ATE477234T1 - Synthese von phenolischen estern von hydroxymethylphenolen - Google Patents

Synthese von phenolischen estern von hydroxymethylphenolen

Info

Publication number
ATE477234T1
ATE477234T1 AT07725843T AT07725843T ATE477234T1 AT E477234 T1 ATE477234 T1 AT E477234T1 AT 07725843 T AT07725843 T AT 07725843T AT 07725843 T AT07725843 T AT 07725843T AT E477234 T1 ATE477234 T1 AT E477234T1
Authority
AT
Austria
Prior art keywords
hydroxymethylphenols
synthesis
compound
formula
phenolic esters
Prior art date
Application number
AT07725843T
Other languages
English (en)
Inventor
Seth Ennis
Roland Drews
Claus Meese
Original Assignee
Schwarz Pharma Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from IES20060433 external-priority patent/IES20060433A2/en
Application filed by Schwarz Pharma Ltd filed Critical Schwarz Pharma Ltd
Application granted granted Critical
Publication of ATE477234T1 publication Critical patent/ATE477234T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C213/00Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
    • C07C213/06Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton from hydroxy amines by reactions involving the etherification or esterification of hydroxy groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AT07725843T 2006-06-09 2007-06-05 Synthese von phenolischen estern von hydroxymethylphenolen ATE477234T1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP06011966 2006-06-09
IES20060433 IES20060433A2 (en) 2006-06-09 2006-06-09 An improved synthesis of phenolic esters of hydroxymethyl phenols
PCT/EP2007/004977 WO2007140986A1 (en) 2006-06-09 2007-06-05 Synthesis of phenolic esters of hydroxymethyl phenols

Publications (1)

Publication Number Publication Date
ATE477234T1 true ATE477234T1 (de) 2010-08-15

Family

ID=38353836

Family Applications (1)

Application Number Title Priority Date Filing Date
AT07725843T ATE477234T1 (de) 2006-06-09 2007-06-05 Synthese von phenolischen estern von hydroxymethylphenolen

Country Status (6)

Country Link
US (1) US7985873B2 (de)
EP (1) EP2004592B1 (de)
AT (1) ATE477234T1 (de)
CA (1) CA2648333C (de)
DE (1) DE602007008389D1 (de)
WO (1) WO2007140986A1 (de)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20110171274A1 (en) * 2008-07-21 2011-07-14 Actavis Group Ptc Ehf Fesoterodine Substantially Free of Dehydroxy Impurity
IT1392082B1 (it) * 2008-12-10 2012-02-09 Chemi Spa Nuove forme solide della fesoterodina fumarato
IT1394217B1 (it) 2009-05-15 2012-06-01 Chemi Spa Metodo di preparazione di fesoterodina e/o fesoterodina fumarato.
IT1394219B1 (it) 2009-05-15 2012-06-01 Chemi Spa Metodo di preparazione di fesoterodina fumarato di elevata purezza.
SI2281801T1 (sl) * 2009-07-27 2014-04-30 Crystal Pharma, S.A.U. Postopek za pridobivanje 3,3-diphenilpropilamina
US20120220655A1 (en) 2009-09-03 2012-08-30 Teva Gyogyszergyar Zartkoruen Mukodo Reszvenytarsasag Crystalline forms of fesoterodine fumarate and fesoterodine base
IT1396373B1 (it) 2009-10-29 2012-11-19 Dipharma Francis Srl Procedimento per la preparazione di fesoterodina.
IT1397521B1 (it) 2009-12-21 2013-01-16 Dipharma Francis Srl Procedimento per la preparazione di fesoterodina con un basso contenuto di impurezze.
IT1397920B1 (it) * 2010-02-08 2013-02-04 Dipharma Francis Srl Forma cristallina di fesoterodina fumarato e procedimento per la sua preparazione
WO2011141932A2 (en) 2010-05-11 2011-11-17 Intas Pharmaceuticals Limited Process for preparation of phenolic monoesters of hydroxymethyl phenols
WO2012025941A2 (en) 2010-08-25 2012-03-01 Cadila Healthcare Limited Processes for the preparation of fesoterodine
IT1403094B1 (it) * 2010-12-09 2013-10-04 Dipharma Francis Srl Procedimento per la preparazione di fesoterodina o un suo sale

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE9203318D0 (sv) 1992-11-06 1992-11-06 Kabi Pharmacia Ab Novel 3,3-diphenylpropylamines, their use and preparation
SE9701144D0 (sv) 1997-03-27 1997-03-27 Pharmacia & Upjohn Ab Novel compounds, their use and preparation
EP0957073A1 (de) * 1998-05-12 1999-11-17 Schwarz Pharma Ag 3,3-Diphenylpropylaminderivate
DE29923134U1 (de) 1999-11-16 2000-06-29 Schwarz Pharma Ag, 40789 Monheim Stabile Salze neuartiger Derviate von 3,3-Diphenylpropylaminen

Also Published As

Publication number Publication date
DE602007008389D1 (de) 2010-09-23
WO2007140986A1 (en) 2007-12-13
US7985873B2 (en) 2011-07-26
CA2648333A1 (en) 2007-12-13
EP2004592A1 (de) 2008-12-24
EP2004592B1 (de) 2010-08-11
CA2648333C (en) 2014-04-29
US20100168459A1 (en) 2010-07-01

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Legal Events

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