ATE223419T1 - Kondensierte thiadiazolderivate, verfahren zu ihrer herstellung und deren verwendung - Google Patents

Kondensierte thiadiazolderivate, verfahren zu ihrer herstellung und deren verwendung

Info

Publication number
ATE223419T1
ATE223419T1 AT93104939T AT93104939T ATE223419T1 AT E223419 T1 ATE223419 T1 AT E223419T1 AT 93104939 T AT93104939 T AT 93104939T AT 93104939 T AT93104939 T AT 93104939T AT E223419 T1 ATE223419 T1 AT E223419T1
Authority
AT
Austria
Prior art keywords
ring
production
substituted
thiadiazole derivatives
pharmaceutically acceptable
Prior art date
Application number
AT93104939T
Other languages
English (en)
Inventor
Takashi Sohda
Zen-Ichi Terashita
Yu Momose
Yukio Fujisawa
Junji Mizoguchi
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Application granted granted Critical
Publication of ATE223419T1 publication Critical patent/ATE223419T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
AT93104939T 1992-03-25 1993-03-25 Kondensierte thiadiazolderivate, verfahren zu ihrer herstellung und deren verwendung ATE223419T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP6761592 1992-03-25
JP3087293 1993-02-19

Publications (1)

Publication Number Publication Date
ATE223419T1 true ATE223419T1 (de) 2002-09-15

Family

ID=26369305

Family Applications (1)

Application Number Title Priority Date Filing Date
AT93104939T ATE223419T1 (de) 1992-03-25 1993-03-25 Kondensierte thiadiazolderivate, verfahren zu ihrer herstellung und deren verwendung

Country Status (5)

Country Link
US (1) US5550138A (de)
EP (1) EP0562599B1 (de)
AT (1) ATE223419T1 (de)
CA (1) CA2092390A1 (de)
DE (1) DE69332259T2 (de)

Families Citing this family (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5767310A (en) * 1993-03-19 1998-06-16 Merck & Co., Inc. Phenoxyphenylacetic acid derivatives
US5686478A (en) * 1993-07-20 1997-11-11 Merck & Co. Inc. Endothelin antagonists
BR9407933A (pt) * 1993-11-01 1996-11-26 Japat Ltd Antagonistas de receptores de endotelina
US5559135A (en) * 1994-09-14 1996-09-24 Merck & Co., Inc. Endothelin antagonists bearing pyridyl amides
US5538991A (en) * 1994-09-14 1996-07-23 Merck & Co., Inc. Endothelin antagonists bearing 5-membered heterocyclic amides
US5830850A (en) * 1996-08-28 1998-11-03 Mount Sinai School Of Medicine Of The City Of New York Methods for the treatment of bone resorption disorders, including osteoporosis
US5691153A (en) * 1996-09-06 1997-11-25 Creighton University Genetic markers to detect high bone mass
US5916887A (en) * 1996-09-23 1999-06-29 National Research Council Of Canada 4-substituted-3-(2-amino-2-cycloalkyl methyl)-acetamido azetidin-2-one derivatives as cysteine proteinase regulators
US6340683B1 (en) 1999-04-22 2002-01-22 Synaptic Pharmaceutical Corporation Selective NPY (Y5) antagonists (triazines)
PT1183245E (pt) * 1999-04-22 2007-07-12 Lundbeck & Co As H Antagonistas selectivos de npy (y5)
US6218408B1 (en) 1999-06-30 2001-04-17 Synaptic Pharmaceutical Corporation Selective NPY (Y5) antagonists (bicyclics)
US6989379B1 (en) 1999-04-22 2006-01-24 H. Lundbick A/S Selective NPY (Y5) antagonists
US6225330B1 (en) * 1999-06-30 2001-05-01 Synaptic Pharmaceutical Corporation Selective NPY (Y5) antagonists (tricyclics)
US6214853B1 (en) 1999-06-30 2001-04-10 Synaptic Pharmaceutical Corporation Selective NPY (Y5) antagonists (bicyclics)
DE60023141T2 (de) * 1999-06-30 2006-06-14 Lundbeck As Valby H Selektive npy (y5) antagonisten
US7273880B2 (en) * 1999-06-30 2007-09-25 H. Lunbeck A/S Selective NPY (Y5) antagonists
US6222040B1 (en) * 1999-06-30 2001-04-24 Synaptic Pharmaceutical Corporation Selective NPY (Y5) antagonists (tricyclics)
WO2004084830A2 (en) * 2003-03-21 2004-10-07 Buck Institute Method for treating alzheimer’s dementia
EP1632558A1 (de) * 2004-09-06 2006-03-08 The Procter & Gamble Zusammensetzung enthaltend ein kationisches Polymer, welches die Abscheidung auf Oberflächen erhöht
EP1981884B1 (de) * 2006-01-18 2012-06-13 Amgen, Inc Thiazolverbindungen als proteinkinase b (pkb)-inhibitoren
US20100022568A1 (en) * 2006-04-13 2010-01-28 Actelion Pharmaceeuticals Ltd. Endothelin receptor antagonists for early stage idiopathic pulmonary fibrosis
WO2009011871A2 (en) * 2007-07-17 2009-01-22 Amgen Inc. Thiadiazole modulators of pkb
WO2009011880A2 (en) 2007-07-17 2009-01-22 Amgen Inc. Heterocyclic modulators of pkb
US9079866B2 (en) 2013-02-04 2015-07-14 Janssen Pharmaceutica Nv Flap modulators
TWI644899B (zh) 2013-02-04 2018-12-21 健生藥品公司 Ｆｌａｐ調節劑

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS60246389A (ja) * 1984-05-22 1985-12-06 Nippon Soda Co Ltd ２−スルホニルイミノ−２Ｈ−１，２，４−チアジアゾロ〔２，３−ａ〕ピリジン誘導体及びその製造法
JPS6310795A (ja) * 1986-03-25 1988-01-18 Takeda Chem Ind Ltd 選択性除草化合物
JPS62263185A (ja) * 1986-05-07 1987-11-16 Nippon Soda Co Ltd チアジアゾロピリミ（トリア）ジン誘導体、その製造方法及び除草剤

Also Published As

Publication number Publication date
CA2092390A1 (en) 1993-09-26
EP0562599B1 (de) 2002-09-04
EP0562599A1 (de) 1993-09-29
US5550138A (en) 1996-08-27
DE69332259D1 (de) 2002-10-10
DE69332259T2 (de) 2003-07-31

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Legal Events

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RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties