AU2018375378A1 - Methods of inhibiting tumor metastasis - Google Patents
Methods of inhibiting tumor metastasis Download PDFInfo
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- AU2018375378A1 AU2018375378A1 AU2018375378A AU2018375378A AU2018375378A1 AU 2018375378 A1 AU2018375378 A1 AU 2018375378A1 AU 2018375378 A AU2018375378 A AU 2018375378A AU 2018375378 A AU2018375378 A AU 2018375378A AU 2018375378 A1 AU2018375378 A1 AU 2018375378A1
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- Prior art keywords
- cancer
- thromboxane
- receptor antagonist
- pharmaceutically acceptable
- acceptable salt
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- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
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Applications Claiming Priority (3)
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| US201762592365P | 2017-11-29 | 2017-11-29 | |
| US62/592,365 | 2017-11-29 | ||
| PCT/US2018/062967 WO2019108736A1 (en) | 2017-11-29 | 2018-11-29 | Methods of inhibiting tumor metastasis |
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| AU2018375378A1 true AU2018375378A1 (en) | 2020-05-28 |
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| AU2018375378A Abandoned AU2018375378A1 (en) | 2017-11-29 | 2018-11-29 | Methods of inhibiting tumor metastasis |
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| EP (1) | EP3716973A4 (https=) |
| JP (1) | JP7305197B2 (https=) |
| KR (1) | KR102687556B1 (https=) |
| CN (2) | CN111432817B (https=) |
| AU (1) | AU2018375378A1 (https=) |
| CA (1) | CA3082839A1 (https=) |
| TW (1) | TW201924719A (https=) |
| WO (1) | WO2019108736A1 (https=) |
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| KR20220164000A (ko) * | 2020-03-31 | 2022-12-12 | 어플라이드 메디칼 테크놀로지스 엘엘씨 | Pgd2/dp2 및 트롬복산 a2/tp 수용체의 이중 길항제 및 이상 면역 반응 또는 혈전성 체질의 치료를 위한 이의 용도 |
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| US5066480A (en) | 1988-04-11 | 1991-11-19 | E. R. Squibb & Sons, Inc. | Method of preventing or reducing adverse reactions to protamine using a thromboxane a2 receptor antagonist |
| US4839384A (en) | 1988-10-07 | 1989-06-13 | E. R. Squibb & Sons, Inc. | Method of inhibiting onset of or treating migraine headache using a thromboxane A2 receptor antagonist |
| US5153327A (en) | 1988-12-23 | 1992-10-06 | E. R. Squibb & Sons, Inc. | 7-Oxabicycloheptyl substituted heterocyclic amide or ester prostaglandin analogs useful in the treatment of thrombotic and vasospastic disease |
| US5100889A (en) | 1989-04-03 | 1992-03-31 | E. R. Squibb & Sons, Inc. | 7-oxabicycloheptyl substituted heterocyclic amide or ester prostaglandin analogs useful in the treatment of thrombotic and vasospastic disease |
| ZA911453B (en) | 1990-03-19 | 1991-11-27 | Squibb & Sons Inc | Method of protecting against and/or treating ulcerative gastrointestinal conditions using a thromoboxane,a2 receptor antagonist and combination useful in preventing and/or treating ulcers and/or inflammation |
| US5158967A (en) * | 1991-06-12 | 1992-10-27 | E. R. Squibb & Sons, Inc. | 7-oxabicycloheptyl substituted heterocyclic amide prostaglandin analogs useful in the treatment of thrombotic and vasospastic disease |
| US5281716A (en) * | 1992-06-18 | 1994-01-25 | Bristol-Myers Squibb Company | Method for preparing 7-oxabicycloheptyl substituted oxazole amide prostaglandin analog intermediates useful in the preparation of anti-thrombotic and anti-vasospastic compounds |
| US5260449A (en) | 1992-08-12 | 1993-11-09 | E. R. Squibb & Sons, Inc. | Method for preparing 7-oxabicycloheptyl substituted bromooxazole amide prostaglandin analog intermediates useful in the preparation of anti-thrombotic and anti-vasospastic compounds |
| US5399725A (en) | 1993-05-27 | 1995-03-21 | Bristol-Myers Squibb Co. | 7-oxabicycloheptane carboxylic acid prostaglandin analog intermediates useful in the preparation of anti-thrombotic and anti-vasospastic compounds and method for preparing same |
| US5332840A (en) | 1993-05-27 | 1994-07-26 | Bristol-Myers Squibb Company | Method for preparing a benzaldehyde intermediate |
| US5605917A (en) | 1994-12-22 | 1997-02-25 | Bristol-Myers Squibb Company | Method of treating dysmenorrhea employing an interphenylene 7-oxabicycloheptyl substituted heterocyclic amide prostaglandin analog |
| IL137937A0 (en) | 1999-08-27 | 2001-10-31 | Pfizer Prod Inc | A pharmaceutical composition for the prevention and treatment of nicotine addiction in a mammal |
| AU2001264729A1 (en) * | 2000-05-22 | 2001-12-03 | Nitromed, Inc. | Thromboxane inhibitors, compositions and methods of use related applications |
| KR100681763B1 (ko) | 2005-02-28 | 2007-02-15 | 재단법인 목암생명공학연구소 | 인간 리포칼린 2를 유효성분으로 포함하는 암 전이 억제용약학적 조성물, 이를 이용한 암 전이 억제 방법 |
| EP1986675A2 (en) | 2006-02-24 | 2008-11-05 | The Government of the United States of America as represented by the Secretary of the Department of Health and Human Services | Extracellular matrix/metastasis modifer genes for the prevention or inhibition of metastasis or growth of tumor and for characterization of tumor |
| US20080160024A1 (en) | 2006-12-07 | 2008-07-03 | Board Of Trustees Of The University Of Arkansas | Inhibition of cancer metastasis |
| WO2009089098A1 (en) | 2008-01-03 | 2009-07-16 | Musc Foundation For Research Development | Methods for the treatment of cancers |
| US9283266B2 (en) | 2008-02-28 | 2016-03-15 | University Of Notre Dame | Metastasis inhibition preparations and methods |
| US8912167B2 (en) | 2011-05-19 | 2014-12-16 | Eugene J. Oliva | Heparin-based compositions and methods for the inhibition of metastasis |
| US20170226514A1 (en) | 2014-08-13 | 2017-08-10 | MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. | Prevention of tumour metastasis by inhibition of necroptosis |
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2018
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- 2018-11-29 WO PCT/US2018/062967 patent/WO2019108736A1/en not_active Ceased
- 2018-11-29 EP EP18884156.3A patent/EP3716973A4/en active Pending
- 2018-11-29 TW TW107142806A patent/TW201924719A/zh unknown
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- 2018-11-29 JP JP2020529160A patent/JP7305197B2/ja active Active
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2024
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Also Published As
| Publication number | Publication date |
|---|---|
| CN117122687A (zh) | 2023-11-28 |
| JP2021504385A (ja) | 2021-02-15 |
| EP3716973A1 (en) | 2020-10-07 |
| US20250144079A1 (en) | 2025-05-08 |
| CN111432817A (zh) | 2020-07-17 |
| KR20200093575A (ko) | 2020-08-05 |
| KR102687556B1 (ko) | 2024-07-22 |
| US20240041839A1 (en) | 2024-02-08 |
| US11471444B2 (en) | 2022-10-18 |
| US20230090578A1 (en) | 2023-03-23 |
| WO2019108736A1 (en) | 2019-06-06 |
| US20200405694A1 (en) | 2020-12-31 |
| JP7305197B2 (ja) | 2023-07-10 |
| CA3082839A1 (en) | 2019-06-06 |
| CN111432817B (zh) | 2023-10-31 |
| EP3716973A4 (en) | 2021-11-10 |
| TW201924719A (zh) | 2019-07-01 |
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| MK1 | Application lapsed section 142(2)(a) - no request for examination in relevant period |