BE777689A - Nouveaux derives de l'imidazoline, compositions therapeutiques les contenant ainsi que le procede de preparation de ces derives et de ces compositions - Google Patents
Nouveaux derives de l'imidazoline, compositions therapeutiques les contenant ainsi que le procede de preparation de ces derives et de ces compositionsInfo
- Publication number
- BE777689A BE777689A BE777689A BE777689A BE777689A BE 777689 A BE777689 A BE 777689A BE 777689 A BE777689 A BE 777689A BE 777689 A BE777689 A BE 777689A BE 777689 A BE777689 A BE 777689A
- Authority
- BE
- Belgium
- Prior art keywords
- derivatives
- imidazoline
- preparation
- compositions
- compositions containing
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title 2
- 150000002462 imidazolines Chemical class 0.000 title 1
- 230000001225 therapeutic effect Effects 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB332771 | 1971-01-27 |
Publications (1)
Publication Number | Publication Date |
---|---|
BE777689A true BE777689A (fr) | 1972-07-05 |
Family
ID=9756227
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE777689A BE777689A (fr) | 1971-01-27 | 1972-01-05 | Nouveaux derives de l'imidazoline, compositions therapeutiques les contenant ainsi que le procede de preparation de ces derives et de ces compositions |
Country Status (17)
Country | Link |
---|---|
US (1) | US3818035A (en:Method) |
JP (1) | JPS4938273B1 (en:Method) |
AT (1) | AT311336B (en:Method) |
BE (1) | BE777689A (en:Method) |
CA (1) | CA962273A (en:Method) |
CH (1) | CH535254A (en:Method) |
DE (1) | DE2203373C3 (en:Method) |
DK (1) | DK138496B (en:Method) |
FI (1) | FI55841C (en:Method) |
GB (1) | GB1333471A (en:Method) |
HU (1) | HU162823B (en:Method) |
NL (1) | NL150454B (en:Method) |
NO (1) | NO134115C (en:Method) |
SE (1) | SE378426B (en:Method) |
SU (1) | SU474145A3 (en:Method) |
YU (1) | YU34694B (en:Method) |
ZA (1) | ZA72286B (en:Method) |
Families Citing this family (28)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3927023A (en) * | 1974-05-24 | 1975-12-16 | Warner Lambert Co | Imidazolyl benzofurans |
DE3049542A1 (de) * | 1980-12-31 | 1982-07-29 | Basf Ag, 6700 Ludwigshafen | Azolylalkyl-2,3-dihydrobenzofurane, diese enthaltende fungizide und verfahren zu ihrer herstellung |
ZA825413B (en) * | 1981-08-26 | 1983-06-29 | Pfizer | Thromboxane synthetase inhibitors, processes for their production, and pharmaceutical compositions comprising them |
US4851554A (en) * | 1987-04-06 | 1989-07-25 | University Of Tennessee Research Corporation | Certain 3-substituted 2-alkyl benzofuran derivatives |
US4806663A (en) * | 1987-04-06 | 1989-02-21 | The University Of Tennessee Research Corporation | Certain 3-substituted 2-alkyl benzofuran derivatives |
US4831156A (en) * | 1987-09-30 | 1989-05-16 | The University Of Tennessee Research Corp. | 3-substituted 2-alkyl indole derivatives |
CA2315226A1 (en) * | 1997-12-19 | 1999-07-01 | Eli Lilly And Company | Hypoglycemic imidazoline compounds |
US7777035B2 (en) | 2005-06-22 | 2010-08-17 | Chemocentryx, Inc. | Azaindazole compounds and methods of use |
CA2637312A1 (en) * | 2006-01-27 | 2007-08-02 | F. Hoffmann-La Roche Ag | Use of substituted 2-imidazole of imidazoline derivatives |
CA2665255A1 (en) * | 2006-10-19 | 2008-04-24 | F. Hoffmann-La Roche Ag | Aminomethyl-2-imidazoles with affinity with the trace amine associated receptors |
JP5335681B2 (ja) * | 2006-10-19 | 2013-11-06 | エフ.ホフマン−ラ ロシュ アーゲー | アミノメチル−4−イミダゾール |
ES2375578T3 (es) * | 2006-11-02 | 2012-03-02 | F. Hoffmann-La Roche Ag | 2-imidazoles sustituidos como moduladores de receptores asociados a aminas trazas. |
JP2010510184A (ja) * | 2006-11-16 | 2010-04-02 | エフ.ホフマン−ラ ロシュ アーゲー | 置換4−イミダゾール類 |
KR101189348B1 (ko) * | 2006-12-13 | 2012-10-09 | 에프. 호프만-라 로슈 아게 | 미량 아민 결합 수용체(taar)에 대한 리간드로서의 신규한 2-이미다졸 |
US20080146523A1 (en) | 2006-12-18 | 2008-06-19 | Guido Galley | Imidazole derivatives |
ES2510546T3 (es) * | 2007-02-02 | 2014-10-21 | F. Hoffmann-La Roche Ag | Nuevas 2-aminooxazolinas como ligandos TAAR1 para trastornos del SNC |
AU2008214774A1 (en) * | 2007-02-15 | 2008-08-21 | F. Hoffmann-La Roche Ag | 2-aminooxazolines as TAAR1 ligands |
EP2173720A2 (en) | 2007-07-02 | 2010-04-14 | F. Hoffmann-Roche AG | 2-imidazolines having a good affinity to the trace amine associated receptors (taars) |
BRPI0812833A2 (pt) * | 2007-07-03 | 2014-12-09 | Hoffmann La Roche | 4-imidazolinas e seu uso como antidepressivos |
EP2183216A1 (en) * | 2007-07-27 | 2010-05-12 | F. Hoffmann-Roche AG | 2-azetidinemethaneamines and 2-pyrrolidinemethaneamines as taar-ligands |
EP2182935A1 (en) * | 2007-08-02 | 2010-05-12 | F. Hoffmann-Roche AG | The use of benzamide derivatives for the treatment of cns disorders |
JP5341084B2 (ja) * | 2007-08-03 | 2013-11-13 | エフ.ホフマン−ラ ロシュ アーゲー | Taar1リガンドとしてのピリジンカルボキシアミド及びベンズアミド誘導体 |
US8242153B2 (en) * | 2008-07-24 | 2012-08-14 | Hoffmann-La Roche Inc. | 4,5-dihydro-oxazol-2YL derivatives |
CA2728480A1 (en) * | 2008-07-24 | 2010-01-28 | F. Hoffmann-La Roche Ag | 4,5-dihydro-oxazol-2-yl derivatives |
US20100311798A1 (en) * | 2009-06-05 | 2010-12-09 | Decoret Guillaume | 2-aminooxazolines as taar1 ligands |
US8354441B2 (en) * | 2009-11-11 | 2013-01-15 | Hoffmann-La Roche Inc. | Oxazoline derivatives |
US9452980B2 (en) | 2009-12-22 | 2016-09-27 | Hoffmann-La Roche Inc. | Substituted benzamides |
HRP20201405T1 (hr) | 2016-03-17 | 2020-11-27 | F. Hoffmann - La Roche Ag | Derivat 5-etil-4-metil-pirazol-3-karboksamida, koji djeluje kao agonist taar-a |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE1121054B (de) * | 1960-11-23 | 1962-01-04 | Merck Ag E | Verfahren zur Herstellung eines neuen Imidazolinderivates und dessen Saeureadditionssalzen |
-
1971
- 1971-01-27 GB GB332771A patent/GB1333471A/en not_active Expired
-
1972
- 1972-01-05 BE BE777689A patent/BE777689A/xx not_active IP Right Cessation
- 1972-01-06 CH CH17272A patent/CH535254A/fr not_active IP Right Cessation
- 1972-01-10 US US00216795A patent/US3818035A/en not_active Expired - Lifetime
- 1972-01-17 ZA ZA720286A patent/ZA72286B/xx unknown
- 1972-01-25 DE DE2203373A patent/DE2203373C3/de not_active Expired
- 1972-01-26 NO NO192/72A patent/NO134115C/no unknown
- 1972-01-26 YU YU181/72A patent/YU34694B/xx unknown
- 1972-01-26 HU HULA791A patent/HU162823B/hu not_active IP Right Cessation
- 1972-01-26 DK DK34572AA patent/DK138496B/da unknown
- 1972-01-26 SE SE7200867A patent/SE378426B/xx unknown
- 1972-01-27 SU SU1742351A patent/SU474145A3/ru active
- 1972-01-27 FI FI219/72A patent/FI55841C/fi active
- 1972-01-27 NL NL727201121A patent/NL150454B/xx not_active IP Right Cessation
- 1972-01-27 JP JP47010207A patent/JPS4938273B1/ja active Pending
- 1972-01-27 AT AT64772A patent/AT311336B/de not_active IP Right Cessation
- 1972-01-27 CA CA133,337A patent/CA962273A/en not_active Expired
Also Published As
Publication number | Publication date |
---|---|
AU3817772A (en) | 1973-07-26 |
DE2203373A1 (de) | 1972-08-17 |
DE2203373C3 (de) | 1978-04-13 |
AT311336B (de) | 1973-11-12 |
DK138496C (en:Method) | 1979-02-26 |
SU474145A3 (ru) | 1975-06-14 |
CA962273A (en) | 1975-02-04 |
CH535254A (fr) | 1973-03-31 |
SE378426B (en:Method) | 1975-09-01 |
DK138496B (da) | 1978-09-18 |
DE2203373B2 (de) | 1977-08-11 |
NO134115B (en:Method) | 1976-05-10 |
NL7201121A (en:Method) | 1972-07-31 |
JPS4938273B1 (en:Method) | 1974-10-16 |
US3818035A (en) | 1974-06-18 |
FI55841C (fi) | 1979-10-10 |
YU18172A (en) | 1979-07-10 |
ZA72286B (en) | 1972-09-27 |
GB1333471A (en) | 1973-10-10 |
HU162823B (en:Method) | 1973-04-28 |
YU34694B (en) | 1979-12-31 |
NL150454B (nl) | 1976-08-16 |
NO134115C (en:Method) | 1976-08-18 |
FI55841B (fi) | 1979-06-29 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RE | Patent lapsed |
Owner name: SANOFI Effective date: 19900131 |