DE3561947D1 - Process for the preparation of 5-azaindole and intermediates - Google Patents

Process for the preparation of 5-azaindole and intermediates

Info

Publication number
DE3561947D1
DE3561947D1 DE8585870072T DE3561947T DE3561947D1 DE 3561947 D1 DE3561947 D1 DE 3561947D1 DE 8585870072 T DE8585870072 T DE 8585870072T DE 3561947 T DE3561947 T DE 3561947T DE 3561947 D1 DE3561947 D1 DE 3561947D1
Authority
DE
Germany
Prior art keywords
group
azaindole
intermediates
preparation
enamine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
DE8585870072T
Other languages
English (en)
Inventor
Jean-Robert Dormoy
Alain Heymes
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi SA
Original Assignee
Sanofi SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi SA filed Critical Sanofi SA
Application granted granted Critical
Publication of DE3561947D1 publication Critical patent/DE3561947D1/de
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/89—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to the ring nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Design And Manufacture Of Integrated Circuits (AREA)
  • Thin Film Transistor (AREA)
  • Crystals, And After-Treatments Of Crystals (AREA)
DE8585870072T 1984-05-25 1985-05-23 Process for the preparation of 5-azaindole and intermediates Expired DE3561947D1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8408275A FR2564836B1 (fr) 1984-05-25 1984-05-25 Procede de preparation de l'aza-5 indole et compose obtenu par ce procede

Publications (1)

Publication Number Publication Date
DE3561947D1 true DE3561947D1 (en) 1988-04-28

Family

ID=9304427

Family Applications (1)

Application Number Title Priority Date Filing Date
DE8585870072T Expired DE3561947D1 (en) 1984-05-25 1985-05-23 Process for the preparation of 5-azaindole and intermediates

Country Status (9)

Country Link
US (1) US4625033A (de)
EP (1) EP0165225B1 (de)
JP (1) JPS60258181A (de)
AT (1) ATE33138T1 (de)
CA (1) CA1259311A (de)
DE (1) DE3561947D1 (de)
ES (1) ES8604217A1 (de)
FR (1) FR2564836B1 (de)
PT (1) PT80485B (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1321118C (zh) * 2005-08-02 2007-06-13 浙江大学 5－氮杂吲哚的制备方法
CN103980273A (zh) * 2014-06-03 2014-08-13 重庆邮电大学 5-氮杂吲哚的制备方法
CN105646486B (zh) * 2016-03-01 2017-10-13 苏州艾缇克药物化学有限公司 一种5‑氮杂吲哚的合成方法

Also Published As

Publication number Publication date
US4625033A (en) 1986-11-25
JPS60258181A (ja) 1985-12-20
ES543461A0 (es) 1986-01-16
CA1259311A (en) 1989-09-12
EP0165225B1 (de) 1988-03-23
ES8604217A1 (es) 1986-01-16
PT80485B (en) 1987-04-21
FR2564836B1 (fr) 1986-09-26
PT80485A (en) 1985-06-01
EP0165225A1 (de) 1985-12-18
FR2564836A1 (fr) 1985-11-29
ATE33138T1 (de) 1988-04-15

Similar Documents

Publication Publication Date Title
ES8400422A1 (es) "procedimiento de preparacion de eteres triciclicos, asi como de sus sales de adicion con un acido mineral u organico terapeuticamente compatible".
CS725686A3 (en) Process for preparing novel imidazole derivatives
PT73601A (en) Process for the preparation of piperidilydene derivatives having pharmaceutical properties
PT77370B (en) Process for preparing new pyrazolo <3,4-b> piridine derivatives and pharmaceutical preparations containing the same
HUT38340A (en) Process for producing benzyl-phtalazinone derivatives and pharmaceutical compositions containing them
HUT38927A (en) Process for producing 5-alkyl-1-phenyl-2-/piperazino-alkyl/-pyrazolin-3-one derivatives
YU182581A (en) Process for preparing new 5,10-dihydro-11h-dibenzo-(b,e)(1,4)diazepine-11-ones substituted in position 5
DE3561947D1 (en) Process for the preparation of 5-azaindole and intermediates
HUT38945A (en) Process for production of derivatives of furo /3,2-c/ piridin and medical preparatives containing thereof
CA1274825C (en) AMIDINES, AND THEIR MANUFACTURE
ES8406067A1 (es) Un procedimiento de preparacion de un nuevo derivado de (2,4,6-trimetoxifenil)-(3-piperidinopropil)cetona
DE3065305D1 (en) Spiro-derivatives, process for their preparation and medicines containing them
PL238869A1 (en) Process for preparing novel 1-furyl-3,4-dihydroisoquinolines
DE3378980D1 (en) Benzazepine derivatives, process for their preparation and their use as pharmaceutical compounds
PH19310A (en) 1,2-fused 1,4-benzodiazepine compounds,process for their preparation and compositions containing them
HUT48599A (en) Process for producing 2-aminoisoquinoline derivatives and pharmaceutical compositions comprising the compounds
ES8506679A2 (es) Mejoras en el objeto de la patente de invencion n 514.340 que se refiere a: procedimiento de obtencion de nuevos derivados de piperazina
PT71895A (en) Process for the preparation of nb-quaternary 10-bromosanduicine and 10-bromoisosanduicine derivatives

Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8339 Ceased/non-payment of the annual fee