AU2006247581B2 - Method for preparing substituted pyrimidines - Google Patents

Method for preparing substituted pyrimidines Download PDF

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Publication number
AU2006247581B2
AU2006247581B2 AU2006247581A AU2006247581A AU2006247581B2 AU 2006247581 B2 AU2006247581 B2 AU 2006247581B2 AU 2006247581 A AU2006247581 A AU 2006247581A AU 2006247581 A AU2006247581 A AU 2006247581A AU 2006247581 B2 AU2006247581 B2 AU 2006247581B2
Authority
AU
Australia
Prior art keywords
compound
formula
preparing
solvent
persulfate
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU2006247581A
Other languages
English (en)
Other versions
AU2006247581A1 (en
Inventor
Gary David Annis
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
EIDP Inc
Original Assignee
EI Du Pont de Nemours and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by EI Du Pont de Nemours and Co filed Critical EI Du Pont de Nemours and Co
Publication of AU2006247581A1 publication Critical patent/AU2006247581A1/en
Application granted granted Critical
Publication of AU2006247581B2 publication Critical patent/AU2006247581B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/42—One nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/30—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/34—One oxygen atom
    • C07D239/36—One oxygen atom as doubly bound oxygen atom or as unsubstituted hydroxy radical

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
AU2006247581A 2005-05-16 2006-05-12 Method for preparing substituted pyrimidines Ceased AU2006247581B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US68129805P 2005-05-16 2005-05-16
US60/681,298 2005-05-16
PCT/US2006/018522 WO2006124657A1 (en) 2005-05-16 2006-05-12 Method for preparing substituted pyrimidines

Publications (2)

Publication Number Publication Date
AU2006247581A1 AU2006247581A1 (en) 2006-11-23
AU2006247581B2 true AU2006247581B2 (en) 2011-10-20

Family

ID=36867439

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2006247581A Ceased AU2006247581B2 (en) 2005-05-16 2006-05-12 Method for preparing substituted pyrimidines

Country Status (13)

Country Link
US (1) US8013155B2 (https=)
EP (1) EP1888536B1 (https=)
JP (1) JP5069677B2 (https=)
KR (1) KR101348458B1 (https=)
CN (1) CN101175730B (https=)
AT (1) ATE465999T1 (https=)
AU (1) AU2006247581B2 (https=)
BR (1) BRPI0612414A2 (https=)
DE (1) DE602006013970D1 (https=)
IL (1) IL185884A (https=)
PL (1) PL1888536T3 (https=)
WO (1) WO2006124657A1 (https=)
ZA (1) ZA200707974B (https=)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GEP20105099B (en) * 2005-05-06 2010-10-25 Du Pont Method for preparation of optionally 2-substituted 1,6- dihydrocarboxil acids
KR20090024120A (ko) * 2006-04-10 2009-03-06 이 아이 듀폰 디 네모아 앤드 캄파니 제초성 혼합물
WO2013124246A1 (de) 2012-02-22 2013-08-29 Bayer Intellectual Property Gmbh Herbizid wirksame 4-dialkoxymethyl-2-phenylpyrimidine
CN102977050B (zh) * 2012-11-20 2015-04-22 浙江工业大学 一种2-苯并噻唑二甲缩醛和2-苯并噻唑甲醛的合成方法
CN116063179A (zh) * 2023-02-20 2023-05-05 南京杰运医药科技有限公司 一种4-甲氧基乙酰乙酸甲酯的合成方法

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2004309325A1 (en) * 2003-12-19 2005-07-14 Corteva Agriscience Llc Herbicidal pyrimidines

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA207185A (en) 1921-01-04 C. Wagner Virgil Warming plate
GB2095240A (en) * 1981-03-05 1982-09-29 Fujisawa Pharmaceutical Co Dihydropyrimidine derivatives, processes for preparation thereof and pharmaceutical composition comprising the same
JPS57158779A (en) * 1981-03-05 1982-09-30 Fujisawa Pharmaceut Co Ltd Dihydropyrimidine derivative and its salt, their preparation and antiallergic containing the same
DE3935277A1 (de) 1989-10-24 1991-05-02 Hoechst Ag Sulfonierte heterocyclische carboxamide, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung als herbizide oder wachstumsregulatoren
CN1071049A (zh) * 1991-10-09 1993-04-21 纳幕尔杜邦公司 用于稻中杂草防治的除草剂
BR9908004A (pt) 1998-02-17 2001-12-18 Tularik Inc Composto, composição e método para prevençãoou supressão de uma infecção viral
ES2240093T3 (es) 1999-04-15 2005-10-16 Basf Aktiengesellschaft Procedimiento para la preparacion de pirimidinas substituidas.
AU2002258400A1 (en) 2001-02-16 2002-08-28 Tularik Inc. Methods of using pyrimidine-based antiviral agents
DE602004022819D1 (de) 2003-06-06 2009-10-08 Vertex Pharma Von atp-bindende kassette transportern
GEP20105099B (en) * 2005-05-06 2010-10-25 Du Pont Method for preparation of optionally 2-substituted 1,6- dihydrocarboxil acids

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2004309325A1 (en) * 2003-12-19 2005-07-14 Corteva Agriscience Llc Herbicidal pyrimidines

Also Published As

Publication number Publication date
IL185884A0 (en) 2008-01-06
DE602006013970D1 (de) 2010-06-10
CN101175730B (zh) 2011-05-25
EP1888536A1 (en) 2008-02-20
IL185884A (en) 2012-03-29
JP5069677B2 (ja) 2012-11-07
ATE465999T1 (de) 2010-05-15
BRPI0612414A2 (pt) 2010-11-09
US20090054647A1 (en) 2009-02-26
AU2006247581A1 (en) 2006-11-23
EP1888536B1 (en) 2010-04-28
CN101175730A (zh) 2008-05-07
US8013155B2 (en) 2011-09-06
JP2008540655A (ja) 2008-11-20
KR101348458B1 (ko) 2014-01-07
KR20080016640A (ko) 2008-02-21
WO2006124657A1 (en) 2006-11-23
ZA200707974B (en) 2008-11-26
PL1888536T3 (pl) 2010-09-30

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Legal Events

Date Code Title Description
FGA Letters patent sealed or granted (standard patent)
MK14 Patent ceased section 143(a) (annual fees not paid) or expired