BE1002179A5 - Compositions pharmaceutiques contenant des pyranoquinoleines. - Google Patents

Compositions pharmaceutiques contenant des pyranoquinoleines. Download PDF

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Publication number
BE1002179A5
BE1002179A5 BE8701471A BE8701471A BE1002179A5 BE 1002179 A5 BE1002179 A5 BE 1002179A5 BE 8701471 A BE8701471 A BE 8701471A BE 8701471 A BE8701471 A BE 8701471A BE 1002179 A5 BE1002179 A5 BE 1002179A5
Authority
BE
Belgium
Prior art keywords
pyranoquinoleins
pharmaceutical compositions
compositions containing
allergic
proctitis
Prior art date
Application number
BE8701471A
Other languages
English (en)
Original Assignee
Fisons Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB868630769A external-priority patent/GB8630769D0/en
Priority claimed from GB868630767A external-priority patent/GB8630767D0/en
Priority claimed from GB868630904A external-priority patent/GB8630904D0/en
Priority claimed from GB878706684A external-priority patent/GB8706684D0/en
Application filed by Fisons Plc filed Critical Fisons Plc
Application granted granted Critical
Publication of BE1002179A5 publication Critical patent/BE1002179A5/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/14Decongestants or antiallergics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/16Otologicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medical Preparation Storing Or Oral Administration Devices (AREA)

Abstract

Utilisation de l'acide 9-éthyl-6,9-dihydro-4,6-dioxo-10-propyl-4H-pyrano(3,2-g)quinoléine-2,8-carboxylique ou d'un sel pharmaceutiquement acceptable de celui-ci en solution aqueuse contre la conjonctivite, la kératite, "l'oeil allergique", les infections par adénovirus, le rejet de l'homogreffe de cornée, l'uvéïte antérieure, les polypes nasaux, la rhinite vasomotrice, les manifestations allergiques du nasopharynx, l'obstruction réversible des voies respiratoires, la maladie de Crohn, la colite distale ou la proctite.
BE8701471A 1986-12-23 1987-12-22 Compositions pharmaceutiques contenant des pyranoquinoleines. BE1002179A5 (fr)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB868630769A GB8630769D0 (en) 1986-12-23 1986-12-23 Pharmaceutical formulation
GB868630767A GB8630767D0 (en) 1986-12-23 1986-12-23 Pharmaceutical formulation
GB868630904A GB8630904D0 (en) 1986-12-24 1986-12-24 Pharmaceutical formulation
GB878706684A GB8706684D0 (en) 1987-03-20 1987-03-20 Pharmaceutical formulation

Publications (1)

Publication Number Publication Date
BE1002179A5 true BE1002179A5 (fr) 1990-10-02

Family

ID=27449862

Family Applications (2)

Application Number Title Priority Date Filing Date
BE8701471A BE1002179A5 (fr) 1986-12-23 1987-12-22 Compositions pharmaceutiques contenant des pyranoquinoleines.
BE9000682A BE1003466A3 (fr) 1986-12-23 1990-07-04 Compositions pharmaceutiques contenant des pyranoquinoleines.

Family Applications After (1)

Application Number Title Priority Date Filing Date
BE9000682A BE1003466A3 (fr) 1986-12-23 1990-07-04 Compositions pharmaceutiques contenant des pyranoquinoleines.

Country Status (22)

Country Link
US (1) US5443833A (fr)
EP (1) EP0279121B1 (fr)
JP (2) JP2568233B2 (fr)
KR (1) KR960001370B1 (fr)
AU (1) AU595969B2 (fr)
BE (2) BE1002179A5 (fr)
CA (1) CA1296635C (fr)
CH (1) CH674937A5 (fr)
DE (1) DE3787274T2 (fr)
DK (1) DK175032B1 (fr)
ES (1) ES2058129T3 (fr)
FI (1) FI875616A (fr)
FR (1) FR2609392B1 (fr)
GR (1) GR871999B (fr)
IE (3) IE63213B1 (fr)
IL (1) IL84893A (fr)
LU (1) LU87087A1 (fr)
MY (1) MY101535A (fr)
NO (1) NO875359L (fr)
NZ (1) NZ223026A (fr)
PT (1) PT86455B (fr)
SA (1) SA90110074B1 (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8704773D0 (en) * 1987-02-28 1987-04-01 Fisons Plc Compounds
GB2202145B (en) * 1987-03-17 1991-01-02 Fisons Plc Compositions of nedocromil for dermatological use.
GB8727590D0 (en) * 1987-11-25 1987-12-31 Fisons Plc Formulation
US5976573A (en) * 1996-07-03 1999-11-02 Rorer Pharmaceutical Products Inc. Aqueous-based pharmaceutical composition
US7977376B2 (en) 2001-06-27 2011-07-12 Novartis Ag Olopatadine formulations for topical nasal administration
CA2781923C (fr) * 2009-12-03 2018-08-14 Opko Health, Inc. Formulations de disaccharides hypersulfates

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2022078A (en) * 1977-05-04 1979-12-12 Fisons Ltd 4,6-Dioxo-4H,6H-pyrano[3,2- g]quinoline-2,8-dicarbocyclic Acids

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4474787A (en) * 1977-05-04 1984-10-02 Fisons Limited 7,6 Dioxo-4H,6H-pyrano[3,2-g]quinoline dicarboxylic acids and anti-allergic use thereof
IL54614A (en) * 1977-05-04 1983-07-31 Fisons Ltd Dihydrodioxo-pyranoquinoline dicarboxylic acid derivatives,their production and pharmaceutical compositions containing them
FR2440371A1 (fr) * 1978-10-31 1980-05-30 Fisons Ltd Nouveaux composes azotes heterocycliques, des compositions pharmaceutiques en contenant et des procedes pour les preparer
ATE11774T1 (de) * 1979-12-07 1985-02-15 Fisons Plc Verfahren zur herstellung von 1,4-dihydro-4-oxo- chinolin-2-carbonsaeuren oder salzen, estern oder amiden davon und zwischenverbindungen dafuer.
AU8468782A (en) * 1981-06-25 1983-01-06 Fisons Plc Compounds with sodium cromoglycate activity
GB8402047D0 (en) * 1984-01-26 1984-02-29 Fisons Plc Nitrogen heterocycles
EP0162556B1 (fr) * 1984-04-13 1991-11-06 FISONS plc Formes et formulations des sels de sodium de nédocromil
GB8630419D0 (en) * 1986-12-19 1987-01-28 Fisons Plc Pharmaceutical formulation
GB8704089D0 (en) * 1987-02-21 1987-03-25 Fisons Plc Method of treatment
GB8704773D0 (en) * 1987-02-28 1987-04-01 Fisons Plc Compounds
GB2202145B (en) * 1987-03-17 1991-01-02 Fisons Plc Compositions of nedocromil for dermatological use.

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2022078A (en) * 1977-05-04 1979-12-12 Fisons Ltd 4,6-Dioxo-4H,6H-pyrano[3,2- g]quinoline-2,8-dicarbocyclic Acids

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
BR. J. CLIN. PHARMAC., vol. 24, octobre 1987, pages 493-501; M.G. NEALE et al.: "The pharmacokinetics of nedocromil sodium, a new drug for the treatment of reversible obstructive airways disease, in human volunteers and patients with reversible obstructive airways disease" *
J. MED. CHEM., vol. 28, no. 12, 1985, pages 1832-1842, American Chemical Society; H. CAIRNS et al.: "New antiallergic pyrano[3,2-g]quinoline-2,8-dicarboxylic acids with potential for the topical treatment of asthma" *

Also Published As

Publication number Publication date
NO875359L (no) 1988-06-24
CA1296635C (fr) 1992-03-03
JP2568233B2 (ja) 1996-12-25
KR960001370B1 (ko) 1996-01-26
PT86455B (pt) 1990-11-20
DE3787274D1 (de) 1993-10-07
IE873507L (en) 1988-06-23
IL84893A0 (en) 1988-06-30
IE63213B1 (en) 1995-04-05
DK680787D0 (da) 1987-12-22
IE940371L (en) 1988-06-23
MY101535A (en) 1991-11-30
LU87087A1 (fr) 1989-07-07
DE3787274T2 (de) 1994-01-27
GR871999B (en) 1988-04-26
SA90110074B1 (ar) 2006-03-06
KR880007082A (ko) 1988-08-26
IE940372L (en) 1988-06-23
AU8292987A (en) 1988-06-23
NZ223026A (en) 1989-09-27
BE1003466A3 (fr) 1992-03-31
US5443833A (en) 1995-08-22
EP0279121B1 (fr) 1993-09-01
DK175032B1 (da) 2004-05-03
JP2504926B2 (ja) 1996-06-05
ES2058129T3 (es) 1994-11-01
JPS63233918A (ja) 1988-09-29
JPH07231926A (ja) 1995-09-05
EP0279121A2 (fr) 1988-08-24
FR2609392B1 (fr) 1994-04-08
NO875359D0 (no) 1987-12-21
FI875616A (fi) 1988-06-24
IL84893A (en) 1991-11-21
PT86455A (en) 1988-01-01
FR2609392A1 (fr) 1988-07-15
CH674937A5 (fr) 1990-08-15
FI875616A0 (fi) 1987-12-21
DK680787A (da) 1988-06-24
AU595969B2 (en) 1990-04-12
EP0279121A3 (en) 1990-09-12

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Legal Events

Date Code Title Description
RE20 Patent expired

Owner name: *FISONS PLC.

Effective date: 20071222