AU2001262081A1 - Method for producing beta-alaninamides - Google Patents

Method for producing beta-alaninamides

Info

Publication number
AU2001262081A1
AU2001262081A1 AU2001262081A AU6208101A AU2001262081A1 AU 2001262081 A1 AU2001262081 A1 AU 2001262081A1 AU 2001262081 A AU2001262081 A AU 2001262081A AU 6208101 A AU6208101 A AU 6208101A AU 2001262081 A1 AU2001262081 A1 AU 2001262081A1
Authority
AU
Australia
Prior art keywords
alaninamides
producing beta
sup
formula
salts
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2001262081A
Other languages
English (en)
Inventor
Stefan Hildbrand
Thomas Ruppen
Dario Veghini
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Lonza AG
Original Assignee
Lonza AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lonza AG filed Critical Lonza AG
Publication of AU2001262081A1 publication Critical patent/AU2001262081A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00Preparation of carboxylic acid amides
    • C07C231/14Preparation of carboxylic acid amides by formation of carboxamide groups together with reactions not involving the carboxamide groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00Carboxylic acid nitriles
    • C07C255/01Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms
    • C07C255/19Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms containing cyano groups and carboxyl groups, other than cyano groups, bound to the same saturated acyclic carbon skeleton
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Peptides Or Proteins (AREA)
  • Pyrrole Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AU2001262081A 2000-03-03 2001-03-02 Method for producing beta-alaninamides Abandoned AU2001262081A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP00104643 2000-03-03
EP00104643 2000-03-03
PCT/EP2001/002349 WO2001064638A1 (de) 2000-03-03 2001-03-02 VERFAHREN ZUR HERSTELLUNG VON β-ALANINAMIDEN

Publications (1)

Publication Number Publication Date
AU2001262081A1 true AU2001262081A1 (en) 2001-09-12

Family

ID=8168028

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2001262081A Abandoned AU2001262081A1 (en) 2000-03-03 2001-03-02 Method for producing beta-alaninamides

Country Status (6)

Country Link
US (2) US6878829B2 (de)
EP (1) EP1259483B1 (de)
JP (1) JP2004509834A (de)
AT (1) ATE392413T1 (de)
AU (1) AU2001262081A1 (de)
WO (1) WO2001064638A1 (de)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE493379T1 (de) 2001-09-06 2011-01-15 Lonza Ag Verfahren zur herstellung von beta-alaninamiden
CN107602661B (zh) * 2017-08-24 2020-03-17 烟台万润药业有限公司 一种聚普瑞锌的制备方法
CN111051289A (zh) 2017-09-05 2020-04-21 株式会社德山 被保护的l-肌肽衍生物、l-肌肽以及结晶性l-肌肽锌络合物的制造方法
CN114213335B (zh) * 2021-12-23 2023-08-15 浙江湃肽生物股份有限公司 肌肽中间体及其肌肽的制备、用途
CN114573470B (zh) * 2022-03-17 2023-12-15 浙江海洲制药有限公司 一种合成n-三氟乙酰叔亮氨酸的方法
CN116283604A (zh) * 2022-12-25 2023-06-23 苏州永健生物医药有限公司 一种亚精胺的制备方法
CN117164519A (zh) * 2023-08-18 2023-12-05 杭州小蓓医药科技有限公司 一种l-肌肽的合成方法

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4093738A (en) * 1974-04-09 1978-06-06 Ciba-Geigy Corporation Microbicidally-active acylated anilino-carboxylic acid esters and their compositions
US4204002A (en) * 1974-04-09 1980-05-20 Ciba-Geigy Corporation Methods of using N-(substituted)-N-alkoxy carbonyl anilino compounds
SE429917B (sv) * 1974-04-09 1983-10-10 Ciba Geigy Ag Anvendning av vissa n-acyl-anilinettiksyraestrar for bekempning av fytopatogena svampar
DE3124091C2 (de) * 1981-06-19 1983-06-01 Degussa Ag, 6000 Frankfurt N-(3-Cyanopropanoyl)-aminocarbonsäureester und deren Verwendung
US4359416A (en) * 1981-07-13 1982-11-16 Pfizer Inc. Process for preparing L-carnosine
DE3702282A1 (de) * 1987-01-27 1988-08-04 Bayer Ag 2-cyan-2-oximino-acetamide
DE3719226A1 (de) 1987-06-09 1988-12-22 Bayer Ag (2-cyan-2-oximinoacetyl)-aminosaeure-derivate
WO1991005555A2 (en) * 1989-10-13 1991-05-02 The Salk Institute Biotechnology/Industrial Associates, Inc. N-acyl peptide metalloendopeptidase inhibitors and methods of using same
US5238930A (en) * 1991-02-06 1993-08-24 Board Of Governors Of Wayne State University Alkenoic acid compounds for mechanism-based inactivation of dehydropeptidase activity
US5112751A (en) * 1991-02-06 1992-05-12 Board Of Governors Of Wayne State University Method for inactivating dehydropepidase activity irreversibly with alkenoic acid compounds
DE4114238A1 (de) * 1991-04-26 1992-10-29 Zentralinstitut Fuer Organisch Neue substituierte 2,2 -pentamethylen-(delta)(pfeil hoch)3(pfeil hoch)-imidazolin-5-one bzw. 2,2 -pentamethylen-imidazolidin-5-one und verfahren zu deren herstellung
US5238893A (en) * 1991-12-30 1993-08-24 Bridgestone Corporation Method of preparing an anionic polymerization initiator

Also Published As

Publication number Publication date
US6878829B2 (en) 2005-04-12
US20050192354A1 (en) 2005-09-01
US7164028B2 (en) 2007-01-16
EP1259483B1 (de) 2008-04-16
WO2001064638A1 (de) 2001-09-07
US20030105335A1 (en) 2003-06-05
ATE392413T1 (de) 2008-05-15
JP2004509834A (ja) 2004-04-02
EP1259483A1 (de) 2002-11-27

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