AU2020247255A1 - Androgen receptor modulators and methods for use as Proteolysis Targeting Chimera ligands - Google Patents

Androgen receptor modulators and methods for use as Proteolysis Targeting Chimera ligands Download PDF

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AU2020247255A1
AU2020247255A1 AU2020247255A AU2020247255A AU2020247255A1 AU 2020247255 A1 AU2020247255 A1 AU 2020247255A1 AU 2020247255 A AU2020247255 A AU 2020247255A AU 2020247255 A AU2020247255 A AU 2020247255A AU 2020247255 A1 AU2020247255 A1 AU 2020247255A1
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alkyl
optionally substituted
independently
bond
compound
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Raymond John Andersen
Han-Jie Zhou
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University of British Columbia
ESSA Pharma Inc
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University of British Columbia
ESSA Pharma Inc
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    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D491/04—Ortho-condensed systems
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