ATE188702T1 - Thienodiazepinverbindungen und ihre verwendung - Google Patents

Thienodiazepinverbindungen und ihre verwendung

Info

Publication number
ATE188702T1
ATE188702T1 AT91916944T AT91916944T ATE188702T1 AT E188702 T1 ATE188702 T1 AT E188702T1 AT 91916944 T AT91916944 T AT 91916944T AT 91916944 T AT91916944 T AT 91916944T AT E188702 T1 ATE188702 T1 AT E188702T1
Authority
AT
Austria
Prior art keywords
antidemential
cholecystokinin
useful
inhibitory action
medicine
Prior art date
Application number
AT91916944T
Other languages
English (en)
Inventor
Yoichi Naka
Keiichiro Haga
Masahiro Hosoya
Original Assignee
Yoshitomi Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Yoshitomi Pharmaceutical filed Critical Yoshitomi Pharmaceutical
Application granted granted Critical
Publication of ATE188702T1 publication Critical patent/ATE188702T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D495/14—Ortho-condensed systems
AT91916944T 1991-09-30 1991-09-30 Thienodiazepinverbindungen und ihre verwendung ATE188702T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CA002097285A CA2097285C (en) 1991-09-30 1991-09-30 Thienodiazepine compounds and their use
PCT/JP1991/001315 WO1993007152A1 (fr) 1991-09-30 1991-09-30 Compose a base de thienodiazepine et son utilisation

Publications (1)

Publication Number Publication Date
ATE188702T1 true ATE188702T1 (de) 2000-01-15

Family

ID=25676237

Family Applications (1)

Application Number Title Priority Date Filing Date
AT91916944T ATE188702T1 (de) 1991-09-30 1991-09-30 Thienodiazepinverbindungen und ihre verwendung

Country Status (8)

Country Link
US (1) US5439905A (de)
EP (1) EP0559891B1 (de)
KR (1) KR970002640B1 (de)
AT (1) ATE188702T1 (de)
CA (1) CA2097285C (de)
DE (1) DE69131907T2 (de)
ES (1) ES2140396T3 (de)
WO (1) WO1993007152A1 (de)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0692483A1 (de) * 1993-03-30 1996-01-17 Yoshitomi Pharmaceutical Industries, Ltd. Zelladhäsionsinhibitor und thienotriazoldiazepin-derivat
US5426185A (en) * 1993-11-22 1995-06-20 Merck & Co., Inc. Antiarrhythmic benzodiazepines
WO1995032963A1 (fr) * 1994-06-01 1995-12-07 Yoshitomi Pharmaceutical Industries, Ltd. Compose de thienylazole et compose de thienotriazolodiazepine
BR9508608A (pt) * 1994-08-18 1997-12-30 Merck & Co Inc Composto formulação farmacêutica e processo para prevenir ou tratar arritmia
US5700797A (en) * 1995-06-07 1997-12-23 Merck & Co, Inc. N-(2,4-dioxo-2,3,4,5-tetrahydro-1H-1,5-benzodiazepin-3-yl)-3-amides
US5691331A (en) * 1995-06-07 1997-11-25 Merck & Co., Inc. N-(2,4-Dioxo-2,3,4,5-tetrahydro-1H-1,5-benzodiazepin-3yl) -3- amides
US5631251A (en) * 1995-06-07 1997-05-20 Merck & Co., Inc. 5-cyclopropyl-1,4 benzodiazepine-2-ones
AU720378B2 (en) * 1995-06-07 2000-06-01 Merck & Co., Inc. Novel N-(4-oxo-2,3,4,5-tetrahydro-1H-1, 5-benzodiazepin-3yl)-3-amides
US5726171A (en) * 1995-06-07 1998-03-10 Merck & Co Inc N-(1-alkyl-5-phenyl-2,3,4,5-tetrahydro-1H-benzo B! 1,4!diazepin-3yl)-acetamides
US5776930A (en) * 1996-06-28 1998-07-07 Merck & Company, Inc. Pharmaceutical preparation
JP2000510155A (ja) * 1996-06-28 2000-08-08 メルク エンド カンパニー インコーポレーテッド 医薬製剤
WO2012075456A1 (en) 2010-12-02 2012-06-07 Constellation Pharmaceuticals Bromodomain inhibitors and uses thereof
AR084070A1 (es) 2010-12-02 2013-04-17 Constellation Pharmaceuticals Inc Inhibidores del bromodominio y usos de los mismos
EP2705039B1 (de) 2011-05-04 2017-07-26 Constellation Pharmaceuticals, Inc. Bromodomainhemmer und ihre verwendung
WO2012174487A2 (en) 2011-06-17 2012-12-20 Constellation Pharmaceuticals, Inc. Bromodomain inhibitors and uses thereof
EP2864336B1 (de) 2012-06-06 2016-11-23 Constellation Pharmaceuticals, Inc. Benzo[b]isoxazolazepinbromdomänenhemmer und verwendungen davon
TWI602820B (zh) 2012-06-06 2017-10-21 星宿藥物公司 溴域抑制劑及其用途
ES2725928T3 (es) 2014-06-20 2019-09-30 Constellation Pharmaceuticals Inc Formas cristalinas de 2-((4S)-6-(4-clorofenil)-1-metil-4H-benzo[c]isoxazolo[4,5-e]azepin-4-il)acetamida
KR101675984B1 (ko) 2015-02-23 2016-11-14 한양대학교 에리카산학협력단 티에노디아제핀 유도체 또는 이의 약학적으로 허용가능한 염, 및 이를 유효성분으로 포함하는 약학적 조성물

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1989005812A1 (en) * 1987-12-22 1989-06-29 Yoshitomi Pharmaceutical Industries, Ltd. Thienodiazepine compounds and their medicinal use
JP2953045B2 (ja) * 1989-12-01 1999-09-27 吉富製薬株式会社 チエノジアゼピン化合物
IL96613A0 (en) * 1989-12-18 1991-09-16 Merck & Co Inc Pharmaceutical compositions containing benzodiazepine analogs

Also Published As

Publication number Publication date
KR970002640B1 (ko) 1997-03-07
CA2097285A1 (en) 1993-03-31
EP0559891B1 (de) 2000-01-12
ES2140396T3 (es) 2000-03-01
US5439905A (en) 1995-08-08
WO1993007152A1 (fr) 1993-04-15
CA2097285C (en) 2000-03-14
DE69131907T2 (de) 2000-06-15
EP0559891A1 (de) 1993-09-15
EP0559891A4 (de) 1994-03-16
DE69131907D1 (de) 2000-02-17

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Legal Events

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