ATE37552T1 - Peptid- und pseudopeptid-derivate. - Google Patents
Peptid- und pseudopeptid-derivate.Info
- Publication number
- ATE37552T1 ATE37552T1 AT83304507T AT83304507T ATE37552T1 AT E37552 T1 ATE37552 T1 AT E37552T1 AT 83304507 T AT83304507 T AT 83304507T AT 83304507 T AT83304507 T AT 83304507T AT E37552 T1 ATE37552 T1 AT E37552T1
- Authority
- AT
- Austria
- Prior art keywords
- sup
- compounds
- radical
- alkyl
- stands
- Prior art date
Links
- 108090000765 processed proteins & peptides Proteins 0.000 title abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 4
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- 125000004432 carbon atom Chemical group C* 0.000 abstract 2
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- 101100244562 Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22644 / CIP 104116 / JCM 14847 / LMG 12228 / 1C / PRS 101 / PAO1) oprD gene Proteins 0.000 abstract 1
- 125000000539 amino acid group Chemical group 0.000 abstract 1
- 150000001413 amino acids Chemical class 0.000 abstract 1
- 108700023159 delta Opioid Receptors Proteins 0.000 abstract 1
- 102000048124 delta Opioid Receptors Human genes 0.000 abstract 1
- 239000003085 diluting agent Substances 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 229940127240 opiate Drugs 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 239000002464 receptor antagonist Substances 0.000 abstract 1
- 229940044551 receptor antagonist Drugs 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/665—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
- C07K14/70—Enkephalins
- C07K14/702—Enkephalins with at least 1 amino acid in D-form
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Genetics & Genomics (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Neurology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biomedical Technology (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Neurosurgery (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Molecular Biology (AREA)
- Toxicology (AREA)
- Zoology (AREA)
- Gastroenterology & Hepatology (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Animal Behavior & Ethology (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB8229723 | 1982-10-18 | ||
| EP83304507A EP0109142B1 (de) | 1982-10-18 | 1983-08-04 | Peptid- und Pseudopeptid-Derivate |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE37552T1 true ATE37552T1 (de) | 1988-10-15 |
Family
ID=10533671
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT83304507T ATE37552T1 (de) | 1982-10-18 | 1983-08-04 | Peptid- und pseudopeptid-derivate. |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US4474767A (de) |
| EP (1) | EP0109142B1 (de) |
| JP (1) | JPS5973551A (de) |
| AT (1) | ATE37552T1 (de) |
| DE (1) | DE3378121D1 (de) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3711335A1 (de) * | 1987-04-03 | 1988-10-20 | Merck Patent Gmbh | Aminosaeurederivate |
| US5877277A (en) | 1987-09-24 | 1999-03-02 | Biomeasure, Inc. | Octapeptide bombesin analogs |
| US5084555A (en) * | 1989-08-21 | 1992-01-28 | The Administrators Of The Tulane Educational Fund | An octapeptide bombesin analog |
| US5162497A (en) * | 1987-09-24 | 1992-11-10 | The Administrators Of The Tulane Educational Fund | Bradykinin analogs with non-peptide bond |
| US6218364B1 (en) * | 1988-06-20 | 2001-04-17 | Scott L. Harbeson | Fluorinated neurokinin A antagonists |
| US5830863A (en) * | 1988-06-20 | 1998-11-03 | Merrell Pharmaceuticals Inc. | Neurokinin A antagonists |
| US5767236A (en) * | 1990-05-09 | 1998-06-16 | Biomeasure, Inc. | Linear therapeutic peptides |
| WO2012158962A2 (en) * | 2011-05-18 | 2012-11-22 | Eumederis Pharmaceuticals, Inc. | Improved peptide pharmaceuticals |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1577115A (en) * | 1976-07-27 | 1980-10-22 | Reckitt & Colmann Prod Ltd | Container closure units |
| US4254106A (en) * | 1976-01-26 | 1981-03-03 | Burroughs Wellcome Co. | Biologically active amides |
| US4322342A (en) * | 1977-06-20 | 1982-03-30 | Eli Lilly And Company | Analgesic compounds |
| GB1604850A (en) * | 1977-11-24 | 1981-12-16 | Wellcome Found | Biologically active peptides |
| US4331593A (en) * | 1977-10-03 | 1982-05-25 | Smithwick Jr Edward L | Analgesic compounds |
| US4221682A (en) * | 1979-08-06 | 1980-09-09 | American Home Products Corporation | Tetrapeptides having analgesic activity |
| US4320051A (en) * | 1979-12-26 | 1982-03-16 | American Home Products Corporation | Analgesic tripeptide amides |
-
1983
- 1983-08-04 DE DE8383304507T patent/DE3378121D1/de not_active Expired
- 1983-08-04 EP EP83304507A patent/EP0109142B1/de not_active Expired
- 1983-08-04 AT AT83304507T patent/ATE37552T1/de not_active IP Right Cessation
- 1983-08-16 US US06/523,773 patent/US4474767A/en not_active Expired - Lifetime
- 1983-08-29 JP JP58156550A patent/JPS5973551A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| JPS5973551A (ja) | 1984-04-25 |
| EP0109142A3 (en) | 1985-08-21 |
| DE3378121D1 (de) | 1988-11-03 |
| EP0109142B1 (de) | 1988-09-28 |
| EP0109142A2 (de) | 1984-05-23 |
| US4474767A (en) | 1984-10-02 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification | ||
| REN | Ceased due to non-payment of the annual fee |