ATE452630T1 - Fungizide medikamente enthaltend arylamidinderivate - Google Patents

Fungizide medikamente enthaltend arylamidinderivate

Info

Publication number
ATE452630T1
ATE452630T1 AT03767675T AT03767675T ATE452630T1 AT E452630 T1 ATE452630 T1 AT E452630T1 AT 03767675 T AT03767675 T AT 03767675T AT 03767675 T AT03767675 T AT 03767675T AT E452630 T1 ATE452630 T1 AT E452630T1
Authority
AT
Austria
Prior art keywords
optionally substituted
alkyl
alkynyl
acyl
alkenyl
Prior art date
Application number
AT03767675T
Other languages
English (en)
Inventor
Jean-Pierre Vors
Elizabeth O'neill
Gilbert Labourdette
Gillian Mansfield
John Pillmoor
Thierry Barchietto
Original Assignee
Bayer Cropscience Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Sa filed Critical Bayer Cropscience Sa
Application granted granted Critical
Publication of ATE452630T1 publication Critical patent/ATE452630T1/de

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/155Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
AT03767675T 2002-10-24 2003-10-24 Fungizide medikamente enthaltend arylamidinderivate ATE452630T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP02356210A EP1413301A1 (de) 2002-10-24 2002-10-24 Antimykotische Medikamente auf der Basis von Arylamidinderivaten
PCT/EP2003/013335 WO2004037239A1 (en) 2002-10-24 2003-10-24 Antifungal medicaments based on arylamidine derivatives

Publications (1)

Publication Number Publication Date
ATE452630T1 true ATE452630T1 (de) 2010-01-15

Family

ID=32050123

Family Applications (1)

Application Number Title Priority Date Filing Date
AT03767675T ATE452630T1 (de) 2002-10-24 2003-10-24 Fungizide medikamente enthaltend arylamidinderivate

Country Status (8)

Country Link
US (1) US20060052459A1 (de)
EP (2) EP1413301A1 (de)
JP (1) JP4624105B2 (de)
AT (1) ATE452630T1 (de)
AU (1) AU2003292131A1 (de)
CA (1) CA2502433A1 (de)
DE (1) DE60330702D1 (de)
WO (1) WO2004037239A1 (de)

Families Citing this family (34)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1570736A1 (de) * 2004-03-05 2005-09-07 Bayer CropScience S.A. Fungizid-Zusammensetzung enthaltend ein Arylamidin und bekannte Fungizid-Verbindungen
JP5261181B2 (ja) * 2005-09-13 2013-08-14 バイエル・クロップサイエンス・アーゲー 殺虫剤フェニルオキシ置換フェニルアミジン誘導体
EP2120558B1 (de) * 2007-03-12 2016-02-10 Bayer Intellectual Property GmbH 3,4-Disubstituierte Phenoxyphenylamidin-Derivate und deren Verwendung als Fungizide
EP1969930A1 (de) * 2007-03-12 2008-09-17 Bayer CropScience AG Phenoxyphenylamidine und deren Verwendung als Fungizide
EP1969932A1 (de) * 2007-03-12 2008-09-17 Bayer CropScience AG Phenoxyphenylamidine und deren Verwendung als Fungizide
EP1969933A1 (de) * 2007-03-12 2008-09-17 Bayer CropScience AG Dihalogenphenoxyphenylamidine und deren Verwendung als Fungizide
EP1969929A1 (de) 2007-03-12 2008-09-17 Bayer CropScience AG Substituierte Phenylamidine und deren Verwendung als Fungizide
EP1969931A1 (de) 2007-03-12 2008-09-17 Bayer CropScience Aktiengesellschaft Fluoalkylphenylamidine und deren Verwendung als Fungizide
EP1969934A1 (de) * 2007-03-12 2008-09-17 Bayer CropScience AG 4-Cycloalkyl-oder 4-arylsubstituierte Phenoxyphenylamidine und deren Verwendung als Fungizide
EP2136628B1 (de) 2007-03-12 2015-07-01 Bayer Intellectual Property GmbH Phenoxy-substituierte phenylamidin-derivate und deren verwendung als fungizide
WO2008110279A1 (de) * 2007-03-12 2008-09-18 Bayer Cropscience Ag Dihalogenphenoxyphenylamidine und deren verwendung als fungizide
EP1969935A1 (de) * 2007-03-12 2008-09-17 Bayer CropScience AG 3,4-Disubstituierte Phenoxyphenylamidine und deren Verwendung als Fungizide
JP2010524869A (ja) * 2007-04-19 2010-07-22 バイエル・クロツプサイエンス・アクチエンゲゼルシヤフト チアジアゾリルオキシフェニルアミジンおよび殺菌剤としてのこれらの使用
EP2072506A1 (de) 2007-12-21 2009-06-24 Bayer CropScience AG Thiazolyloxyphenylamidine oder Thiadiazolyloxyphenylamidine und deren Verwendung als Fungizide
CA2729432A1 (en) 2008-06-27 2009-12-30 Bayer Cropscience Ag Thiadiazolyloxyphenylamidines and use thereof as fungicides
BRPI0913885A8 (pt) 2008-06-27 2016-08-02 Bayer Cropscience Ag tiadiazoliloxifenilamidinas e seu uso como fungicidas
EP2223917A1 (de) 2009-02-02 2010-09-01 Bayer CropScience AG Isothiazolyloxyphenylamidine und deren Verwendung als Fungizide
EP2264011A1 (de) 2009-06-03 2010-12-22 Bayer CropScience AG Heteroarylamidine und deren Verwendung als Fungizide
EP2264012A1 (de) 2009-06-03 2010-12-22 Bayer CropScience AG Heteroarylamidine und deren Verwendung als Fungizide
WO2011006604A1 (de) 2009-07-17 2011-01-20 Bayer Cropscience Ag Substituierte aminothiazole und deren verwendung als fungizide
WO2011082941A1 (de) 2009-12-16 2011-07-14 Bayer Cropscience Ag Benzylsubstituierte thiadiazolyloxyphenylamidiniumsalze als fungizide
WO2012019998A1 (de) 2010-08-10 2012-02-16 Bayer Cropscience Ag Herstellung von n'-(4-{[3-(4-chlorbenzyl)-1,2,4-thiadiazol-5-yl]oxy}-2,5-dimethylphenyl)-n-ethyl-n-methylimidoformamid
KR20140045511A (ko) 2011-07-29 2014-04-16 다이쇼 세이야꾸 가부시끼가이샤 아미딘 화합물 또는 그의 염
US20140315789A1 (en) * 2011-11-23 2014-10-23 Newsouth Innovations Pty Limited Antimicrobial peptides and uses thereof
WO2016043260A1 (ja) * 2014-09-19 2016-03-24 塩野義製薬株式会社 環状グアニジンまたはアミジン化合物
LT3307707T (lt) 2015-06-15 2021-01-11 Syngenta Crop Protection Ag Halogeninti fenoksifenilamidinai ir jų naudojimas kaip fungicidų
US10252977B2 (en) 2015-06-15 2019-04-09 Bayer Cropscience Aktiengesellschaft Halogen-substituted phenoxyphenylamidines and the use thereof as fungicides
BR112018000390A2 (pt) 2015-07-08 2018-09-11 Bayer Cropscience Ag fenoxihalogenofenilamidinas e o uso dessas como fungicidas
EP3335559A1 (de) 2016-12-14 2018-06-20 Bayer CropScience Aktiengesellschaft Wirkstoffkombinationen
WO2018109002A1 (en) 2016-12-14 2018-06-21 Bayer Cropscience Aktiengesellschaft Active compound combinations
US20190308933A1 (en) 2016-12-14 2019-10-10 Bayer Cropscience Aktiengesellschaft Phenylamidines and the use thereof as fungicides
AU2017375006A1 (en) 2016-12-14 2019-07-04 Bayer Aktiengesellschaft Phenoxyphenylamidines and the use thereof as fungicides
EP3708565A1 (de) 2020-03-04 2020-09-16 Bayer AG Pyrimidinyloxyphenylamidine und ihre verwendung als fungizide
EP3915971A1 (de) 2020-12-16 2021-12-01 Bayer Aktiengesellschaft Phenyl-s(o)n-phenylamidine und verwendung davon als fungizide

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3217770A1 (de) * 1982-05-12 1983-11-17 Hoechst Ag, 6230 Frankfurt 1-(1,3-dioxolan-2-yl-methyl)-1h-imidazole und -1h-1,2,4-triazole und deren salze, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung
EP0957101A1 (de) * 1998-05-14 1999-11-17 Janssen Pharmaceutica N.V. Wasserlösliche Azole als Breitspektrum-antifungus
GB9902592D0 (en) * 1999-02-06 1999-03-24 Hoechst Schering Agrevo Gmbh Fungicides
JP2004501867A (ja) * 2000-03-07 2004-01-22 ランバクシー ラボラトリーズ リミテッド 真菌感染症に対する治療薬としてのアゾール化合物
EP1178038A1 (de) * 2000-08-04 2002-02-06 Aventis Cropscience S.A. Fungizide Phenylamidin Derivative
AU2002246600B2 (en) * 2000-11-06 2005-08-25 Duke University Synthesis and antimicrobial activity of novel dicationic "Reversed amidines"

Also Published As

Publication number Publication date
WO2004037239A1 (en) 2004-05-06
EP1562569A1 (de) 2005-08-17
JP2006505576A (ja) 2006-02-16
JP4624105B2 (ja) 2011-02-02
EP1562569B1 (de) 2009-12-23
DE60330702D1 (de) 2010-02-04
EP1413301A1 (de) 2004-04-28
US20060052459A1 (en) 2006-03-09
CA2502433A1 (en) 2004-05-06
AU2003292131A1 (en) 2004-05-13

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