AU2007274710A1 - Tartrate salt of (7S)-7-[(5-fluoro-2-methyl-benzyl)oxy]-2-[(2R)-2-methylpiperazin-1-yl]-6,7-dihydro-5H-cyclopenta[b]pyridine - Google Patents

Tartrate salt of (7S)-7-[(5-fluoro-2-methyl-benzyl)oxy]-2-[(2R)-2-methylpiperazin-1-yl]-6,7-dihydro-5H-cyclopenta[b]pyridine Download PDF

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AU2007274710A1
AU2007274710A1 AU2007274710A AU2007274710A AU2007274710A1 AU 2007274710 A1 AU2007274710 A1 AU 2007274710A1 AU 2007274710 A AU2007274710 A AU 2007274710A AU 2007274710 A AU2007274710 A AU 2007274710A AU 2007274710 A1 AU2007274710 A1 AU 2007274710A1
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disorder
disease
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dementia
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Kevin Kun-Chin Liu
Yuan Zeng
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Pfizer Products Inc
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Pfizer Products Inc
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D221/00Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/04Ortho- or peri-condensed ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
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    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/10Drugs for disorders of the urinary system of the bladder
    • AHUMAN NECESSITIES
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10Drugs for genital or sexual disorders; Contraceptives for impotence
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P25/00Drugs for disorders of the nervous system
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    • A61P25/06Antimigraine agents
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    • A61P25/00Drugs for disorders of the nervous system
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    • A61P25/16Anti-Parkinson drugs
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    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
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    • C07B2200/13Crystalline forms, e.g. polymorphs

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  • Health & Medical Sciences (AREA)
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  • General Health & Medical Sciences (AREA)
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  • Urology & Nephrology (AREA)
  • Anesthesiology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
AU2007274710A 2006-07-14 2007-07-09 Tartrate salt of (7S)-7-[(5-fluoro-2-methyl-benzyl)oxy]-2-[(2R)-2-methylpiperazin-1-yl]-6,7-dihydro-5H-cyclopenta[b]pyridine Abandoned AU2007274710A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US83089006P 2006-07-14 2006-07-14
US60/830,890 2006-07-14
PCT/IB2007/002025 WO2008010073A1 (en) 2006-07-14 2007-07-09 Tartrate salt of (7s)-7-[(5-fluoro-2-methyl-benzyl)oxy]-2-[(2r)-2-methylpiperazin-1-yl]-6,7-dihydro-5h-cyclopenta[b]pyridine

Publications (1)

Publication Number Publication Date
AU2007274710A1 true AU2007274710A1 (en) 2008-01-24

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AU2007274710A Abandoned AU2007274710A1 (en) 2006-07-14 2007-07-09 Tartrate salt of (7S)-7-[(5-fluoro-2-methyl-benzyl)oxy]-2-[(2R)-2-methylpiperazin-1-yl]-6,7-dihydro-5H-cyclopenta[b]pyridine

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Country Link
US (1) US20100004259A1 (enExample)
EP (1) EP2044029B1 (enExample)
JP (1) JP4312243B2 (enExample)
KR (1) KR20090029299A (enExample)
CN (1) CN101506172A (enExample)
AR (1) AR062068A1 (enExample)
AT (1) ATE496894T1 (enExample)
AU (1) AU2007274710A1 (enExample)
CA (1) CA2657640A1 (enExample)
DE (1) DE602007012254D1 (enExample)
IL (1) IL196417A0 (enExample)
MX (1) MX2009000508A (enExample)
NO (1) NO20090667L (enExample)
TW (1) TW200821293A (enExample)
WO (1) WO2008010073A1 (enExample)
ZA (1) ZA200901051B (enExample)

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MX2009000508A (es) 2009-01-27
ATE496894T1 (de) 2011-02-15
DE602007012254D1 (de) 2011-03-10
JP2008044931A (ja) 2008-02-28
EP2044029A1 (en) 2009-04-08
ZA200901051B (en) 2010-01-27
WO2008010073A8 (en) 2009-03-05
IL196417A0 (en) 2009-09-22
JP4312243B2 (ja) 2009-08-12
TW200821293A (en) 2008-05-16
WO2008010073A1 (en) 2008-01-24
KR20090029299A (ko) 2009-03-20
CA2657640A1 (en) 2008-01-24
CN101506172A (zh) 2009-08-12
EP2044029B1 (en) 2011-01-26
AR062068A1 (es) 2008-10-15
NO20090667L (no) 2009-02-11
US20100004259A1 (en) 2010-01-07

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