ATE218568T1 - Hetero-biaryl-pyridochinazolinonderivate als antikrebsmittel - Google Patents

Hetero-biaryl-pyridochinazolinonderivate als antikrebsmittel

Info

Publication number
ATE218568T1
ATE218568T1 AT97948622T AT97948622T ATE218568T1 AT E218568 T1 ATE218568 T1 AT E218568T1 AT 97948622 T AT97948622 T AT 97948622T AT 97948622 T AT97948622 T AT 97948622T AT E218568 T1 ATE218568 T1 AT E218568T1
Authority
AT
Austria
Prior art keywords
pyridoquinazolinone
ch2ch2nh2
group
alkyl
biaryl
Prior art date
Application number
AT97948622T
Other languages
English (en)
Inventor
Michael Peter Trova
Nan Zhang
Original Assignee
American Cyanamid Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Cyanamid Co filed Critical American Cyanamid Co
Application granted granted Critical
Publication of ATE218568T1 publication Critical patent/ATE218568T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AT97948622T 1996-11-26 1997-11-24 Hetero-biaryl-pyridochinazolinonderivate als antikrebsmittel ATE218568T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US75584596A 1996-11-26 1996-11-26
PCT/US1997/022502 WO1998023617A1 (en) 1996-11-26 1997-11-24 Hetero-biaryl-pyridoquinazolinone derivatives as anti-cancer agents

Publications (1)

Publication Number Publication Date
ATE218568T1 true ATE218568T1 (de) 2002-06-15

Family

ID=25040889

Family Applications (1)

Application Number Title Priority Date Filing Date
AT97948622T ATE218568T1 (de) 1996-11-26 1997-11-24 Hetero-biaryl-pyridochinazolinonderivate als antikrebsmittel

Country Status (11)

Country Link
EP (1) EP0944628B1 (de)
JP (1) JP2001507341A (de)
AT (1) ATE218568T1 (de)
AU (1) AU5465198A (de)
CA (1) CA2272915A1 (de)
DE (1) DE69713139T2 (de)
DK (1) DK0944628T3 (de)
ES (1) ES2176800T3 (de)
HK (1) HK1021373A1 (de)
PT (1) PT944628E (de)
WO (1) WO1998023617A1 (de)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2314583B1 (de) * 2008-08-12 2015-02-25 Nippon Soda Co., Ltd. Nitrogeniertes heterozyklisches derivat sowie bakterizid-wirkstoff für landwirtschaft und gartenbau
KR101435729B1 (ko) 2009-09-28 2014-09-01 닛뽕소다 가부시키가이샤 함질소 헤테로 고리 화합물 및 그의 염, 그리고 농원예용 살균제
ES2692433A1 (es) * 2017-06-01 2018-12-03 Oncostellae, S.L. Derivados de ácidos carboxílicos como inhibidores de proteinas quinasa
JP7110335B2 (ja) * 2017-06-01 2022-08-01 オンコステラ、ソシエダッド、リミターダ プロテインキナーゼ阻害剤として有用なピリドキナゾリン誘導体

Also Published As

Publication number Publication date
JP2001507341A (ja) 2001-06-05
WO1998023617A1 (en) 1998-06-04
CA2272915A1 (en) 1998-06-04
DK0944628T3 (da) 2002-08-26
DE69713139T2 (de) 2002-12-19
ES2176800T3 (es) 2002-12-01
DE69713139D1 (de) 2002-07-11
HK1021373A1 (en) 2000-06-09
PT944628E (pt) 2002-09-30
AU5465198A (en) 1998-06-22
EP0944628A1 (de) 1999-09-29
EP0944628B1 (de) 2002-06-05

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Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification
EEFA Change of the company name
REN Ceased due to non-payment of the annual fee