AU2006304283B2 - Biphenyl derivatives as modulators of voltage gated ion channels - Google Patents
Biphenyl derivatives as modulators of voltage gated ion channels Download PDFInfo
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- AU2006304283B2 AU2006304283B2 AU2006304283A AU2006304283A AU2006304283B2 AU 2006304283 B2 AU2006304283 B2 AU 2006304283B2 AU 2006304283 A AU2006304283 A AU 2006304283A AU 2006304283 A AU2006304283 A AU 2006304283A AU 2006304283 B2 AU2006304283 B2 AU 2006304283B2
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Classifications
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- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
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Landscapes
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| US72568605P | 2005-10-12 | 2005-10-12 | |
| US60/725,686 | 2005-10-12 | ||
| PCT/US2006/040156 WO2007047474A2 (en) | 2005-10-12 | 2006-10-12 | Biphenyl derivatives as modulators of voltage gated ion channels |
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| AU2006304283A1 AU2006304283A1 (en) | 2007-04-26 |
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| KR20080021030A (ko) * | 2005-05-16 | 2008-03-06 | 버텍스 파마슈티칼스 인코포레이티드 | 이온 채널 조절인자로서의 바이사이클릭 유도체 |
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| WO2009133641A1 (ja) * | 2008-04-30 | 2009-11-05 | シャープ株式会社 | 照明装置、及び表示装置 |
| WO2010002956A2 (en) * | 2008-07-01 | 2010-01-07 | Vertex Pharmaceuticals Incorporated | Heterocyclic derivatives as modulators of ion channels |
| GB201209015D0 (en) * | 2012-05-22 | 2012-07-04 | Convergence Pharmaceuticals | Novel compounds |
| US9714252B2 (en) | 2012-12-20 | 2017-07-25 | Purdue Pharma L.P. | Cyclic sulfonamides as sodium channel blockers |
| CN105026373B (zh) | 2013-01-31 | 2018-03-30 | 沃泰克斯药物股份有限公司 | 作为钠通道调节剂的吡啶酮酰胺 |
| US20200270237A1 (en) * | 2017-10-19 | 2020-08-27 | Esteve Pharmaceuticals, S.A. | New alkoxyamino compounds for treating pain and pain related conditions |
| CA3105748A1 (en) | 2018-07-09 | 2020-01-16 | Lieber Institute, Inc. | Pyridazine compounds for inhibiting nav1.8 |
| KR20210019581A (ko) | 2018-07-09 | 2021-02-22 | 리버 인스티튜트, 아이엔씨 | Nav1.8을 억제하기 위한 피리딘 카르복스아미드 화합물 |
| WO2020163236A1 (en) * | 2019-02-04 | 2020-08-13 | The General Hospital Corporation | Treating long qt syndrome |
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| SE0001899D0 (sv) * | 2000-05-22 | 2000-05-22 | Pharmacia & Upjohn Ab | New compounds |
| WO2002039987A2 (en) * | 2000-11-14 | 2002-05-23 | Neurosearch A/S | Use of malaria parasite anion channel blockers for treating malaria |
| MXPA04004837A (es) * | 2001-11-22 | 2004-08-02 | Biovitrum Ab | Inhibidores de 11-??-hidroxiesteroide deshidrogenasa de tipo 1. |
| EP1461327A1 (en) * | 2001-11-22 | 2004-09-29 | Biovitrum Ab | Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 |
| US7135575B2 (en) * | 2003-03-03 | 2006-11-14 | Array Biopharma, Inc. | P38 inhibitors and methods of use thereof |
| AR045238A1 (es) * | 2003-08-08 | 2005-10-19 | Vertex Pharma | Compuestos utiles como inhibidores de canales ionicos regulados por voltaje |
| KR20060101772A (ko) * | 2003-12-19 | 2006-09-26 | 화이자 인코포레이티드 | 당뇨병 및 비만을 치료하기 위한,11-베타-하이드록시스테로이드 데하이드로게나제 유형1(11-베타-ｈｓｄ-1)의 저해제로서의벤젠설폰일아미노-피리딘-2-일 유도체 및 관련 화합물 |
| WO2006089871A2 (en) | 2005-02-23 | 2006-08-31 | Neurosearch A/S | Diphenylurea derivatives useful as erg channel openers for the treatment of cardiac arrhythmias |
| US7683083B2 (en) * | 2005-10-12 | 2010-03-23 | Vertex Pharmaceuticals Incorporated | Biphenyl derivatives as modulators of voltage gated ion channels |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5514696A (en) * | 1992-05-06 | 1996-05-07 | Bristol-Myers Squibb Co. | Phenyl sulfonamide endothelin antagonists |
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| CA2624831A1 (en) | 2007-04-26 |
| NZ567570A (en) | 2011-02-25 |
| AU2006304283A1 (en) | 2007-04-26 |
| US20100130548A1 (en) | 2010-05-27 |
| CN101365690A (zh) | 2009-02-11 |
| US8236833B2 (en) | 2012-08-07 |
| EP1934191B1 (en) | 2012-03-28 |
| ATE551333T1 (de) | 2012-04-15 |
| NO20082165L (no) | 2008-07-09 |
| US7683083B2 (en) | 2010-03-23 |
| KR20080059292A (ko) | 2008-06-26 |
| JP2009511599A (ja) | 2009-03-19 |
| US20080113990A1 (en) | 2008-05-15 |
| WO2007047474A3 (en) | 2007-07-05 |
| IL190632A0 (en) | 2008-11-03 |
| ZA200803704B (en) | 2009-09-30 |
| ES2383090T3 (es) | 2012-06-18 |
| WO2007047474A2 (en) | 2007-04-26 |
| EP1934191A2 (en) | 2008-06-25 |
| RU2008118350A (ru) | 2009-11-20 |
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