ATE352295T1 - Verwendung von quinazolinen zur behandlung von t- zell vermittelten krankheiten - Google Patents
Verwendung von quinazolinen zur behandlung von t- zell vermittelten krankheitenInfo
- Publication number
- ATE352295T1 ATE352295T1 AT02777571T AT02777571T ATE352295T1 AT E352295 T1 ATE352295 T1 AT E352295T1 AT 02777571 T AT02777571 T AT 02777571T AT 02777571 T AT02777571 T AT 02777571T AT E352295 T1 ATE352295 T1 AT E352295T1
- Authority
- AT
- Austria
- Prior art keywords
- sub
- mediated diseases
- cell
- quinazolines
- treat
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Immunology (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Transplantation (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0128109.6A GB0128109D0 (en) | 2001-11-23 | 2001-11-23 | Therapeutic use |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE352295T1 true ATE352295T1 (de) | 2007-02-15 |
Family
ID=9926330
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT02777571T ATE352295T1 (de) | 2001-11-23 | 2002-11-20 | Verwendung von quinazolinen zur behandlung von t- zell vermittelten krankheiten |
Country Status (7)
Country | Link |
---|---|
US (1) | US7157467B2 (de) |
EP (1) | EP1453492B1 (de) |
AT (1) | ATE352295T1 (de) |
AU (1) | AU2002339194A1 (de) |
DE (1) | DE60217904T2 (de) |
GB (1) | GB0128109D0 (de) |
WO (1) | WO2003045364A2 (de) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU2002217999A1 (en) | 2000-11-01 | 2002-05-15 | Cor Therapeutics, Inc. | Process for the production of 4-quinazolinylpiperazin-1-carboxylic acid phenylamides |
US6924285B2 (en) | 2002-03-30 | 2005-08-02 | Boehringer Ingelheim Pharma Gmbh & Co. | Bicyclic heterocyclic compounds, pharmaceutical compositions containing these compounds, their use and process for preparing them |
JP2005536486A (ja) * | 2002-07-09 | 2005-12-02 | アストラゼネカ アクチボラグ | 癌の処置に使用するためのキナゾリン誘導体 |
GB0317665D0 (en) | 2003-07-29 | 2003-09-03 | Astrazeneca Ab | Qinazoline derivatives |
EP1921070A1 (de) | 2006-11-10 | 2008-05-14 | Boehringer Ingelheim Pharma GmbH & Co. KG | Bicyclische Heterocyclen, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstelllung |
WO2008095847A1 (de) | 2007-02-06 | 2008-08-14 | Boehringer Ingelheim International Gmbh | Bicyclische heterocyclen, diese verbindungen enthaltende arzneimittel, deren verwendung und verfahren zu ihrer herstellung |
EP2245026B1 (de) | 2008-02-07 | 2012-08-01 | Boehringer Ingelheim International GmbH | Spirocyclische heterocyclen, diese verbindungen enthaltende arzneimittel, deren verwendung und verfahren zu ihrer herstellung |
JP5739802B2 (ja) | 2008-05-13 | 2015-06-24 | アストラゼネカ アクチボラグ | 4−(3−クロロ−2−フルオロアニリノ)−7−メトキシ−6−{[1−(n−メチルカルバモイルメチル)ピペリジン−4−イル]オキシ}キナゾリンのフマル酸塩 |
EP2313397B1 (de) | 2008-08-08 | 2016-04-20 | Boehringer Ingelheim International GmbH | Cyclohexyloxy-substituierte heterocyclen, diese verbindungen enthaltende arzneimittel, deren verwendung und verfahren zu ihrer herstellung |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6046206A (en) * | 1995-06-07 | 2000-04-04 | Cell Pathways, Inc. | Method of treating a patient having a precancerous lesions with amide quinazoline derivatives |
GB9718972D0 (en) | 1996-09-25 | 1997-11-12 | Zeneca Ltd | Chemical compounds |
JPH11209350A (ja) | 1998-01-26 | 1999-08-03 | Eisai Co Ltd | 含窒素複素環誘導体およびその医薬 |
PL205557B1 (pl) * | 1999-02-10 | 2010-05-31 | Astrazeneca Ab | Pochodne indolu |
RU2267489C2 (ru) * | 2000-08-21 | 2006-01-10 | Астразенека Аб | Производные хиназолина, способ их получения и фармацевтическая композиция |
-
2001
- 2001-11-23 GB GBGB0128109.6A patent/GB0128109D0/en not_active Ceased
-
2002
- 2002-11-20 US US10/496,464 patent/US7157467B2/en not_active Expired - Fee Related
- 2002-11-20 AU AU2002339194A patent/AU2002339194A1/en not_active Abandoned
- 2002-11-20 EP EP02777571A patent/EP1453492B1/de not_active Expired - Lifetime
- 2002-11-20 DE DE60217904T patent/DE60217904T2/de not_active Expired - Fee Related
- 2002-11-20 AT AT02777571T patent/ATE352295T1/de not_active IP Right Cessation
- 2002-11-20 WO PCT/GB2002/005217 patent/WO2003045364A2/en active IP Right Grant
Also Published As
Publication number | Publication date |
---|---|
US20050014773A1 (en) | 2005-01-20 |
US7157467B2 (en) | 2007-01-02 |
EP1453492B1 (de) | 2007-01-24 |
GB0128109D0 (en) | 2002-01-16 |
DE60217904T2 (de) | 2007-11-15 |
WO2003045364A2 (en) | 2003-06-05 |
EP1453492A2 (de) | 2004-09-08 |
DE60217904D1 (de) | 2007-03-15 |
WO2003045364A3 (en) | 2003-08-28 |
AU2002339194A1 (en) | 2003-06-10 |
AU2002339194A8 (en) | 2003-06-10 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |