ATE452630T1 - Fungizide medikamente enthaltend arylamidinderivate - Google Patents
Fungizide medikamente enthaltend arylamidinderivateInfo
- Publication number
- ATE452630T1 ATE452630T1 AT03767675T AT03767675T ATE452630T1 AT E452630 T1 ATE452630 T1 AT E452630T1 AT 03767675 T AT03767675 T AT 03767675T AT 03767675 T AT03767675 T AT 03767675T AT E452630 T1 ATE452630 T1 AT E452630T1
- Authority
- AT
- Austria
- Prior art keywords
- optionally substituted
- alkyl
- alkynyl
- acyl
- alkenyl
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP02356210A EP1413301A1 (de) | 2002-10-24 | 2002-10-24 | Antimykotische Medikamente auf der Basis von Arylamidinderivaten |
PCT/EP2003/013335 WO2004037239A1 (en) | 2002-10-24 | 2003-10-24 | Antifungal medicaments based on arylamidine derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE452630T1 true ATE452630T1 (de) | 2010-01-15 |
Family
ID=32050123
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT03767675T ATE452630T1 (de) | 2002-10-24 | 2003-10-24 | Fungizide medikamente enthaltend arylamidinderivate |
Country Status (8)
Country | Link |
---|---|
US (1) | US20060052459A1 (de) |
EP (2) | EP1413301A1 (de) |
JP (1) | JP4624105B2 (de) |
AT (1) | ATE452630T1 (de) |
AU (1) | AU2003292131A1 (de) |
CA (1) | CA2502433A1 (de) |
DE (1) | DE60330702D1 (de) |
WO (1) | WO2004037239A1 (de) |
Families Citing this family (34)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1570736A1 (de) * | 2004-03-05 | 2005-09-07 | Bayer CropScience S.A. | Fungizid-Zusammensetzung enthaltend ein Arylamidin und bekannte Fungizid-Verbindungen |
JP5261181B2 (ja) * | 2005-09-13 | 2013-08-14 | バイエル・クロップサイエンス・アーゲー | 殺虫剤フェニルオキシ置換フェニルアミジン誘導体 |
EP2120558B1 (de) * | 2007-03-12 | 2016-02-10 | Bayer Intellectual Property GmbH | 3,4-Disubstituierte Phenoxyphenylamidin-Derivate und deren Verwendung als Fungizide |
EP1969930A1 (de) * | 2007-03-12 | 2008-09-17 | Bayer CropScience AG | Phenoxyphenylamidine und deren Verwendung als Fungizide |
EP1969932A1 (de) * | 2007-03-12 | 2008-09-17 | Bayer CropScience AG | Phenoxyphenylamidine und deren Verwendung als Fungizide |
EP1969933A1 (de) * | 2007-03-12 | 2008-09-17 | Bayer CropScience AG | Dihalogenphenoxyphenylamidine und deren Verwendung als Fungizide |
EP1969929A1 (de) | 2007-03-12 | 2008-09-17 | Bayer CropScience AG | Substituierte Phenylamidine und deren Verwendung als Fungizide |
EP1969931A1 (de) | 2007-03-12 | 2008-09-17 | Bayer CropScience Aktiengesellschaft | Fluoalkylphenylamidine und deren Verwendung als Fungizide |
EP1969934A1 (de) * | 2007-03-12 | 2008-09-17 | Bayer CropScience AG | 4-Cycloalkyl-oder 4-arylsubstituierte Phenoxyphenylamidine und deren Verwendung als Fungizide |
EP2136628B1 (de) | 2007-03-12 | 2015-07-01 | Bayer Intellectual Property GmbH | Phenoxy-substituierte phenylamidin-derivate und deren verwendung als fungizide |
WO2008110279A1 (de) * | 2007-03-12 | 2008-09-18 | Bayer Cropscience Ag | Dihalogenphenoxyphenylamidine und deren verwendung als fungizide |
EP1969935A1 (de) * | 2007-03-12 | 2008-09-17 | Bayer CropScience AG | 3,4-Disubstituierte Phenoxyphenylamidine und deren Verwendung als Fungizide |
JP2010524869A (ja) * | 2007-04-19 | 2010-07-22 | バイエル・クロツプサイエンス・アクチエンゲゼルシヤフト | チアジアゾリルオキシフェニルアミジンおよび殺菌剤としてのこれらの使用 |
EP2072506A1 (de) | 2007-12-21 | 2009-06-24 | Bayer CropScience AG | Thiazolyloxyphenylamidine oder Thiadiazolyloxyphenylamidine und deren Verwendung als Fungizide |
CA2729432A1 (en) | 2008-06-27 | 2009-12-30 | Bayer Cropscience Ag | Thiadiazolyloxyphenylamidines and use thereof as fungicides |
BRPI0913885A8 (pt) | 2008-06-27 | 2016-08-02 | Bayer Cropscience Ag | tiadiazoliloxifenilamidinas e seu uso como fungicidas |
EP2223917A1 (de) | 2009-02-02 | 2010-09-01 | Bayer CropScience AG | Isothiazolyloxyphenylamidine und deren Verwendung als Fungizide |
EP2264011A1 (de) | 2009-06-03 | 2010-12-22 | Bayer CropScience AG | Heteroarylamidine und deren Verwendung als Fungizide |
EP2264012A1 (de) | 2009-06-03 | 2010-12-22 | Bayer CropScience AG | Heteroarylamidine und deren Verwendung als Fungizide |
WO2011006604A1 (de) | 2009-07-17 | 2011-01-20 | Bayer Cropscience Ag | Substituierte aminothiazole und deren verwendung als fungizide |
WO2011082941A1 (de) | 2009-12-16 | 2011-07-14 | Bayer Cropscience Ag | Benzylsubstituierte thiadiazolyloxyphenylamidiniumsalze als fungizide |
WO2012019998A1 (de) | 2010-08-10 | 2012-02-16 | Bayer Cropscience Ag | Herstellung von n'-(4-{[3-(4-chlorbenzyl)-1,2,4-thiadiazol-5-yl]oxy}-2,5-dimethylphenyl)-n-ethyl-n-methylimidoformamid |
KR20140045511A (ko) | 2011-07-29 | 2014-04-16 | 다이쇼 세이야꾸 가부시끼가이샤 | 아미딘 화합물 또는 그의 염 |
US20140315789A1 (en) * | 2011-11-23 | 2014-10-23 | Newsouth Innovations Pty Limited | Antimicrobial peptides and uses thereof |
WO2016043260A1 (ja) * | 2014-09-19 | 2016-03-24 | 塩野義製薬株式会社 | 環状グアニジンまたはアミジン化合物 |
LT3307707T (lt) | 2015-06-15 | 2021-01-11 | Syngenta Crop Protection Ag | Halogeninti fenoksifenilamidinai ir jų naudojimas kaip fungicidų |
US10252977B2 (en) | 2015-06-15 | 2019-04-09 | Bayer Cropscience Aktiengesellschaft | Halogen-substituted phenoxyphenylamidines and the use thereof as fungicides |
BR112018000390A2 (pt) | 2015-07-08 | 2018-09-11 | Bayer Cropscience Ag | fenoxihalogenofenilamidinas e o uso dessas como fungicidas |
EP3335559A1 (de) | 2016-12-14 | 2018-06-20 | Bayer CropScience Aktiengesellschaft | Wirkstoffkombinationen |
WO2018109002A1 (en) | 2016-12-14 | 2018-06-21 | Bayer Cropscience Aktiengesellschaft | Active compound combinations |
US20190308933A1 (en) | 2016-12-14 | 2019-10-10 | Bayer Cropscience Aktiengesellschaft | Phenylamidines and the use thereof as fungicides |
AU2017375006A1 (en) | 2016-12-14 | 2019-07-04 | Bayer Aktiengesellschaft | Phenoxyphenylamidines and the use thereof as fungicides |
EP3708565A1 (de) | 2020-03-04 | 2020-09-16 | Bayer AG | Pyrimidinyloxyphenylamidine und ihre verwendung als fungizide |
EP3915971A1 (de) | 2020-12-16 | 2021-12-01 | Bayer Aktiengesellschaft | Phenyl-s(o)n-phenylamidine und verwendung davon als fungizide |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3217770A1 (de) * | 1982-05-12 | 1983-11-17 | Hoechst Ag, 6230 Frankfurt | 1-(1,3-dioxolan-2-yl-methyl)-1h-imidazole und -1h-1,2,4-triazole und deren salze, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung |
EP0957101A1 (de) * | 1998-05-14 | 1999-11-17 | Janssen Pharmaceutica N.V. | Wasserlösliche Azole als Breitspektrum-antifungus |
GB9902592D0 (en) * | 1999-02-06 | 1999-03-24 | Hoechst Schering Agrevo Gmbh | Fungicides |
JP2004501867A (ja) * | 2000-03-07 | 2004-01-22 | ランバクシー ラボラトリーズ リミテッド | 真菌感染症に対する治療薬としてのアゾール化合物 |
EP1178038A1 (de) * | 2000-08-04 | 2002-02-06 | Aventis Cropscience S.A. | Fungizide Phenylamidin Derivative |
AU2002246600B2 (en) * | 2000-11-06 | 2005-08-25 | Duke University | Synthesis and antimicrobial activity of novel dicationic "Reversed amidines" |
-
2002
- 2002-10-24 EP EP02356210A patent/EP1413301A1/de not_active Withdrawn
-
2003
- 2003-10-24 AT AT03767675T patent/ATE452630T1/de not_active IP Right Cessation
- 2003-10-24 WO PCT/EP2003/013335 patent/WO2004037239A1/en active Application Filing
- 2003-10-24 US US10/532,033 patent/US20060052459A1/en not_active Abandoned
- 2003-10-24 EP EP03767675A patent/EP1562569B1/de not_active Expired - Lifetime
- 2003-10-24 AU AU2003292131A patent/AU2003292131A1/en not_active Abandoned
- 2003-10-24 CA CA002502433A patent/CA2502433A1/en not_active Abandoned
- 2003-10-24 JP JP2004546028A patent/JP4624105B2/ja not_active Expired - Fee Related
- 2003-10-24 DE DE60330702T patent/DE60330702D1/de not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
WO2004037239A1 (en) | 2004-05-06 |
EP1562569A1 (de) | 2005-08-17 |
JP2006505576A (ja) | 2006-02-16 |
JP4624105B2 (ja) | 2011-02-02 |
EP1562569B1 (de) | 2009-12-23 |
DE60330702D1 (de) | 2010-02-04 |
EP1413301A1 (de) | 2004-04-28 |
US20060052459A1 (en) | 2006-03-09 |
CA2502433A1 (en) | 2004-05-06 |
AU2003292131A1 (en) | 2004-05-13 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |