BE790287A - Acides pyrimidin-6yl acethydroxamiques, leur procede de preparation et leur application en therapeutique - Google Patents

Acides pyrimidin-6yl acethydroxamiques, leur procede de preparation et leur application en therapeutique

Info

Publication number
BE790287A
BE790287A BE790287DA BE790287A BE 790287 A BE790287 A BE 790287A BE 790287D A BE790287D A BE 790287DA BE 790287 A BE790287 A BE 790287A
Authority
BE
Belgium
Prior art keywords
acethydroxamic
pyrimidin
acids
preparation process
therapeutic application
Prior art date
Application number
Other languages
English (en)
French (fr)
Inventor
C Fauran
G Raynaud
G Bourgery
C Couret
J Eberle
Original Assignee
Delalande Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Publication date
Publication of BE790287A publication Critical patent/BE790287A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32One oxygen, sulfur or nitrogen atom
    • C07D239/42One nitrogen atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
BE790287D 1971-10-28 Acides pyrimidin-6yl acethydroxamiques, leur procede de preparation et leur application en therapeutique BE790287A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7138788A FR2158081B1 (de) 1971-10-28 1971-10-28

Publications (1)

Publication Number Publication Date
BE790287A true BE790287A (fr) 1973-04-19

Family

ID=9085023

Family Applications (1)

Application Number Title Priority Date Filing Date
BE790287D BE790287A (fr) 1971-10-28 Acides pyrimidin-6yl acethydroxamiques, leur procede de preparation et leur application en therapeutique

Country Status (15)

Country Link
US (1) US3876636A (de)
JP (1) JPS535677B2 (de)
AU (1) AU465951B2 (de)
BE (1) BE790287A (de)
CA (1) CA980775A (de)
CH (1) CH551418A (de)
DE (1) DE2252822C3 (de)
ES (1) ES407913A1 (de)
FR (2) FR2158081B1 (de)
GB (1) GB1339389A (de)
LU (1) LU66378A1 (de)
NL (1) NL7214533A (de)
SE (1) SE398349B (de)
SU (1) SU490290A3 (de)
ZA (1) ZA727579B (de)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE826017R (fr) * 1974-03-19 1975-08-26 Acides pyrimidin-6yl acethydroxamiques, leur procede de preparation et leur application en therapeutique
IT1192287B (it) * 1977-11-14 1988-03-31 Fujisawa Pharmaceutical Co Derivati di acido cefalosporanico ad azione farmaceutica e relativo procedimento di preparazione
US4604466A (en) * 1983-08-02 1986-08-05 Riker Laboratories, Inc. Piperidine-substituted pyrimidines
JPH0720943B2 (ja) * 1988-08-19 1995-03-08 宇部興産株式会社 アミノピリミジン誘導体、その製法及び殺虫・殺菌剤
JPH0567317A (ja) * 1991-09-06 1993-03-19 Pioneer Electron Corp 細部クリーニング用ブラシ及びその製造方法
US6369222B1 (en) * 2000-07-18 2002-04-09 Hoffmann-La Roche Inc. mGluR antagonists and a method for their synthesis
JP5543354B2 (ja) * 2007-10-19 2014-07-09 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ γ−セクレターゼのアミン結合調節物質
EP2215043B1 (de) * 2007-10-19 2013-03-06 Janssen Pharmaceutica, N.V. Kohlenstoffgebundene modulatoren von y-sekretase
EA017119B1 (ru) * 2007-10-19 2012-09-28 Янссен Фармацевтика, Н.В. МОДУЛЯТОРЫ АКТИВНОСТИ γ-СЕКРЕТАЗЫ ИЗ ГРУППЫ ПИПЕРИДИНИЛА И ПИПЕРАЗИНИЛА

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR819596A (fr) * 1936-03-31 1937-10-21 Ig Farbenindustrie Ag Dérivés pyrimidiques
GB1174165A (en) * 1966-04-20 1969-12-17 Basf Ag Production of Pyrimidines Bearing a Halogen as Substituent in the 5-Position
FR1526533A (fr) * 1966-06-09 1968-05-24 Takeda Chemical Industries Ltd Procédé de production de 4-amino-5-acylamidométhyl pyrimidines 2-substituées
GB1121922A (en) * 1966-06-17 1968-07-31 Ici Ltd Pyrimidine derivatives

Also Published As

Publication number Publication date
CA980775A (en) 1975-12-30
SE398349B (sv) 1977-12-19
FR2225154B2 (de) 1976-07-02
CH551418A (fr) 1974-07-15
NL7214533A (de) 1973-05-02
DE2252822B2 (de) 1975-09-18
SU490290A3 (ru) 1975-10-30
US3876636A (en) 1975-04-08
FR2158081A1 (de) 1973-06-15
AU4811072A (en) 1974-04-26
JPS535677B2 (de) 1978-03-01
LU66378A1 (de) 1973-05-03
JPS495979A (de) 1974-01-19
FR2158081B1 (de) 1975-06-06
DE2252822C3 (de) 1976-05-06
FR2225154A2 (en) 1974-11-08
AU465951B2 (en) 1975-10-09
ZA727579B (en) 1973-07-25
DE2252822A1 (de) 1973-05-03
GB1339389A (en) 1973-12-05
ES407913A1 (es) 1975-11-16

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