ATE425161T1 - Mercaptoimidazole als ccr2-rezeptorantagonisten - Google Patents

Mercaptoimidazole als ccr2-rezeptorantagonisten

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Publication number
ATE425161T1
ATE425161T1 AT05755042T AT05755042T ATE425161T1 AT E425161 T1 ATE425161 T1 AT E425161T1 AT 05755042 T AT05755042 T AT 05755042T AT 05755042 T AT05755042 T AT 05755042T AT E425161 T1 ATE425161 T1 AT E425161T1
Authority
AT
Austria
Prior art keywords
mercaptoimidazole
receptor antagonists
ccr2 receptor
ccr2
antagonists
Prior art date
Application number
AT05755042T
Other languages
English (en)
Inventor
Gustaaf Maria Boeckx
Lommen Guy R E Van
Julien G P Doyon
Erwin Coesemans
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34957884&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE425161(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Application granted granted Critical
Publication of ATE425161T1 publication Critical patent/ATE425161T1/de

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    • C07C211/01—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms
    • C07C211/26—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an unsaturated carbon skeleton containing at least one six-membered aromatic ring
    • C07C211/29—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an unsaturated carbon skeleton containing at least one six-membered aromatic ring the carbon skeleton being further substituted by halogen atoms or by nitro or nitroso groups
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    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/84—Sulfur atoms
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
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    • A61K31/4245—Oxadiazoles
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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AT05755042T 2004-05-26 2005-05-24 Mercaptoimidazole als ccr2-rezeptorantagonisten ATE425161T1 (de)

Applications Claiming Priority (1)

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EP2004050933 2004-05-26

Publications (1)

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ATE425161T1 true ATE425161T1 (de) 2009-03-15

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US (1) US20070249691A1 (de)
EP (1) EP1753758B1 (de)
JP (1) JP2008500310A (de)
KR (1) KR20070020070A (de)
CN (1) CN1956980A (de)
AR (1) AR049386A1 (de)
AT (1) ATE425161T1 (de)
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ATE411989T1 (de) * 2004-05-26 2008-11-15 Janssen Pharmaceutica Nv Mercaptoimidazole als ccr2-rezeptorantagonisten
ES2764840T3 (es) 2015-01-28 2020-06-04 Univ Bordeaux Uso de plerixafor para tratar y/o prevenir exacerbaciones agudas de la enfermedad pulmonar obstructiva crónica
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JP2021534101A (ja) 2018-08-09 2021-12-09 ヴェルソー セラピューティクス， インコーポレイテッド Ｃｃｒ２及びｃｓｆ１ｒを標的とするためのオリゴヌクレオチド組成物ならびにその使用
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FR1487326A (fr) 1966-01-18 1967-07-07 Clin Byla Ets Dérivés imidazoliques et leur préparation
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US4770689A (en) * 1986-03-10 1988-09-13 Janssen Pharmaceutica N.V. Herbicidal imidazole-5-carboxylic acid derivatives
DE10107683A1 (de) 2001-02-19 2002-08-29 Merckle Gmbh Chem Pharm Fabrik 2-Thio-substituierte Imidazolderivate und ihre Verwendung in der Pharmazie
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PA8634401A1 (es) 2006-05-16
WO2005118578A1 (en) 2005-12-15
IL179518A0 (en) 2007-05-15
CN1956980A (zh) 2007-05-02
AR049386A1 (es) 2006-07-26
EA200602193A1 (ru) 2007-04-27
JP2008500310A (ja) 2008-01-10
AU2005250156A1 (en) 2005-12-15
MXPA06013764A (es) 2007-02-08
DE602005013216D1 (de) 2009-04-23
US20070249691A1 (en) 2007-10-25
TW200606154A (en) 2006-02-16
ZA200609846B (en) 2008-07-30
NO20066011L (no) 2007-02-23
EP1753758B1 (de) 2009-03-11
EP1753758A1 (de) 2007-02-21
CA2566187A1 (en) 2005-12-15
MY140571A (en) 2009-12-31
KR20070020070A (ko) 2007-02-16

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