ATE452630T1 - Fungizide medikamente enthaltend arylamidinderivate - Google Patents
Fungizide medikamente enthaltend arylamidinderivateInfo
- Publication number
- ATE452630T1 ATE452630T1 AT03767675T AT03767675T ATE452630T1 AT E452630 T1 ATE452630 T1 AT E452630T1 AT 03767675 T AT03767675 T AT 03767675T AT 03767675 T AT03767675 T AT 03767675T AT E452630 T1 ATE452630 T1 AT E452630T1
- Authority
- AT
- Austria
- Prior art keywords
- optionally substituted
- alkyl
- alkynyl
- acyl
- alkenyl
- Prior art date
Links
- 239000003814 drug Substances 0.000 title 1
- 229940079593 drug Drugs 0.000 title 1
- 230000000855 fungicidal effect Effects 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 abstract 6
- 125000000623 heterocyclic group Chemical group 0.000 abstract 6
- 229910052760 oxygen Inorganic materials 0.000 abstract 5
- 125000002252 acyl group Chemical group 0.000 abstract 4
- 125000003342 alkenyl group Chemical group 0.000 abstract 4
- 125000000304 alkynyl group Chemical group 0.000 abstract 4
- 125000002837 carbocyclic group Chemical group 0.000 abstract 4
- 229910052739 hydrogen Inorganic materials 0.000 abstract 4
- 239000001257 hydrogen Substances 0.000 abstract 4
- 150000003839 salts Chemical class 0.000 abstract 4
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 3
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 3
- 239000001301 oxygen Substances 0.000 abstract 3
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 2
- 239000002253 acid Substances 0.000 abstract 2
- 150000007513 acids Chemical class 0.000 abstract 2
- 239000012871 anti-fungal composition Substances 0.000 abstract 2
- MPVDXIMFBOLMNW-UHFFFAOYSA-N chembl1615565 Chemical compound OC1=CC=C2C=C(S(O)(=O)=O)C=C(S(O)(=O)=O)C2=C1N=NC1=CC=CC=C1 MPVDXIMFBOLMNW-UHFFFAOYSA-N 0.000 abstract 2
- 125000001475 halogen functional group Chemical group 0.000 abstract 2
- 150000002431 hydrogen Chemical group 0.000 abstract 2
- -1 hydroxy, mercapto Chemical class 0.000 abstract 2
- 230000003287 optical effect Effects 0.000 abstract 2
- 229910052717 sulfur Inorganic materials 0.000 abstract 2
- HCMJWOGOISXSDL-UHFFFAOYSA-N (2-isothiocyanato-1-phenylethyl)benzene Chemical compound C=1C=CC=CC=1C(CN=C=S)C1=CC=CC=C1 HCMJWOGOISXSDL-UHFFFAOYSA-N 0.000 abstract 1
- 101100439663 Arabidopsis thaliana CHR7 gene Proteins 0.000 abstract 1
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical group [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 125000004414 alkyl thio group Chemical group 0.000 abstract 1
- 125000000852 azido group Chemical group *N=[N+]=[N-] 0.000 abstract 1
- 125000005677 ethinylene group Chemical group [*:2]C#C[*:1] 0.000 abstract 1
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1
- 239000011593 sulfur Chemical group 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP02356210A EP1413301A1 (fr) | 2002-10-24 | 2002-10-24 | Médicaments antifongiques à base de dérivés d'arylamidine |
| PCT/EP2003/013335 WO2004037239A1 (en) | 2002-10-24 | 2003-10-24 | Antifungal medicaments based on arylamidine derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE452630T1 true ATE452630T1 (de) | 2010-01-15 |
Family
ID=32050123
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT03767675T ATE452630T1 (de) | 2002-10-24 | 2003-10-24 | Fungizide medikamente enthaltend arylamidinderivate |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20060052459A1 (enExample) |
| EP (2) | EP1413301A1 (enExample) |
| JP (1) | JP4624105B2 (enExample) |
| AT (1) | ATE452630T1 (enExample) |
| AU (1) | AU2003292131A1 (enExample) |
| CA (1) | CA2502433A1 (enExample) |
| DE (1) | DE60330702D1 (enExample) |
| WO (1) | WO2004037239A1 (enExample) |
Families Citing this family (35)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1570736A1 (en) * | 2004-03-05 | 2005-09-07 | Bayer CropScience S.A. | Fungicide composition comprising an arylamidine derivative and known fungicide compounds |
| BRPI0616000B1 (pt) * | 2005-09-13 | 2016-04-19 | Bayer Cropscience Ag | composto derivado de fenil-amidina, processo de preparação de composto, composto derivado de nitrofeniléter, composto derivado de aminofeniléter, método de controle de fungos fitopatogênicos de safras e método de controle de insetos daninhos. |
| EP1969931A1 (de) | 2007-03-12 | 2008-09-17 | Bayer CropScience Aktiengesellschaft | Fluoalkylphenylamidine und deren Verwendung als Fungizide |
| BRPI0808798A2 (pt) | 2007-03-12 | 2014-10-07 | Bayer Cropscience Ag | Fenoxifenilamidinas 3,5-dissubstituídas e seu uso como fungicidas |
| EP1969929A1 (de) | 2007-03-12 | 2008-09-17 | Bayer CropScience AG | Substituierte Phenylamidine und deren Verwendung als Fungizide |
| EP1969934A1 (de) * | 2007-03-12 | 2008-09-17 | Bayer CropScience AG | 4-Cycloalkyl-oder 4-arylsubstituierte Phenoxyphenylamidine und deren Verwendung als Fungizide |
| EP1969933A1 (de) * | 2007-03-12 | 2008-09-17 | Bayer CropScience AG | Dihalogenphenoxyphenylamidine und deren Verwendung als Fungizide |
| EP1969935A1 (de) * | 2007-03-12 | 2008-09-17 | Bayer CropScience AG | 3,4-Disubstituierte Phenoxyphenylamidine und deren Verwendung als Fungizide |
| WO2008110279A1 (de) * | 2007-03-12 | 2008-09-18 | Bayer Cropscience Ag | Dihalogenphenoxyphenylamidine und deren verwendung als fungizide |
| EP1969930A1 (de) * | 2007-03-12 | 2008-09-17 | Bayer CropScience AG | Phenoxyphenylamidine und deren Verwendung als Fungizide |
| EP1969932A1 (de) * | 2007-03-12 | 2008-09-17 | Bayer CropScience AG | Phenoxyphenylamidine und deren Verwendung als Fungizide |
| BRPI0808846A2 (pt) | 2007-03-12 | 2019-09-24 | Bayer Cropscience Ag | fenoxifenilamidinas 3-substituídas e seu uso como fungicidas |
| US8168567B2 (en) * | 2007-04-19 | 2012-05-01 | Bayer Cropscience Ag | Thiadiazolyl oxyphenyl amidines and the use thereof as a fungicide |
| EP2072506A1 (de) | 2007-12-21 | 2009-06-24 | Bayer CropScience AG | Thiazolyloxyphenylamidine oder Thiadiazolyloxyphenylamidine und deren Verwendung als Fungizide |
| CN102066347B (zh) * | 2008-06-27 | 2016-06-08 | 拜耳知识产权有限责任公司 | 噻二唑氧苯基脒及其作为杀菌剂的应用 |
| UA106875C2 (uk) | 2008-06-27 | 2014-10-27 | Баєр Кропсаєнс Аг | Тіадіазолілоксифеніламідини та їх застосування як фунгіцидів |
| EP2223917A1 (de) | 2009-02-02 | 2010-09-01 | Bayer CropScience AG | Isothiazolyloxyphenylamidine und deren Verwendung als Fungizide |
| EP2264011A1 (de) | 2009-06-03 | 2010-12-22 | Bayer CropScience AG | Heteroarylamidine und deren Verwendung als Fungizide |
| EP2264012A1 (de) | 2009-06-03 | 2010-12-22 | Bayer CropScience AG | Heteroarylamidine und deren Verwendung als Fungizide |
| WO2011006604A1 (de) | 2009-07-17 | 2011-01-20 | Bayer Cropscience Ag | Substituierte aminothiazole und deren verwendung als fungizide |
| WO2011082941A1 (de) | 2009-12-16 | 2011-07-14 | Bayer Cropscience Ag | Benzylsubstituierte thiadiazolyloxyphenylamidiniumsalze als fungizide |
| WO2012019998A1 (de) | 2010-08-10 | 2012-02-16 | Bayer Cropscience Ag | Herstellung von n'-(4-{[3-(4-chlorbenzyl)-1,2,4-thiadiazol-5-yl]oxy}-2,5-dimethylphenyl)-n-ethyl-n-methylimidoformamid |
| ES2563232T3 (es) | 2011-07-29 | 2016-03-11 | Taisho Pharmaceutical Co., Ltd. | Compuesto de amidina o sal del mismo |
| WO2013076666A1 (en) * | 2011-11-23 | 2013-05-30 | Newsouth Innovations Pty Limited | Antimicrobial peptides and uses thereof |
| WO2016043260A1 (ja) * | 2014-09-19 | 2016-03-24 | 塩野義製薬株式会社 | 環状グアニジンまたはアミジン化合物 |
| HUE051950T2 (hu) | 2015-06-15 | 2021-04-28 | Bayer Cropscience Ag | Halogén-szubsztituált fenoxifenilamidinok és alkalmazásuk fungicidként |
| EP3307706B1 (en) | 2015-06-15 | 2019-07-24 | Bayer CropScience AG | Halogen-substituted phenoxyphenylamidines and the use thereof as fungicides |
| EP3319937A1 (en) | 2015-07-08 | 2018-05-16 | Bayer CropScience Aktiengesellschaft | Phenoxyhalogenphenylamidines and the use thereof as fungicides |
| EP3335559A1 (en) | 2016-12-14 | 2018-06-20 | Bayer CropScience Aktiengesellschaft | Active compound combinations |
| BR112019012272A2 (pt) | 2016-12-14 | 2019-12-03 | Bayer Ag | fenilamidinas e seu uso como fungicidas |
| BR112019012219A2 (pt) | 2016-12-14 | 2019-11-12 | Bayer Cropscience Aktiengesellschaft | fenoxifenilamidinas e o uso das mesmas como fungicidas |
| WO2018109002A1 (en) | 2016-12-14 | 2018-06-21 | Bayer Cropscience Aktiengesellschaft | Active compound combinations |
| EP3708565A1 (en) | 2020-03-04 | 2020-09-16 | Bayer AG | Pyrimidinyloxyphenylamidines and the use thereof as fungicides |
| EP3915971A1 (en) | 2020-12-16 | 2021-12-01 | Bayer Aktiengesellschaft | Phenyl-s(o)n-phenylamidines and the use thereof as fungicides |
| CN121717732A (zh) * | 2024-09-21 | 2026-03-24 | 青岛清原化合物有限公司 | 苯基脒类化合物及其应用 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3217770A1 (de) * | 1982-05-12 | 1983-11-17 | Hoechst Ag, 6230 Frankfurt | 1-(1,3-dioxolan-2-yl-methyl)-1h-imidazole und -1h-1,2,4-triazole und deren salze, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung |
| EP0957101A1 (en) * | 1998-05-14 | 1999-11-17 | Janssen Pharmaceutica N.V. | Water soluble azoles as broad-spectrum antifungals |
| GB9902592D0 (en) * | 1999-02-06 | 1999-03-24 | Hoechst Schering Agrevo Gmbh | Fungicides |
| EP1278755A2 (en) * | 2000-03-07 | 2003-01-29 | Ranbaxy Laboratories, Limited | Azole compounds as therapeutic agents for fungal infections |
| EP1178038A1 (en) * | 2000-08-04 | 2002-02-06 | Aventis Cropscience S.A. | Fungicidal phenylamidine derivatives |
| EP1337510A4 (en) * | 2000-11-06 | 2005-02-23 | Univ North Carolina | SYNTHESIS AND ANTIMICROBIAL ACTIVITY OF NEW DICATIONIC REVERSED AMIDINES |
-
2002
- 2002-10-24 EP EP02356210A patent/EP1413301A1/fr not_active Withdrawn
-
2003
- 2003-10-24 WO PCT/EP2003/013335 patent/WO2004037239A1/en not_active Ceased
- 2003-10-24 JP JP2004546028A patent/JP4624105B2/ja not_active Expired - Fee Related
- 2003-10-24 AT AT03767675T patent/ATE452630T1/de not_active IP Right Cessation
- 2003-10-24 DE DE60330702T patent/DE60330702D1/de not_active Expired - Lifetime
- 2003-10-24 US US10/532,033 patent/US20060052459A1/en not_active Abandoned
- 2003-10-24 CA CA002502433A patent/CA2502433A1/en not_active Abandoned
- 2003-10-24 EP EP03767675A patent/EP1562569B1/en not_active Expired - Lifetime
- 2003-10-24 AU AU2003292131A patent/AU2003292131A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| JP4624105B2 (ja) | 2011-02-02 |
| US20060052459A1 (en) | 2006-03-09 |
| EP1413301A1 (fr) | 2004-04-28 |
| EP1562569A1 (en) | 2005-08-17 |
| JP2006505576A (ja) | 2006-02-16 |
| CA2502433A1 (en) | 2004-05-06 |
| AU2003292131A1 (en) | 2004-05-13 |
| EP1562569B1 (en) | 2009-12-23 |
| WO2004037239A1 (en) | 2004-05-06 |
| DE60330702D1 (de) | 2010-02-04 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |