AU2019384802A1 - Pharmaceutical methods - Google Patents
Pharmaceutical methods Download PDFInfo
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- AU2019384802A1 AU2019384802A1 AU2019384802A AU2019384802A AU2019384802A1 AU 2019384802 A1 AU2019384802 A1 AU 2019384802A1 AU 2019384802 A AU2019384802 A AU 2019384802A AU 2019384802 A AU2019384802 A AU 2019384802A AU 2019384802 A1 AU2019384802 A1 AU 2019384802A1
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- Prior art keywords
- cancer
- administered
- tumor
- cell
- rivoceranib
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- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
- C07D213/82—Amides; Imides in position 3
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
- C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Physics & Mathematics (AREA)
- Biomedical Technology (AREA)
- Nanotechnology (AREA)
- Optics & Photonics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862770437P | 2018-11-21 | 2018-11-21 | |
| US62/770,437 | 2018-11-21 | ||
| PCT/US2019/062494 WO2020106898A1 (en) | 2018-11-21 | 2019-11-20 | Pharmaceutical methods |
Publications (1)
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| AU2019384802A1 true AU2019384802A1 (en) | 2021-06-17 |
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| AU2019384802A Abandoned AU2019384802A1 (en) | 2018-11-21 | 2019-11-20 | Pharmaceutical methods |
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| US (1) | US20230149377A1 (https=) |
| EP (1) | EP3883561A4 (https=) |
| JP (1) | JP2022507686A (https=) |
| KR (1) | KR20210099022A (https=) |
| AU (1) | AU2019384802A1 (https=) |
| CA (1) | CA3120366A1 (https=) |
| IL (1) | IL283273A (https=) |
| MX (1) | MX2021005936A (https=) |
| SG (1) | SG11202105221XA (https=) |
| TW (1) | TW202033189A (https=) |
| WO (1) | WO2020106898A1 (https=) |
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| WO2024137821A1 (en) * | 2022-12-21 | 2024-06-27 | Elevar Therapeutics, Inc. | Effect of rivoceranib on cytochrome p450 enzyme substrates |
| WO2025261988A1 (fr) * | 2024-06-17 | 2025-12-26 | Assistance Publique Hopitaux De Paris | Utilisation de nintédanib pour le traitement de la maladie de castleman |
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| US6245805B1 (en) * | 1995-10-26 | 2001-06-12 | Baker Norton Pharmaceuticals, Inc. | Method, compositions and kits for increasing the oral bioavailability of pharmaceutical agents |
| AU2013204181A1 (en) * | 2006-11-06 | 2013-05-16 | Abraxis Bioscience, Llc | Nanoparticles of paclitaxel and albumin in combination with bevacizumab against cancer |
| CN101675930B (zh) * | 2008-09-16 | 2012-04-25 | 江苏恒瑞医药股份有限公司 | 用于治疗增生性疾病的药物组合物 |
| EP3141245A1 (en) * | 2010-03-29 | 2017-03-15 | Abraxis BioScience, LLC | Methods of treating cancer |
| CN106038566B (zh) * | 2016-06-10 | 2018-11-27 | 江阴市人民医院 | 一种用于胃癌治疗的药物组合物及其应用 |
| CN107669685A (zh) * | 2016-08-02 | 2018-02-09 | 江苏恒瑞医药股份有限公司 | 阿帕替尼与替加氟和紫杉类药物联合用于制备治疗胃癌的药物中的用途 |
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2019
- 2019-11-20 CA CA3120366A patent/CA3120366A1/en active Pending
- 2019-11-20 JP JP2021527084A patent/JP2022507686A/ja active Pending
- 2019-11-20 WO PCT/US2019/062494 patent/WO2020106898A1/en not_active Ceased
- 2019-11-20 MX MX2021005936A patent/MX2021005936A/es unknown
- 2019-11-20 KR KR1020217018983A patent/KR20210099022A/ko not_active Abandoned
- 2019-11-20 SG SG11202105221XA patent/SG11202105221XA/en unknown
- 2019-11-20 TW TW108142221A patent/TW202033189A/zh unknown
- 2019-11-20 EP EP19887000.8A patent/EP3883561A4/en not_active Withdrawn
- 2019-11-20 US US17/295,848 patent/US20230149377A1/en not_active Abandoned
- 2019-11-20 AU AU2019384802A patent/AU2019384802A1/en not_active Abandoned
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2021
- 2021-05-19 IL IL283273A patent/IL283273A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| IL283273A (en) | 2021-07-29 |
| KR20210099022A (ko) | 2021-08-11 |
| CA3120366A1 (en) | 2020-05-28 |
| US20230149377A1 (en) | 2023-05-18 |
| WO2020106898A1 (en) | 2020-05-28 |
| EP3883561A1 (en) | 2021-09-29 |
| EP3883561A4 (en) | 2022-07-27 |
| MX2021005936A (es) | 2021-08-24 |
| JP2022507686A (ja) | 2022-01-18 |
| SG11202105221XA (en) | 2021-06-29 |
| TW202033189A (zh) | 2020-09-16 |
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