AU2006235706B2 - New tricyclic angiotensin II agonists - Google Patents

New tricyclic angiotensin II agonists Download PDF

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Publication number
AU2006235706B2
AU2006235706B2 AU2006235706A AU2006235706A AU2006235706B2 AU 2006235706 B2 AU2006235706 B2 AU 2006235706B2 AU 2006235706 A AU2006235706 A AU 2006235706A AU 2006235706 A AU2006235706 A AU 2006235706A AU 2006235706 B2 AU2006235706 B2 AU 2006235706B2
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Australia
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compound
formula
alkyl
compounds
alkoxy
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AU2006235706A
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AU2006235706A1 (en
Inventor
Mathias Alterman
Anders Hallberg
Xiongyu Wu
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Vicore Pharma AB
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Vicore Pharma AB
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    • C07—ORGANIC CHEMISTRY
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    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
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    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/24—Oxygen or sulfur atoms
    • C07D207/26—2-Pyrrolidones
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    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4025—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
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  • Health & Medical Sciences (AREA)
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  • Engineering & Computer Science (AREA)
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  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Hospice & Palliative Care (AREA)
  • Obesity (AREA)
  • Gynecology & Obstetrics (AREA)
  • Vascular Medicine (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Dermatology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Psychiatry (AREA)
  • Transplantation (AREA)
AU2006235706A 2005-04-12 2006-04-12 New tricyclic angiotensin II agonists Ceased AU2006235706B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US67025705P 2005-04-12 2005-04-12
US60/670,257 2005-04-12
PCT/GB2006/001332 WO2006109056A1 (en) 2005-04-12 2006-04-12 New tricyclic angiotensin ii agonists

Publications (2)

Publication Number Publication Date
AU2006235706A1 AU2006235706A1 (en) 2006-10-19
AU2006235706B2 true AU2006235706B2 (en) 2012-03-08

Family

ID=36616971

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2006235706A Ceased AU2006235706B2 (en) 2005-04-12 2006-04-12 New tricyclic angiotensin II agonists

Country Status (12)

Country Link
US (1) US8067418B2 (enExample)
EP (1) EP1869024B1 (enExample)
JP (2) JP5289043B2 (enExample)
KR (1) KR101284573B1 (enExample)
CN (2) CN104109156A (enExample)
AT (1) ATE487713T1 (enExample)
AU (1) AU2006235706B2 (enExample)
CA (1) CA2604038C (enExample)
DE (1) DE602006018122D1 (enExample)
ES (1) ES2384450T3 (enExample)
MX (1) MX2007012635A (enExample)
WO (1) WO2006109056A1 (enExample)

Families Citing this family (31)

* Cited by examiner, † Cited by third party
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JP5679997B2 (ja) 2009-02-04 2015-03-04 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 11β−ヒドロキシステロイドデヒドロゲナーゼ1の環状阻害剤
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