A1 (fr) 2011-03-14 2012-09-20 Incyte Corporation Dérivés diamino-pyrimidines et diamino-pyridines substituées en tant qu'inhibiteurs de pi3k
WO2012135009A1 (fr) 2011-03-25 2012-10-04 Incyte Corporation Dérivés de pyrimidine-4,6-diamine en tant qu'inhibiteurs de pi3k
HUE043703T2 (hu) 2011-09-02 2019-09-30 Incyte Holdings Corp Heterociklusos aminok PI3K inhibitorokként
AR090548A1 (es) 2012-04-02 2014-11-19 Incyte Corp Azaheterociclobencilaminas biciclicas como inhibidores de pi3k
US10077277B2 (en) 2014-06-11 2018-09-18 Incyte Corporation Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors
TWI764392B (zh) 2015-02-27 2022-05-11 美商英塞特公司 Pi3k抑制劑之鹽及製備方法
WO2016183063A1 (fr) 2015-05-11 2016-11-17 Incyte Corporation Formes cristallines d'un inhibiteur de pi3k
US9732097B2 (en) 2015-05-11 2017-08-15 Incyte Corporation Process for the synthesis of a phosphoinositide 3-kinase inhibitor

Also Published As

Publication number Publication date
JPS50106969A (fr) 1975-08-22
NL7500535A (nl) 1975-07-29
DE2501468A1 (de) 1975-07-31
ATA53175A (de) 1977-08-15
GB1472342A (en) 1977-05-04
AU7756375A (en) 1976-07-29
ZA75522B (en) 1976-01-28
FR2258853A1 (fr) 1975-08-22
IL46505A0 (en) 1975-04-25
SE7500262L (fr) 1975-07-28
FR2258853B1 (fr) 1978-06-30
IE40368L (en) 1975-07-25
IE40368B1 (en) 1979-05-09
DK3375A (fr) 1975-09-15
ES434079A1 (es) 1977-03-01

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