AU2019328599A1 - Compounds and methods for treating fungal infections - Google Patents

Compounds and methods for treating fungal infections Download PDF

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Publication number
AU2019328599A1
AU2019328599A1 AU2019328599A AU2019328599A AU2019328599A1 AU 2019328599 A1 AU2019328599 A1 AU 2019328599A1 AU 2019328599 A AU2019328599 A AU 2019328599A AU 2019328599 A AU2019328599 A AU 2019328599A AU 2019328599 A1 AU2019328599 A1 AU 2019328599A1
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Australia
Prior art keywords
pharmaceutical composition
pharmaceutically acceptable
compound
dosage form
solvate
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AU2019328599A
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English (en)
Inventor
Jason Brittain
Michael GREY
Michael Hodges
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Basilea Pharmaceutica International Ag Allschwil
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Basilea Pharmaceutica International Ag Allschwil
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Publication of AU2019328599A1 publication Critical patent/AU2019328599A1/en
Assigned to BASILEA PHARMACEUTICA INTERNATIONAL AG, ALLSCHWIL reassignment BASILEA PHARMACEUTICA INTERNATIONAL AG, ALLSCHWIL Request for Assignment Assignors: AMPLYX PHARMACEUTICALS, INC.
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    • A—HUMAN NECESSITIES
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/66—Phosphorus compounds
    • A61K31/675—Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4196—1,2,4-Triazoles
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
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    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
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    • A61K47/16—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
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    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Inorganic Chemistry (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Dermatology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Dispersion Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Biochemistry (AREA)
  • Immunology (AREA)
  • Physics & Mathematics (AREA)
  • Biomedical Technology (AREA)
  • Nanotechnology (AREA)
  • Optics & Photonics (AREA)
  • Otolaryngology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AU2019328599A 2018-08-31 2019-08-30 Compounds and methods for treating fungal infections Pending AU2019328599A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862725971P 2018-08-31 2018-08-31
US62/725,971 2018-08-31
PCT/US2019/049223 WO2020047510A1 (en) 2018-08-31 2019-08-30 Compounds and methods for treating fungal infections

Publications (1)

Publication Number Publication Date
AU2019328599A1 true AU2019328599A1 (en) 2021-04-22

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AU2019328599A Pending AU2019328599A1 (en) 2018-08-31 2019-08-30 Compounds and methods for treating fungal infections

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US (1) US20210290644A1 (zh)
EP (1) EP3843769A4 (zh)
JP (3) JP7522098B2 (zh)
KR (1) KR20210088528A (zh)
CN (1) CN112996527A (zh)
AR (1) AR121477A1 (zh)
AU (1) AU2019328599A1 (zh)
BR (1) BR112021003878A2 (zh)
CA (1) CA3110860A1 (zh)
EA (1) EA202190590A1 (zh)
IL (1) IL281140A (zh)
MX (1) MX2021002444A (zh)
TW (1) TW202024058A (zh)
WO (1) WO2020047510A1 (zh)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2023516648A (ja) * 2020-03-04 2023-04-20 アンプリックス ファーマシューティカルズ，インク． 真菌感染症の処置における化合物の使用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10133394A1 (de) * 2001-07-13 2003-01-30 Merck Patent Gmbh Flüssige Formulierung enthaltend Cetuximab
WO2005033079A1 (ja) * 2003-09-30 2005-04-14 Eisai Co., Ltd. ヘテロ環化合物を含有する新規な抗真菌剤
US8513287B2 (en) * 2007-12-27 2013-08-20 Eisai R&D Management Co., Ltd. Heterocyclic ring and phosphonoxymethyl group substituted pyridine derivatives and antifungal agent containing same
EP2636409A1 (en) * 2010-11-05 2013-09-11 Eisai R&D Management Co., Ltd. Combined pharmaceutical composition as antifungal agent

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Publication number Publication date
EP3843769A4 (en) 2022-11-16
EA202190590A1 (ru) 2021-07-16
EP3843769A1 (en) 2021-07-07
KR20210088528A (ko) 2021-07-14
AR121477A1 (es) 2022-06-08
TW202024058A (zh) 2020-07-01
JP2024116313A (ja) 2024-08-27
WO2020047510A1 (en) 2020-03-05
IL281140A (en) 2021-04-29
CN112996527A (zh) 2021-06-18
MX2021002444A (es) 2021-04-28
JP2024116312A (ja) 2024-08-27
CA3110860A1 (en) 2020-03-05
US20210290644A1 (en) 2021-09-23
JP7522098B2 (ja) 2024-07-24
BR112021003878A2 (pt) 2021-05-18
JP2021536446A (ja) 2021-12-27

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