AU3573793A - 3-(1H-tetrazol-5-yl)-4H-pyrido(1,2-a)pyrimidine-4-ones pharmaceutical compositions containing the same and the preparation thereof - Google Patents

3-(1H-tetrazol-5-yl)-4H-pyrido(1,2-a)pyrimidine-4-ones pharmaceutical compositions containing the same and the preparation thereof

Info

Publication number
AU3573793A
AU3573793A AU35737/93A AU3573793A AU3573793A AU 3573793 A AU3573793 A AU 3573793A AU 35737/93 A AU35737/93 A AU 35737/93A AU 3573793 A AU3573793 A AU 3573793A AU 3573793 A AU3573793 A AU 3573793A
Authority
AU
Australia
Prior art keywords
tetrazol
pyrido
pyrimidine
preparation
same
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
AU35737/93A
Other languages
English (en)
Inventor
Maria Balogh
Kinga Boer
Istvan Hermecz
Agnes Horvath
Zoltan Kapui
Geza Kereszturi
Aniko Pajor
Judit Sipos
Lelle Vasvary
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Chinoin Private Co Ltd
Original Assignee
Chinoin Gyogyszer es Vegyeszeti Termekek Gyara Zrt
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chinoin Gyogyszer es Vegyeszeti Termekek Gyara Zrt filed Critical Chinoin Gyogyszer es Vegyeszeti Termekek Gyara Zrt
Publication of AU3573793A publication Critical patent/AU3573793A/en
Withdrawn legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU35737/93A 1992-02-13 1993-02-12 3-(1H-tetrazol-5-yl)-4H-pyrido(1,2-a)pyrimidine-4-ones pharmaceutical compositions containing the same and the preparation thereof Withdrawn AU3573793A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HU9200432A HUT64064A (en) 1992-02-13 1992-02-13 Process for producing puyrido/1,2-a/pyrimidine derivatives and pharmaceutical compositions comprising same as active ingredient
HU9200432 1992-02-13

Publications (1)

Publication Number Publication Date
AU3573793A true AU3573793A (en) 1993-09-03

Family

ID=10981335

Family Applications (1)

Application Number Title Priority Date Filing Date
AU35737/93A Withdrawn AU3573793A (en) 1992-02-13 1993-02-12 3-(1H-tetrazol-5-yl)-4H-pyrido(1,2-a)pyrimidine-4-ones pharmaceutical compositions containing the same and the preparation thereof

Country Status (7)

Country Link
CN (1) CN1080289A (zh)
AU (1) AU3573793A (zh)
HU (1) HUT64064A (zh)
IL (1) IL104706A0 (zh)
MX (1) MX9300779A (zh)
SI (1) SI9300075A (zh)
WO (1) WO1993016076A1 (zh)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU663886B2 (en) * 1990-09-25 1995-10-26 Chinoin Gyogyszer Es Vegyeszeti Termekek Gyara New 3-(substituted tetrazolyl)-4-oxo-4H-pyrido-{1,2-a}pyrimidines, salts thereof, pharmaceutical compositions containing them and process for preparing same

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ITMI20011764A1 (it) * 2001-08-10 2003-02-10 Dinamite Dipharma Spa Metodo per l'ottenimento del pemirolast ad elevata purezza
MXPA05003607A (es) * 2002-10-04 2005-11-17 Prana Biotechnology Ltd Compuestos neurologicamente activos.
EP1818058A3 (en) * 2006-02-13 2007-11-07 Astion Pharma A/S Treatment of mmp-mediated dermatological diseases with pemirolast
WO2007093184A2 (en) * 2006-02-13 2007-08-23 Astion Pharma A/S Treatment of mmp-mediated dermatological diseases with pemirolast
SI2448938T1 (sl) 2009-06-29 2014-08-29 Incyte Corporation Experimental Station Pirimidinoni kot zaviralci pi3k
WO2011075643A1 (en) 2009-12-18 2011-06-23 Incyte Corporation Substituted heteroaryl fused derivatives as pi3k inhibitors
US9193721B2 (en) 2010-04-14 2015-11-24 Incyte Holdings Corporation Fused derivatives as PI3Kδ inhibitors
WO2011163195A1 (en) 2010-06-21 2011-12-29 Incyte Corporation Fused pyrrole derivatives as pi3k inhibitors
JP5961187B2 (ja) 2010-12-20 2016-08-02 インサイト・ホールディングス・コーポレイションＩｎｃｙｔｅ Ｈｏｌｄｉｎｇｓ Ｃｏｒｐｏｒａｔｉｏｎ Ｐｉ３ｋ阻害剤としてのｎ−（１−（置換フェニル）エチル）−９ｈ−プリン−６−アミン
US9108984B2 (en) 2011-03-14 2015-08-18 Incyte Corporation Substituted diamino-pyrimidine and diamino-pyridine derivatives as PI3K inhibitors
WO2012135009A1 (en) 2011-03-25 2012-10-04 Incyte Corporation Pyrimidine-4,6-diamine derivatives as pi3k inhibitors
CA2846652C (en) 2011-09-02 2019-11-05 Incyte Corporation Heterocyclylamines as pi3k inhibitors
AR090548A1 (es) 2012-04-02 2014-11-19 Incyte Corp Azaheterociclobencilaminas biciclicas como inhibidores de pi3k
WO2015191677A1 (en) 2014-06-11 2015-12-17 Incyte Corporation Bicyclic heteroarylaminoalkyl phenyl derivatives as pi3k inhibitors
ES2843522T3 (es) 2015-02-27 2021-07-19 Incyte Corp Sales del inhibidor de PI3K y procesos para su preparación
WO2016183063A1 (en) 2015-05-11 2016-11-17 Incyte Corporation Crystalline forms of a pi3k inhibitor
WO2016183060A1 (en) 2015-05-11 2016-11-17 Incyte Corporation Process for the synthesis of a phosphoinositide 3-kinase inhibitor

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2044796C (en) * 1990-06-21 2001-10-16 Atsunori Sano Process for producing pyrido[1,2-a] pyrimidine derivative

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU663886B2 (en) * 1990-09-25 1995-10-26 Chinoin Gyogyszer Es Vegyeszeti Termekek Gyara New 3-(substituted tetrazolyl)-4-oxo-4H-pyrido-{1,2-a}pyrimidines, salts thereof, pharmaceutical compositions containing them and process for preparing same

Also Published As

Publication number Publication date
SI9300075A (en) 1993-09-30
CN1080289A (zh) 1994-01-05
WO1993016076A1 (en) 1993-08-19
HUT64064A (en) 1993-11-29
MX9300779A (es) 1993-09-30
IL104706A0 (en) 1993-06-10
HU9200432D0 (en) 1992-04-28

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