BE824742A - Nouveaux composes d'indole substitues en positions 1 et 2, leur procede de preparation et les preparations pharmaceutiques les contenant - Google Patents
Nouveaux composes d'indole substitues en positions 1 et 2, leur procede de preparation et les preparations pharmaceutiques les contenantInfo
- Publication number
- BE824742A BE824742A BE152675A BE152675A BE824742A BE 824742 A BE824742 A BE 824742A BE 152675 A BE152675 A BE 152675A BE 152675 A BE152675 A BE 152675A BE 824742 A BE824742 A BE 824742A
- Authority
- BE
- Belgium
- Prior art keywords
- positions
- preparation process
- pharmaceutical preparations
- preparations containing
- compounds substituted
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH104774 | 1974-01-25 |
Publications (1)
Publication Number | Publication Date |
---|---|
BE824742A true BE824742A (fr) | 1975-07-24 |
Family
ID=4201215
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE152675A BE824742A (fr) | 1974-01-25 | 1975-01-24 | Nouveaux composes d'indole substitues en positions 1 et 2, leur procede de preparation et les preparations pharmaceutiques les contenant |
Country Status (14)
Country | Link |
---|---|
JP (1) | JPS50106969A (fr) |
AT (1) | ATA53175A (fr) |
AU (1) | AU7756375A (fr) |
BE (1) | BE824742A (fr) |
DE (1) | DE2501468A1 (fr) |
DK (1) | DK3375A (fr) |
ES (1) | ES434079A1 (fr) |
FR (1) | FR2258853B1 (fr) |
GB (1) | GB1472342A (fr) |
IE (1) | IE40368B1 (fr) |
IL (1) | IL46505A0 (fr) |
NL (1) | NL7500535A (fr) |
SE (1) | SE7500262L (fr) |
ZA (1) | ZA75522B (fr) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4999186A (en) * | 1986-06-27 | 1991-03-12 | The Procter & Gamble Company | Novel sunscreen agents, sunscreen compositions and methods for preventing sunburn |
KR20030024661A (ko) * | 2000-04-28 | 2003-03-26 | 박스터 헬쓰케어 에스.에이. | 2-아실 인돌 유도체 및 항종양제로서의 이의 용도 |
DE10152306A1 (de) * | 2001-10-26 | 2003-07-24 | Asta Medica Ag | 2-Acylindolderivate mit neuen therapeutisch wertvollen Eigenschaften |
US20100298343A1 (en) * | 2007-10-05 | 2010-11-25 | John Howard Hutchinson | 5-lipoxygenase-activating protein (flap) inhibitors |
CN104945420A (zh) | 2009-06-29 | 2015-09-30 | 因塞特公司 | 作为pi3k抑制剂的嘧啶酮类 |
US8759359B2 (en) | 2009-12-18 | 2014-06-24 | Incyte Corporation | Substituted heteroaryl fused derivatives as PI3K inhibitors |
TW201130842A (en) | 2009-12-18 | 2011-09-16 | Incyte Corp | Substituted fused aryl and heteroaryl derivatives as PI3K inhibitors |
JP5816678B2 (ja) | 2010-04-14 | 2015-11-18 | インサイト・コーポレイションIncyte Corporation | PI3Kδ阻害剤としての縮合誘導体 |
US9062055B2 (en) | 2010-06-21 | 2015-06-23 | Incyte Corporation | Fused pyrrole derivatives as PI3K inhibitors |
AR084366A1 (es) | 2010-12-20 | 2013-05-08 | Incyte Corp | N-(1-(fenil sustituido)etil)-9h-purin-6-aminas como inhibidores de pi3k |
WO2012125629A1 (fr) | 2011-03-14 | 2012-09-20 | Incyte Corporation | Dérivés diamino-pyrimidines et diamino-pyridines substituées en tant qu'inhibiteurs de pi3k |
WO2012135009A1 (fr) | 2011-03-25 | 2012-10-04 | Incyte Corporation | Dérivés de pyrimidine-4,6-diamine en tant qu'inhibiteurs de pi3k |
HUE043703T2 (hu) | 2011-09-02 | 2019-09-30 | Incyte Holdings Corp | Heterociklusos aminok PI3K inhibitorokként |
AR090548A1 (es) | 2012-04-02 | 2014-11-19 | Incyte Corp | Azaheterociclobencilaminas biciclicas como inhibidores de pi3k |
US10077277B2 (en) | 2014-06-11 | 2018-09-18 | Incyte Corporation | Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors |
TWI764392B (zh) | 2015-02-27 | 2022-05-11 | 美商英塞特公司 | Pi3k抑制劑之鹽及製備方法 |
WO2016183063A1 (fr) | 2015-05-11 | 2016-11-17 | Incyte Corporation | Formes cristallines d'un inhibiteur de pi3k |
US9732097B2 (en) | 2015-05-11 | 2017-08-15 | Incyte Corporation | Process for the synthesis of a phosphoinositide 3-kinase inhibitor |
-
1975
- 1975-01-08 DK DK3375*BA patent/DK3375A/da unknown
- 1975-01-10 SE SE7500262A patent/SE7500262L/xx unknown
- 1975-01-16 NL NL7500535A patent/NL7500535A/xx unknown
- 1975-01-16 DE DE19752501468 patent/DE2501468A1/de active Pending
- 1975-01-23 ES ES434079A patent/ES434079A1/es not_active Expired
- 1975-01-23 AU AU77563/75A patent/AU7756375A/en not_active Expired
- 1975-01-23 GB GB299475A patent/GB1472342A/en not_active Expired
- 1975-01-23 FR FR7502129A patent/FR2258853B1/fr not_active Expired
- 1975-01-24 IL IL46505A patent/IL46505A0/xx unknown
- 1975-01-24 IE IE137/75A patent/IE40368B1/xx unknown
- 1975-01-24 BE BE152675A patent/BE824742A/fr unknown
- 1975-01-24 ZA ZA00750522A patent/ZA75522B/xx unknown
- 1975-01-24 AT AT53175A patent/ATA53175A/de not_active IP Right Cessation
- 1975-01-25 JP JP50010179A patent/JPS50106969A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
JPS50106969A (fr) | 1975-08-22 |
NL7500535A (nl) | 1975-07-29 |
DE2501468A1 (de) | 1975-07-31 |
ATA53175A (de) | 1977-08-15 |
GB1472342A (en) | 1977-05-04 |
AU7756375A (en) | 1976-07-29 |
ZA75522B (en) | 1976-01-28 |
FR2258853A1 (fr) | 1975-08-22 |
IL46505A0 (en) | 1975-04-25 |
SE7500262L (fr) | 1975-07-28 |
FR2258853B1 (fr) | 1978-06-30 |
IE40368L (en) | 1975-07-25 |
IE40368B1 (en) | 1979-05-09 |
DK3375A (fr) | 1975-09-15 |
ES434079A1 (es) | 1977-03-01 |
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