ATE449773T1 - Homomorpholinoxazolidinone als antibakterielle mittel - Google Patents

Homomorpholinoxazolidinone als antibakterielle mittel

Info

Publication number
ATE449773T1
ATE449773T1 AT06779767T AT06779767T ATE449773T1 AT E449773 T1 ATE449773 T1 AT E449773T1 AT 06779767 T AT06779767 T AT 06779767T AT 06779767 T AT06779767 T AT 06779767T AT E449773 T1 ATE449773 T1 AT E449773T1
Authority
AT
Austria
Prior art keywords
sup
sub
antibacterial agents
homomorpholinoxazolidinones
het
Prior art date
Application number
AT06779767T
Other languages
German (de)
English (en)
Inventor
Vara Prasad Venkata Nagendra Josyula
Frederick Earl Boyer Jr
Ji-Young Kim
Original Assignee
Pharmacia & Upjohn Co Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia & Upjohn Co Llc filed Critical Pharmacia & Upjohn Co Llc
Application granted granted Critical
Publication of ATE449773T1 publication Critical patent/ATE449773T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
AT06779767T 2005-06-29 2006-06-20 Homomorpholinoxazolidinone als antibakterielle mittel ATE449773T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US69486205P 2005-06-29 2005-06-29
PCT/IB2006/001730 WO2007000644A1 (en) 2005-06-29 2006-06-20 Homomorpholine oxazolidinones as antibacterial agents

Publications (1)

Publication Number Publication Date
ATE449773T1 true ATE449773T1 (de) 2009-12-15

Family

ID=37101665

Family Applications (1)

Application Number Title Priority Date Filing Date
AT06779767T ATE449773T1 (de) 2005-06-29 2006-06-20 Homomorpholinoxazolidinone als antibakterielle mittel

Country Status (8)

Country Link
EP (1) EP1899331B1 (enExample)
JP (1) JP2008544979A (enExample)
AT (1) ATE449773T1 (enExample)
CA (1) CA2610978A1 (enExample)
DE (1) DE602006010702D1 (enExample)
DK (1) DK1899331T3 (enExample)
ES (1) ES2335307T3 (enExample)
WO (1) WO2007000644A1 (enExample)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101460495B (zh) 2006-03-31 2013-08-14 财团法人乙卯研究所 具有杂环的化合物
JP5455906B2 (ja) * 2007-08-06 2014-03-26 ミクウルク ファーマシューティカルズ，インコーポレイテッド 細菌感染症治療のための抗微生物性オルト−フルオロフェニルオキサゾリジノン
EP2669283A1 (en) * 2007-10-02 2013-12-04 Shionogi&Co., Ltd. Oxazolidinone derivative having 7-membered hetero ring
CA2939098A1 (en) 2014-02-21 2015-08-27 Micurx Pharmaceuticals, Inc. Water-soluble o-carbonyl phosphoramidate prodrugs for therapeutic administration
CN113603683B (zh) * 2015-07-17 2024-06-14 结核病药物开发全球联盟公司 用于抗微生物治疗的经取代苯基噁唑烷酮

Family Cites Families (33)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SK283420B6 (sk) 1992-05-08 2003-07-01 Pharmacia & Upjohn Company Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny
MY115155A (en) 1993-09-09 2003-04-30 Upjohn Co Substituted oxazine and thiazine oxazolidinone antimicrobials.
US5952324A (en) 1994-11-15 1999-09-14 Pharmacia & Upjohn Company Bicyclic oxazine and thiazine oxazolidinone antibacterials
CN1154644C (zh) 1997-11-12 2004-06-23 法玛西雅厄普约翰美国公司 噁唑烷酮衍生物和药物组合物
JP2000204084A (ja) 1998-11-11 2000-07-25 Hokuriku Seiyaku Co Ltd チオカルバミド酸誘導体
HK1040707A1 (zh) 1998-11-27 2002-06-21 法玛西雅厄普约翰美国公司 具有硫代羰基官能團的噁唑烷酮抗菌劑
US6297242B1 (en) 1999-08-12 2001-10-02 Ortho-Mcneil Pharmaceutical, Inc. N-substituted amidine and guanidine oxazolidinone antibacterials and methods of use thereof
SK7572002A3 (en) 1999-12-21 2002-12-03 Upjohn Co Oxazolidinones having a sulfoximine functionality and their use as antimicrobial agents
AU2001253113B2 (en) 2000-04-20 2005-02-03 Pharmacia & Upjohn Company Use of thioamide oxazolidinones for the treatment of bone resorption and osteoporosis
ATE301474T1 (de) 2000-06-30 2005-08-15 Pharmacia & Upjohn Co Llc Zusammensetzungen zur behandlung baktrieller infektionen, welche ein oxazolidinonderivat, sulbactam und ampicillin enthalten
GB0017225D0 (en) 2000-07-14 2000-08-30 Really Useful Products Limited Container
DE10034627A1 (de) 2000-07-17 2002-01-31 Bayer Ag Aryl-substituierte Oxazolidinone mit Cytokin inhibitorischer Wirkung
HUP0302918A2 (hu) 2000-07-17 2003-12-29 Ranbaxy Laboratories Limited Mikrobaellenes oxazolidinonszármazékok és a vegyületeket tartalmazó gyógyászati készítmények és eljárás a vegyületek előállítására
DE60144522D1 (de) 2000-08-24 2011-06-09 Sirf Tech Inc Vorrichtung zur reduzierung von autokorrelation und kreuzkorrelation bei schwachen cdma-signalen
PE20020578A1 (es) 2000-10-10 2002-08-14 Upjohn Co Una composicion de antibiotico topico para el tratamiento de infecciones oculares
US20030008012A1 (en) 2001-02-05 2003-01-09 Pena Lorraine E. Composition for rectal delivery of an oxazolidinone antibacterial drug
DE10105989A1 (de) 2001-02-09 2002-08-14 Bayer Ag Substituierte Oxazolidinone und ihre Verwendung
ES2268011T3 (es) 2001-04-07 2007-03-16 Astrazeneca Ab Oxazolidinonas que contienen un grupo sulfonimida como antibioticos.
GB0108793D0 (en) 2001-04-07 2001-05-30 Astrazeneca Ab Chemical compounds
EP1409464A4 (en) 2001-07-16 2005-11-02 Ranbaxy Lab Ltd OXAZOLIDINONE DERIVATIVES AS POTENTIAL ANTIMICROBIALS
US6956040B2 (en) 2001-07-16 2005-10-18 Ranbaxy Laboratories Limited Oxazolidinone piperazinyl derivatives as potential antimicrobials
TW200302095A (en) 2002-01-25 2003-08-01 Upjohn Co Oxazolidinone cotherapy
TW200400055A (en) 2002-02-22 2004-01-01 Pharmacia Corp Ophthalmic formulation with novel gum composition
WO2003072141A1 (en) 2002-02-22 2003-09-04 Pharmacia Corporation Ophthalmic antibiotic drug formulations containing a cyclodextrin compound and cetyl pyridinium chloride
AR038536A1 (es) 2002-02-25 2005-01-19 Upjohn Co N-aril-2-oxazolidinona-5- carboxamidas y sus derivados
KR20040086465A (ko) 2002-02-28 2004-10-08 아스트라제네카 아베 화합물
AU2003207340A1 (en) 2002-02-28 2003-09-09 Astrazeneca Ab 3-cyclyl-5-(nitrogen-containing 5-membered ring) methyl-oxazolidinone derivatives and their use as antibacterial agents
EP1490059A1 (en) 2002-03-29 2004-12-29 Pharmacia & Upjohn Company LLC Parenteral, intravenous, and oral administration of oxazolidinones for treating diabetic foot infections
AU2003224345A1 (en) 2002-04-30 2003-11-17 Orchid Chemicals & Pharmaceuticals Antibacterial agents
TW200403240A (en) 2002-06-28 2004-03-01 Upjohn Co Difluorothioacetamides of oxazolidinones as antibacterial agents
WO2004009587A1 (en) 2002-07-22 2004-01-29 Orchid Chemicals & Pharmaceuticals Ltd Oxazolidinone derivatives as antibacterial agents
EA200500283A1 (ru) 2002-07-29 2005-08-25 Рэнбакси Лабораториз Лимитед Производные оксазолидинона как противомикробные средства
AU2003253141A1 (en) 2002-08-22 2004-03-11 Orchid Chemicals And Pharmaceuticals Ltd Novel antibacterial agents

Also Published As

Publication number Publication date
DK1899331T3 (da) 2010-03-08
JP2008544979A (ja) 2008-12-11
ES2335307T3 (es) 2010-03-24
DE602006010702D1 (de) 2010-01-07
WO2007000644A1 (en) 2007-01-04
CA2610978A1 (en) 2007-01-04
EP1899331B1 (en) 2009-11-25
EP1899331A1 (en) 2008-03-19

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Legal Events

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RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties