AU515428B2 - Process for preparing 3-(thiomethy) substituted cephalosporins - Google Patents

Process for preparing 3-(thiomethy) substituted cephalosporins

Info

Publication number
AU515428B2
AU515428B2 AU33828/78A AU3382878A AU515428B2 AU 515428 B2 AU515428 B2 AU 515428B2 AU 33828/78 A AU33828/78 A AU 33828/78A AU 3382878 A AU3382878 A AU 3382878A AU 515428 B2 AU515428 B2 AU 515428B2
Authority
AU
Australia
Prior art keywords
thiomethy
preparing
substituted cephalosporins
cephalosporins
substituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
AU33828/78A
Other languages
English (en)
Other versions
AU3382878A (en
Inventor
L. D Hatfield
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/862,871 external-priority patent/US4144391A/en
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Publication of AU3382878A publication Critical patent/AU3382878A/en
Application granted granted Critical
Publication of AU515428B2 publication Critical patent/AU515428B2/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/36—Methylene radicals, substituted by sulfur atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU33828/78A 1977-03-07 1978-03-03 Process for preparing 3-(thiomethy) substituted cephalosporins Expired AU515428B2 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US77501877A 1977-03-07 1977-03-07
USUS775018 1977-03-07
USUS862871 1977-12-27
US05/862,871 US4144391A (en) 1977-03-07 1977-12-27 Cephalosporin displacement reaction

Publications (2)

Publication Number Publication Date
AU3382878A AU3382878A (en) 1979-09-06
AU515428B2 true AU515428B2 (en) 1981-04-02

Family

ID=27118982

Family Applications (1)

Application Number Title Priority Date Filing Date
AU33828/78A Expired AU515428B2 (en) 1977-03-07 1978-03-03 Process for preparing 3-(thiomethy) substituted cephalosporins

Country Status (30)

Country Link
JP (1) JPS53130689A (fi)
AT (1) AT366696B (fi)
AU (1) AU515428B2 (fi)
BG (1) BG31379A3 (fi)
CA (1) CA1083141A (fi)
CH (1) CH637964A5 (fi)
CS (1) CS205115B2 (fi)
CY (1) CY1196A (fi)
DD (1) DD137356A5 (fi)
DE (1) DE2809058A1 (fi)
DK (1) DK97378A (fi)
EG (1) EG13454A (fi)
ES (1) ES467637A1 (fi)
FI (1) FI69309C (fi)
FR (1) FR2383189A1 (fi)
GB (1) GB1597036A (fi)
GR (1) GR68893B (fi)
HK (1) HK49083A (fi)
HU (1) HU179967B (fi)
IE (1) IE46437B1 (fi)
IL (1) IL54181A (fi)
IT (1) IT1093504B (fi)
MX (1) MX5142E (fi)
NL (1) NL190703C (fi)
NZ (1) NZ186610A (fi)
PH (1) PH14596A (fi)
PL (1) PL122152B1 (fi)
PT (1) PT67732A (fi)
SE (1) SE437991B (fi)
YU (1) YU51478A (fi)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5543043A (en) * 1978-09-22 1980-03-26 Sankyo Co Ltd Preparation of 3-substituted thiomethylcephalosporin derivative
US4576937A (en) * 1984-02-29 1986-03-18 Smithkline Beckman Corporation 7-D-Mandelamido-3(1-sulfomethyltetrazol-5-yl)thiomethyl-3-cephem-4-carboxylic acid monosodium salt
GB8519606D0 (en) * 1985-08-05 1985-09-11 Fujisawa Pharmaceutical Co 3 7-d substituted-3-cephem compounds
JP2503500B2 (ja) * 1986-04-14 1996-06-05 萬有製薬株式会社 新規セフアロスポリン誘導体及びその製造法
JPS62281881A (ja) * 1986-09-08 1987-12-07 Sankyo Co Ltd ３−置換チオメチルセフアロスポリン誘導体の製法
US20120329770A1 (en) * 2010-02-26 2012-12-27 Gary Igor Dmitrienko Cephalosporin derivatives useful as beta-lactamase inhibitors and compositions and methods of use thereof
GB201818410D0 (en) * 2018-11-12 2018-12-26 Imperial Innovations Ltd Compounds

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3641021A (en) * 1969-04-18 1972-02-08 Lilly Co Eli 3 7-(ring-substituted) cephalosporin compounds
JPS5116436B1 (fi) * 1971-05-31 1976-05-24
JPS5143785A (en) * 1974-10-11 1976-04-14 Yamanouchi Pharma Co Ltd Shinsefuarosuhorinkanrenkagobutsuno goseiho
JPS612674B2 (fi) * 1974-06-20 1986-01-27 Meiji Seika Co
CA1100129A (en) * 1974-08-02 1981-04-28 William H.W. Lunn Cephalosporin compounds
AU1303576A (en) * 1975-04-21 1977-10-20 Erba Carlo Spa Cephalosporins

Also Published As

Publication number Publication date
NL190703B (nl) 1994-02-01
FI780716A (fi) 1978-09-08
PL122152B1 (en) 1982-06-30
DK97378A (da) 1978-09-08
FR2383189B1 (fi) 1981-06-26
JPH025758B2 (fi) 1990-02-05
HU179967B (en) 1983-01-28
NZ186610A (en) 1979-11-01
CY1196A (en) 1983-12-31
BG31379A3 (en) 1981-12-15
CA1083141A (en) 1980-08-05
ATA150778A (de) 1981-09-15
AU3382878A (en) 1979-09-06
EG13454A (en) 1981-12-31
DE2809058C2 (fi) 1989-02-09
SE7802530L (sv) 1978-09-08
NL7802376A (nl) 1978-09-11
FI69309C (fi) 1986-01-10
IE46437B1 (en) 1983-06-15
IL54181A0 (en) 1978-06-15
GB1597036A (en) 1981-09-03
NL190703C (nl) 1994-07-01
SE437991B (sv) 1985-03-25
CS205115B2 (en) 1981-04-30
DD137356A5 (de) 1979-08-29
FR2383189A1 (fr) 1978-10-06
AT366696B (de) 1982-04-26
PT67732A (en) 1978-04-01
IT1093504B (it) 1985-07-19
PH14596A (en) 1981-10-02
DE2809058A1 (de) 1978-09-14
ES467637A1 (es) 1980-04-01
YU51478A (en) 1982-10-31
PL205135A1 (pl) 1979-06-04
CH637964A5 (en) 1983-08-31
HK49083A (en) 1983-11-04
FI69309B (fi) 1985-09-30
MX5142E (es) 1983-03-30
GR68893B (fi) 1982-03-15
IL54181A (en) 1981-03-31
IT7820912A0 (it) 1978-03-06
IE780453L (en) 1978-09-07
JPS53130689A (en) 1978-11-14

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