BE688539A - - Google Patents

Info

Publication number
BE688539A
BE688539A BE688539DA BE688539A BE 688539 A BE688539 A BE 688539A BE 688539D A BE688539D A BE 688539DA BE 688539 A BE688539 A BE 688539A
Authority
BE
Belgium
Application number
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of BE688539A publication Critical patent/BE688539A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06Pyrimidine radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BE688539D 1965-10-22 1966-10-20 BE688539A (US08197722-20120612-C00093.png)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US502586A US3309359A (en) 1965-10-22 1965-10-22 N-mono-acyl-5-fluorocytosine derivatives and process

Publications (1)

Publication Number Publication Date
BE688539A true BE688539A (US08197722-20120612-C00093.png) 1967-04-20

Family

ID=23998481

Family Applications (1)

Application Number Title Priority Date Filing Date
BE688539D BE688539A (US08197722-20120612-C00093.png) 1965-10-22 1966-10-20

Country Status (11)

Country Link
US (1) US3309359A (US08197722-20120612-C00093.png)
BE (1) BE688539A (US08197722-20120612-C00093.png)
BR (1) BR6683864D0 (US08197722-20120612-C00093.png)
CH (1) CH475258A (US08197722-20120612-C00093.png)
DE (1) DE1695160A1 (US08197722-20120612-C00093.png)
DK (1) DK115474B (US08197722-20120612-C00093.png)
FR (1) FR5908M (US08197722-20120612-C00093.png)
GB (1) GB1110357A (US08197722-20120612-C00093.png)
IL (1) IL26726A (US08197722-20120612-C00093.png)
NL (1) NL6614240A (US08197722-20120612-C00093.png)
SE (1) SE330176B (US08197722-20120612-C00093.png)

Families Citing this family (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3894000A (en) * 1971-01-27 1975-07-08 Upjohn Co Ara-cytidine derivatives and process of preparation
US3975367A (en) * 1971-06-08 1976-08-17 The Upjohn Company Arabinofuranosyl N4 -aminoacyl cytosine containing compounds
US4022963A (en) * 1972-06-08 1977-05-10 Deutsch Daniel Harold Acetylation process for nucleoside compounds
US3991045A (en) * 1973-05-30 1976-11-09 Asahi Kasei Kogyo Kabushiki Kaisha N4 -acylarabinonucleosides
JPS5159880A (en) * 1974-11-22 1976-05-25 Asahi Chemical Ind N44 ashirunukureoshidojikarubonsanesuteruno seiho
JPS5924999B2 (ja) * 1978-06-10 1984-06-13 富山化学工業株式会社 新規な5−フルオロ−2′−デオキシ−β−ウリジン誘導体の製造法
JPS5535057A (en) * 1978-09-05 1980-03-11 Funai Corp 2'-deoxy-5-fluorouridine derivative, its preparation, and antitumor agent comprising it
JPS59167600A (ja) * 1983-03-14 1984-09-21 Microbial Chem Res Found 2′−デオキシオキザノシンおよびその製造法
KR100978904B1 (ko) 2001-12-14 2010-08-31 파마셋 인코포레이티드 바이러스 감염 치료용 n4-아실사이토신 뉴클레오사이드
JP5749017B2 (ja) * 2008-01-22 2015-07-15 ダウ アグロサイエンシィズ エルエルシー 5−フルオロピリミジン誘導体
RU2536492C2 (ru) * 2008-08-01 2014-12-27 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи Применение 5-фторцитозина в качестве фунгицида
PT2462134E (pt) * 2009-08-07 2014-07-28 Dow Agrosciences Llc Derivados de n1-sulfonil-5-fluoropirimidinona
UA106889C2 (uk) * 2009-08-07 2014-10-27 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Похідні n1-ацил-5-фторпіримідинону
UA107671C2 (en) * 2009-08-07 2015-02-10 Dow Agrosciences Llc N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
UA112284C2 (uk) * 2009-08-07 2016-08-25 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Похідні 5-фторпіримідинону
EP2521452B1 (en) * 2010-01-07 2014-12-24 Dow AgroSciences LLC THIAZOLO[5,4-d]PYRIMIDINES AND THEIR USE AS AGROCHEMICALS
RU2613451C2 (ru) 2011-08-17 2017-03-16 Адама Мактешим Лтд. Производные 5-фтор-4-имино-3-(замещенного)-3, 4-дигидропиримидин-2(1н)она, композиция на их основе и спсоб борьбы с грибковыми заболеваниями
CA2893778A1 (en) 2012-12-28 2014-07-03 Dow Agrosciences Llc N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2h)-carboxylate derivatives
JP6258969B2 (ja) 2012-12-28 2018-01-10 アダマ・マクテシム・リミテッド N−(置換)−5−フルオロ−4−イミノ−3−メチル−2−オキソ−3,4−ジヒドロピリミジン−1(2h)−カルボキサミド誘導体
CN104994859B (zh) 2012-12-28 2018-10-26 阿达玛马克西姆股份有限公司 1-(取代的苯甲酰基)-5-氟-4-亚氨基-3-甲基-3,4-二氢嘧啶-2(1h)-酮衍生物
AU2013370494B2 (en) 2012-12-31 2017-08-17 Adama Makhteshim Ltd. 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1H)-one derivatives as fungicides
BR112016015158A2 (pt) 2013-12-31 2017-08-08 Adama Makhteshim Ltd Misturas fungicidas sinergísticas para controle de fungos em cereais
CA2935601C (en) 2013-12-31 2023-03-14 Adama Makhteshim Ltd. 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
WO2019038583A1 (en) 2017-07-17 2019-02-28 Adama Makhteshim Ltd. 5-FLUORO-4-IMINO-3-METHYL-1-TOSYL-3,4-DIHYDROPYRIMIDIN-2-ONE POLYMORPHS
CN109651467A (zh) * 2019-01-15 2019-04-19 齐鲁天和惠世制药有限公司 一种卡培他滨杂质及其制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2949451A (en) * 1959-04-21 1960-08-16 Hoffmann La Roche Preparation of thymidine and deoxyfluorouridine, and intermediates therefor
NL299755A (US08197722-20120612-C00093.png) * 1959-06-03
GB1070413A (en) * 1962-11-15 1967-06-01 Sankyo Co A process for preparing purine and pyrimidine nucleosides

Also Published As

Publication number Publication date
US3309359A (en) 1967-03-14
CH475258A (de) 1969-07-15
DK115474B (da) 1969-10-13
SE330176B (US08197722-20120612-C00093.png) 1970-11-09
NL6614240A (US08197722-20120612-C00093.png) 1967-04-24
DE1695160A1 (de) 1970-12-17
GB1110357A (en) 1968-04-18
IL26726A (en) 1970-06-17
FR5908M (US08197722-20120612-C00093.png) 1968-03-25
BR6683864D0 (pt) 1973-12-26

Similar Documents

Publication Publication Date Title
FR5908M (US08197722-20120612-C00093.png)
FI43303B (US08197722-20120612-C00093.png)
JPS4318781Y1 (US08197722-20120612-C00093.png)
JPS443838Y1 (US08197722-20120612-C00093.png)
JPS436059Y1 (US08197722-20120612-C00093.png)
JPS465922Y1 (US08197722-20120612-C00093.png)
JPS426556Y1 (US08197722-20120612-C00093.png)
JPS4316451Y1 (US08197722-20120612-C00093.png)
JPS4327560Y1 (US08197722-20120612-C00093.png)
JPS444127Y1 (US08197722-20120612-C00093.png)
JPS4631238Y1 (US08197722-20120612-C00093.png)
AU6702965A (US08197722-20120612-C00093.png)
BE666660A (US08197722-20120612-C00093.png)
BE660222A (US08197722-20120612-C00093.png)
BE665556A (US08197722-20120612-C00093.png)
BE665642A (US08197722-20120612-C00093.png)
LU51005A1 (US08197722-20120612-C00093.png)
BE666481A (US08197722-20120612-C00093.png)
NL6515491A (US08197722-20120612-C00093.png)
NL6603814A (US08197722-20120612-C00093.png)
BE665030A (US08197722-20120612-C00093.png)
BE670827A (US08197722-20120612-C00093.png)
BE664769A (US08197722-20120612-C00093.png)
BE667205A (US08197722-20120612-C00093.png)
BE667503A (US08197722-20120612-C00093.png)