ATE33138T1 - Verfahren zur herstellung von 5-azaindol und zwischenprodukte. - Google Patents
Verfahren zur herstellung von 5-azaindol und zwischenprodukte.Info
- Publication number
- ATE33138T1 ATE33138T1 AT85870072T AT85870072T ATE33138T1 AT E33138 T1 ATE33138 T1 AT E33138T1 AT 85870072 T AT85870072 T AT 85870072T AT 85870072 T AT85870072 T AT 85870072T AT E33138 T1 ATE33138 T1 AT E33138T1
- Authority
- AT
- Austria
- Prior art keywords
- group
- azaindol
- preparation
- intermediate products
- enamine
- Prior art date
Links
- SRSKXJVMVSSSHB-UHFFFAOYSA-N 1h-pyrrolo[3,2-c]pyridine Chemical compound N1=CC=C2NC=CC2=C1 SRSKXJVMVSSSHB-UHFFFAOYSA-N 0.000 title abstract 3
- 239000013067 intermediate product Substances 0.000 title 1
- 150000002081 enamines Chemical class 0.000 abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 2
- SSOURMYKACOBIV-UHFFFAOYSA-N 3-methyl-4-nitro-1-oxidopyridin-1-ium Chemical compound CC1=C[N+]([O-])=CC=C1[N+]([O-])=O SSOURMYKACOBIV-UHFFFAOYSA-N 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- -1 morpholino, piperidino Chemical group 0.000 abstract 1
- 125000002112 pyrrolidino group Chemical group [*]N1C([H])([H])C([H])([H])C([H])([H])C1([H])[H] 0.000 abstract 1
- 238000007363 ring formation reaction Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/89—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to the ring nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Design And Manufacture Of Integrated Circuits (AREA)
- Thin Film Transistor (AREA)
- Crystals, And After-Treatments Of Crystals (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR8408275A FR2564836B1 (fr) | 1984-05-25 | 1984-05-25 | Procede de preparation de l'aza-5 indole et compose obtenu par ce procede |
| EP85870072A EP0165225B1 (de) | 1984-05-25 | 1985-05-23 | Verfahren zur Herstellung von 5-Azaindol und Zwischenprodukte |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE33138T1 true ATE33138T1 (de) | 1988-04-15 |
Family
ID=9304427
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT85870072T ATE33138T1 (de) | 1984-05-25 | 1985-05-23 | Verfahren zur herstellung von 5-azaindol und zwischenprodukte. |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US4625033A (de) |
| EP (1) | EP0165225B1 (de) |
| JP (1) | JPS60258181A (de) |
| AT (1) | ATE33138T1 (de) |
| CA (1) | CA1259311A (de) |
| DE (1) | DE3561947D1 (de) |
| ES (1) | ES8604217A1 (de) |
| FR (1) | FR2564836B1 (de) |
| PT (1) | PT80485B (de) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN1321118C (zh) * | 2005-08-02 | 2007-06-13 | 浙江大学 | 5－氮杂吲哚的制备方法 |
| CN103980273A (zh) * | 2014-06-03 | 2014-08-13 | 重庆邮电大学 | 5-氮杂吲哚的制备方法 |
| CN105646486B (zh) * | 2016-03-01 | 2017-10-13 | 苏州艾缇克药物化学有限公司 | 一种5‑氮杂吲哚的合成方法 |
-
1984
- 1984-05-25 FR FR8408275A patent/FR2564836B1/fr not_active Expired
-
1985
- 1985-05-13 JP JP60102500A patent/JPS60258181A/ja active Pending
- 1985-05-17 PT PT80485A patent/PT80485B/pt not_active IP Right Cessation
- 1985-05-23 DE DE8585870072T patent/DE3561947D1/de not_active Expired
- 1985-05-23 AT AT85870072T patent/ATE33138T1/de not_active IP Right Cessation
- 1985-05-23 EP EP85870072A patent/EP0165225B1/de not_active Expired
- 1985-05-24 ES ES543461A patent/ES8604217A1/es not_active Expired
- 1985-05-24 CA CA000482288A patent/CA1259311A/en not_active Expired
- 1985-05-28 US US06/738,438 patent/US4625033A/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| FR2564836A1 (fr) | 1985-11-29 |
| EP0165225B1 (de) | 1988-03-23 |
| EP0165225A1 (de) | 1985-12-18 |
| ES8604217A1 (es) | 1986-01-16 |
| DE3561947D1 (en) | 1988-04-28 |
| FR2564836B1 (fr) | 1986-09-26 |
| CA1259311A (en) | 1989-09-12 |
| JPS60258181A (ja) | 1985-12-20 |
| PT80485A (en) | 1985-06-01 |
| ES543461A0 (es) | 1986-01-16 |
| US4625033A (en) | 1986-11-25 |
| PT80485B (en) | 1987-04-21 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification | ||
| REN | Ceased due to non-payment of the annual fee |