ATE242333T1 - Verfahren zur herstellung von fexofenadin - Google Patents
Verfahren zur herstellung von fexofenadinInfo
- Publication number
- ATE242333T1 ATE242333T1 AT99909036T AT99909036T ATE242333T1 AT E242333 T1 ATE242333 T1 AT E242333T1 AT 99909036 T AT99909036 T AT 99909036T AT 99909036 T AT99909036 T AT 99909036T AT E242333 T1 ATE242333 T1 AT E242333T1
- Authority
- AT
- Austria
- Prior art keywords
- fexofenadine
- producing
- producing fexofenadine
- Prior art date
Links
- RWTNPBWLLIMQHL-UHFFFAOYSA-N fexofenadine Chemical compound C1=CC(C(C)(C(O)=O)C)=CC=C1C(O)CCCN1CCC(C(O)(C=2C=CC=CC=2)C=2C=CC=CC=2)CC1 RWTNPBWLLIMQHL-UHFFFAOYSA-N 0.000 title 1
- 229960003592 fexofenadine Drugs 0.000 title 1
- 238000004519 manufacturing process Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/70—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
- C07F9/576—Six-membered rings
- C07F9/59—Hydrogenated pyridine rings
-
- C—CHEMISTRY; METALLURGY
- C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
- C12P—FERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
- C12P17/00—Preparation of heterocyclic carbon compounds with only O, N, S, Se or Te as ring hetero atoms
- C12P17/10—Nitrogen as only ring hetero atom
- C12P17/12—Nitrogen as only ring hetero atom containing a six-membered hetero ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Zoology (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Biochemistry (AREA)
- Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Microbiology (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Engineering & Computer Science (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Micro-Organisms Or Cultivation Processes Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9803349A FR2776302B1 (fr) | 1998-03-19 | 1998-03-19 | Nouveau procede de preparation de la fexofenadine |
| PCT/FR1999/000625 WO1999047693A1 (fr) | 1998-03-19 | 1999-03-18 | Nouveau procede de preparation de la fexofenadine |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE242333T1 true ATE242333T1 (de) | 2003-06-15 |
Family
ID=9524214
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT99909036T ATE242333T1 (de) | 1998-03-19 | 1999-03-18 | Verfahren zur herstellung von fexofenadin |
Country Status (15)
| Country | Link |
|---|---|
| US (2) | US6558931B1 (de) |
| EP (1) | EP1062358B1 (de) |
| JP (1) | JP4291511B2 (de) |
| AR (1) | AR014738A1 (de) |
| AT (1) | ATE242333T1 (de) |
| AU (1) | AU2842799A (de) |
| DE (1) | DE69908569T2 (de) |
| DK (1) | DK1062358T3 (de) |
| DZ (1) | DZ2746A1 (de) |
| ES (1) | ES2196783T3 (de) |
| FR (1) | FR2776302B1 (de) |
| MA (1) | MA26615A1 (de) |
| PT (1) | PT1062358E (de) |
| TN (1) | TNSN99042A1 (de) |
| WO (1) | WO1999047693A1 (de) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2776302B1 (fr) * | 1998-03-19 | 2002-04-12 | Hoechst Marion Roussel Inc | Nouveau procede de preparation de la fexofenadine |
| GB0013368D0 (en) * | 2000-05-31 | 2000-07-26 | Pfizer Ltd | Enzymatic oxidations |
| US6610518B2 (en) | 2000-05-31 | 2003-08-26 | Pfizer Inc. | Enzymatic oxidations |
| US6613906B1 (en) * | 2000-06-06 | 2003-09-02 | Geneva Pharmaceuticals, Inc. | Crystal modification |
| GB0018691D0 (en) * | 2000-07-28 | 2000-09-20 | Rolabo Sl | Process |
| US6613907B2 (en) | 2000-11-08 | 2003-09-02 | Amr Technology, Inc. | Process for the production of piperidine derivatives with microorganisms |
| AU2003209673B2 (en) * | 2002-03-08 | 2007-10-18 | M/S. Ind-Swift Limited | Tasteless directly compressible fast-dissolving complexes and pharmaceutical formulations thereof |
| US20090076080A1 (en) * | 2007-09-19 | 2009-03-19 | Protia, Llc | Deuterium-enriched fexofenadine |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6147216A (en) | 1993-06-25 | 2000-11-14 | Merrell Pharmaceuticals Inc. | Intermediates useful for the preparation of antihistaminic piperidine derivatives |
| HU226037B1 (en) | 1993-06-25 | 2008-03-28 | Aventis Inc | Process for producing antihistaminic 4-diphenylmethyl/diphenylmethoxy piperidine derivatives and novel intermediates |
| ES2216191T3 (es) * | 1997-03-11 | 2004-10-16 | Aventis Pharmaceuticals Inc. | Procedimiento para preparar acido 4-(4-(hidroxidifenil)-1-piperidinil)-1-hidroxibutil)-alfa,alfa-dimetilfenilacetico y derivados fosforilados. |
| FR2776302B1 (fr) * | 1998-03-19 | 2002-04-12 | Hoechst Marion Roussel Inc | Nouveau procede de preparation de la fexofenadine |
-
1998
- 1998-03-19 FR FR9803349A patent/FR2776302B1/fr not_active Expired - Lifetime
-
1999
- 1999-03-17 DZ DZ990047A patent/DZ2746A1/xx active
- 1999-03-17 AR ARP990101165A patent/AR014738A1/es unknown
- 1999-03-17 MA MA25501A patent/MA26615A1/fr unknown
- 1999-03-18 WO PCT/FR1999/000625 patent/WO1999047693A1/fr active IP Right Grant
- 1999-03-18 AU AU28427/99A patent/AU2842799A/en not_active Abandoned
- 1999-03-18 US US09/646,517 patent/US6558931B1/en not_active Expired - Lifetime
- 1999-03-18 TN TNTNSN99042A patent/TNSN99042A1/fr unknown
- 1999-03-18 DE DE69908569T patent/DE69908569T2/de not_active Expired - Lifetime
- 1999-03-18 PT PT99909036T patent/PT1062358E/pt unknown
- 1999-03-18 EP EP99909036A patent/EP1062358B1/de not_active Expired - Lifetime
- 1999-03-18 ES ES99909036T patent/ES2196783T3/es not_active Expired - Lifetime
- 1999-03-18 JP JP2000536876A patent/JP4291511B2/ja not_active Expired - Lifetime
- 1999-03-18 DK DK99909036T patent/DK1062358T3/da active
- 1999-03-18 AT AT99909036T patent/ATE242333T1/de active
-
2003
- 2003-03-20 US US10/392,699 patent/US7241601B2/en not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| JP2002506653A (ja) | 2002-03-05 |
| EP1062358A1 (de) | 2000-12-27 |
| PT1062358E (pt) | 2003-10-31 |
| AR014738A1 (es) | 2001-03-28 |
| EP1062358B1 (de) | 2003-06-04 |
| AU2842799A (en) | 1999-10-11 |
| FR2776302B1 (fr) | 2002-04-12 |
| MA26615A1 (fr) | 2004-12-20 |
| ES2196783T3 (es) | 2003-12-16 |
| US6558931B1 (en) | 2003-05-06 |
| DK1062358T3 (da) | 2003-09-29 |
| FR2776302A1 (fr) | 1999-09-24 |
| DE69908569T2 (de) | 2004-05-13 |
| JP4291511B2 (ja) | 2009-07-08 |
| TNSN99042A1 (fr) | 2005-11-10 |
| US7241601B2 (en) | 2007-07-10 |
| DZ2746A1 (fr) | 2003-09-08 |
| DE69908569D1 (de) | 2003-07-10 |
| WO1999047693A1 (fr) | 1999-09-23 |
| US20060019358A1 (en) | 2006-01-26 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification |
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