ATE45937T1 - Mit radioaktivhalogen markierte verbindungen, insbesondere estradiolderivate, ihre herstellung und die erhaltenen zwischenprodukte. - Google Patents

Mit radioaktivhalogen markierte verbindungen, insbesondere estradiolderivate, ihre herstellung und die erhaltenen zwischenprodukte.

Info

Publication number
ATE45937T1
ATE45937T1 AT85113214T AT85113214T ATE45937T1 AT E45937 T1 ATE45937 T1 AT E45937T1 AT 85113214 T AT85113214 T AT 85113214T AT 85113214 T AT85113214 T AT 85113214T AT E45937 T1 ATE45937 T1 AT E45937T1
Authority
AT
Austria
Prior art keywords
sup
beta
estradiol
labeled
estradiols
Prior art date
Application number
AT85113214T
Other languages
English (en)
Inventor
Richard J Baranczuk
Jay Spicer
William P Duncan
Gary A Rotert
Original Assignee
Bio Medical Research Lab Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bio Medical Research Lab Inc filed Critical Bio Medical Research Lab Inc
Application granted granted Critical
Publication of ATE45937T1 publication Critical patent/ATE45937T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0066—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa
    • C07J1/007—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J13/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17
    • C07J13/005—Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17 with double bond in position 16 (17)
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
AT85113214T 1984-10-22 1985-10-17 Mit radioaktivhalogen markierte verbindungen, insbesondere estradiolderivate, ihre herstellung und die erhaltenen zwischenprodukte. ATE45937T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US06/663,600 US4659517A (en) 1984-10-22 1984-10-22 Halogen labeled compounds including estradiol derivatives, their synthetic intermediates and the syntheses thereof
EP85113214A EP0182104B1 (de) 1984-10-22 1985-10-17 Mit Radioaktivhalogen markierte Verbindungen, insbesondere Estradiolderivate, ihre Herstellung und die erhaltenen Zwischenprodukte

Publications (1)

Publication Number Publication Date
ATE45937T1 true ATE45937T1 (de) 1989-09-15

Family

ID=24662522

Family Applications (1)

Application Number Title Priority Date Filing Date
AT85113214T ATE45937T1 (de) 1984-10-22 1985-10-17 Mit radioaktivhalogen markierte verbindungen, insbesondere estradiolderivate, ihre herstellung und die erhaltenen zwischenprodukte.

Country Status (5)

Country Link
US (1) US4659517A (de)
EP (1) EP0182104B1 (de)
JP (1) JPS62273994A (de)
AT (1) ATE45937T1 (de)
DE (1) DE3572648D1 (de)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4882141A (en) * 1984-10-22 1989-11-21 Bio-Medical Research Laboratories, Inc. Tissue imaging utilizing labelled steroids
FR2690443B1 (fr) * 1992-04-10 1995-06-30 Wallone Region Marquage des hormones par le rhenium et le technetium.
AU7013296A (en) * 1995-08-30 1997-03-19 Eli Lilly And Company N-butylsulfonate esters of estrogens
KR100368103B1 (ko) * 1998-05-28 2004-05-20 주식회사 태평양 에스트로겐유도체및그의염,및이를함유하는모발생장촉진조성물
US20050049487A1 (en) * 2003-08-26 2005-03-03 Johnson Bruce Fletcher Compounds and kits for preparing imaging agents and methods of imaging
US20070059239A1 (en) * 2005-09-15 2007-03-15 Estradiol Images, Llc A Missouri Limited Liability Company Process for the preparation of radioactive labeled estradiol

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4465676A (en) * 1980-04-09 1984-08-14 New England Nuclear Corporation 16α Halogen substituted 3,17β-dihydroxy steroidal estrogens

Also Published As

Publication number Publication date
EP0182104B1 (de) 1989-08-30
US4659517A (en) 1987-04-21
DE3572648D1 (en) 1989-10-05
EP0182104A1 (de) 1986-05-28
JPS62273994A (ja) 1987-11-28

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Legal Events

Date Code Title Description
RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties