BE762758A - Nouvelles 1-polyfluoroalcoyl-benzodiazepines et leurs procede de preparation - Google Patents

Nouvelles 1-polyfluoroalcoyl-benzodiazepines et leurs procede de preparation

Info

Publication number
BE762758A
BE762758A BE762758A BE762758A BE762758A BE 762758 A BE762758 A BE 762758A BE 762758 A BE762758 A BE 762758A BE 762758 A BE762758 A BE 762758A BE 762758 A BE762758 A BE 762758A
Authority
BE
Belgium
Prior art keywords
polyfluoroalcoyl
benzodiazepines
new
preparation process
preparation
Prior art date
Application number
BE762758A
Other languages
English (en)
Inventor
M Steinman Qui A C Corporation
Original Assignee
Scherico Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Scherico Ltd filed Critical Scherico Ltd
Publication of BE762758A publication Critical patent/BE762758A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BE762758A 1970-02-13 1971-02-10 Nouvelles 1-polyfluoroalcoyl-benzodiazepines et leurs procede de preparation BE762758A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US1133670A 1970-02-13 1970-02-13

Publications (1)

Publication Number Publication Date
BE762758A true BE762758A (fr) 1971-08-10

Family

ID=21749938

Family Applications (1)

Application Number Title Priority Date Filing Date
BE762758A BE762758A (fr) 1970-02-13 1971-02-10 Nouvelles 1-polyfluoroalcoyl-benzodiazepines et leurs procede de preparation

Country Status (22)

Country Link
US (1) US3723414A (fr)
AT (1) AT305286B (fr)
BE (1) BE762758A (fr)
CA (1) CA967152A (fr)
CH (1) CH581636A5 (fr)
CY (1) CY835A (fr)
DE (2) DE2115906A1 (fr)
ES (1) ES388129A1 (fr)
FI (1) FI52978C (fr)
FR (1) FR2081510B1 (fr)
GB (1) GB1297206A (fr)
HK (1) HK13576A (fr)
IE (1) IE35306B1 (fr)
IL (1) IL36163A (fr)
KE (1) KE2597A (fr)
MY (1) MY7600086A (fr)
NL (1) NL7101705A (fr)
NO (1) NO132799C (fr)
PL (1) PL88933B1 (fr)
SE (1) SE384858B (fr)
SU (1) SU437295A3 (fr)
ZA (1) ZA71812B (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2221558A1 (de) 1972-05-03 1973-11-15 Kali Chemie Ag Neue benzodiazepinderivate und verfahren zu deren herstellung

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU678503B2 (en) * 1993-09-24 1997-05-29 Takeda Chemical Industries Ltd. Condensed heterocyclic compounds and their use as squalene synthetase inhibitors

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3131178A (en) * 1964-04-28 Process for producing s-phenyl-l
US3501460A (en) * 1966-06-03 1970-03-17 Hoffmann La Roche Dehydration process for forming benzodiazepines
US3429874A (en) * 1966-12-22 1969-02-25 Schering Corp 1-polyhalogenoalkyl-2-oxo-1,3-dihydro-2h-1,4-benzodiazepines
US3523939A (en) * 1967-07-03 1970-08-11 Hoffmann La Roche 5-(2,6-disubstituted phenyl)-1,4-benzodiazepines and methods for their preparation
US3546212A (en) * 1968-06-12 1970-12-08 Hoffmann La Roche Oxidation of benzodiazepines with ruthenium tetroxide
FR2024239B1 (fr) * 1968-11-26 1973-01-12 Scherico Ltd

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2221558A1 (de) 1972-05-03 1973-11-15 Kali Chemie Ag Neue benzodiazepinderivate und verfahren zu deren herstellung
DE2265370C2 (de) * 1972-05-03 1982-12-02 Kali-Chemie Ag, 3000 Hannover 6-Phenyl-1,2,3,4-tetrahydro-1,5-benzodiazocinderivate

Also Published As

Publication number Publication date
DE2115906A1 (de) 1971-10-21
PL88933B1 (fr) 1976-10-30
NO132799C (fr) 1976-01-07
DE2106175A1 (de) 1971-09-30
SU437295A3 (ru) 1974-07-25
FR2081510B1 (fr) 1974-09-27
IL36163A (en) 1976-09-30
MY7600086A (en) 1976-12-31
FI52978C (fr) 1978-01-10
FI52978B (fr) 1977-09-30
SE384858B (sv) 1976-05-24
ES388129A1 (es) 1973-05-01
US3723414A (en) 1973-03-27
CA967152A (en) 1975-05-06
IE35306B1 (en) 1976-01-07
NL7101705A (fr) 1971-08-17
IE35306L (en) 1971-08-13
FR2081510A1 (fr) 1971-12-03
NO132799B (fr) 1975-09-29
KE2597A (en) 1976-02-27
ZA71812B (en) 1971-10-27
CY835A (en) 1976-09-10
GB1297206A (fr) 1972-11-22
AT305286B (de) 1973-02-26
IL36163A0 (en) 1971-04-28
HK13576A (en) 1976-03-19
CH581636A5 (fr) 1976-11-15

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