AU2006287528A1 - 1 , 4 and 1 , 5-disubstituted indole derivatives for use as PPAR active compounds - Google Patents

1 , 4 and 1 , 5-disubstituted indole derivatives for use as PPAR active compounds Download PDF

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Publication number
AU2006287528A1
AU2006287528A1 AU2006287528A AU2006287528A AU2006287528A1 AU 2006287528 A1 AU2006287528 A1 AU 2006287528A1 AU 2006287528 A AU2006287528 A AU 2006287528A AU 2006287528 A AU2006287528 A AU 2006287528A AU 2006287528 A1 AU2006287528 A1 AU 2006287528A1
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optionally substituted
substituted lower
group
bound
fluoro
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AU2006287528A
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Inventor
Dean R. Artis
Prabha N. Ibrahim
Byunghun Lee
Jack Lin
Shenghua Shi
Chao Zhang
Rebecca Zuckerman
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Plexxikon Inc
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Plexxikon Inc
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    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
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    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
    • C—CHEMISTRY; METALLURGY
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    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings

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  • Dermatology (AREA)
  • Cardiology (AREA)
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  • Heart & Thoracic Surgery (AREA)
  • Obesity (AREA)
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  • Ophthalmology & Optometry (AREA)
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  • Child & Adolescent Psychology (AREA)
AU2006287528A 2005-09-07 2006-09-06 1 , 4 and 1 , 5-disubstituted indole derivatives for use as PPAR active compounds Abandoned AU2006287528A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US71525905P 2005-09-07 2005-09-07
US60/715,259 2005-09-07
PCT/US2006/034780 WO2007030574A2 (en) 2005-09-07 2006-09-06 1 , 4 and 1 , 5-disubstituted indole derivatives for use as ppar active compounds

Publications (1)

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AU2006287528A1 true AU2006287528A1 (en) 2007-03-15

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AU2006287528A Abandoned AU2006287528A1 (en) 2005-09-07 2006-09-06 1 , 4 and 1 , 5-disubstituted indole derivatives for use as PPAR active compounds

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Country Link
US (1) US20080234349A1 (https=)
EP (1) EP1931658A2 (https=)
JP (1) JP2009509932A (https=)
AU (1) AU2006287528A1 (https=)
CA (1) CA2621275A1 (https=)
WO (1) WO2007030574A2 (https=)

Cited By (2)

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AU2007221020B2 (en) * 2006-02-28 2013-02-14 Dart Neuroscience (Cayman) Ltd. Therapeutic compounds
AU2013200480B2 (en) * 2006-02-28 2016-06-09 Dart Neuroscience (Cayman) Ltd. Therapeutic compounds

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CA2774476A1 (en) * 2009-10-07 2011-04-14 Francis Barany Coferons and methods of making and using them
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TW201815766A (zh) 2016-09-22 2018-05-01 美商普雷辛肯公司 用於ｉｄｏ及ｔｄｏ調節之化合物及方法以及其適應症
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AU2018307910B2 (en) 2017-07-25 2024-07-25 Daiichi Sankyo Company, Limited Formulations of a compound modulating kinases
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EP3768666A1 (en) 2018-03-20 2021-01-27 Plexxikon Inc. Compounds and methods for ido and tdo modulation, and indications therefor
MX2022007265A (es) 2019-12-20 2022-09-09 Nuevolution As Compuestos activos frente a receptores nucleares.
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US20080234349A1 (en) 2008-09-25
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