ATE101150T1 - Thiophen-2-carboxamid-derivate und ihre verwendung als pharmazeutische mittel. - Google Patents
Thiophen-2-carboxamid-derivate und ihre verwendung als pharmazeutische mittel.Info
- Publication number
- ATE101150T1 ATE101150T1 AT89309970T AT89309970T ATE101150T1 AT E101150 T1 ATE101150 T1 AT E101150T1 AT 89309970 T AT89309970 T AT 89309970T AT 89309970 T AT89309970 T AT 89309970T AT E101150 T1 ATE101150 T1 AT E101150T1
- Authority
- AT
- Austria
- Prior art keywords
- alkyl
- thiophene
- pharmaceutical agents
- carboxamide derivatives
- ch2oc1
- Prior art date
Links
- 239000008177 pharmaceutical agent Substances 0.000 title 1
- DENPQNAWGQXKCU-UHFFFAOYSA-N thiophene-2-carboxamide Chemical class NC(=O)C1=CC=CS1 DENPQNAWGQXKCU-UHFFFAOYSA-N 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 abstract 4
- 125000006273 (C1-C3) alkyl group Chemical group 0.000 abstract 2
- 125000004178 (C1-C4) alkyl group Chemical group 0.000 abstract 2
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 125000000719 pyrrolidinyl group Chemical group 0.000 abstract 1
- -1 pyrrolidinylmethyl Chemical group 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Hospice & Palliative Care (AREA)
- Otolaryngology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB888823040A GB8823040D0 (en) | 1988-09-30 | 1988-09-30 | Organic compounds & their use as pharmaceuticals |
| EP89309970A EP0368464B1 (de) | 1988-09-30 | 1989-09-29 | Thiophen-2-carboxamid-Derivate und ihre Verwendung als pharmazeutische Mittel |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE101150T1 true ATE101150T1 (de) | 1994-02-15 |
Family
ID=10644554
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT89309970T ATE101150T1 (de) | 1988-09-30 | 1989-09-29 | Thiophen-2-carboxamid-derivate und ihre verwendung als pharmazeutische mittel. |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US5021449A (de) |
| EP (1) | EP0368464B1 (de) |
| JP (1) | JP2740296B2 (de) |
| AT (1) | ATE101150T1 (de) |
| CA (1) | CA1338845C (de) |
| DE (1) | DE68912887T2 (de) |
| GB (1) | GB8823040D0 (de) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20040011427A (ko) * | 2000-11-08 | 2004-02-05 | 신젠타 파티서페이션즈 아게 | 피롤카르복시아미드 및 피롤카르보티오아미드 및 그의농화학적 용도 |
| US7521473B2 (en) * | 2004-02-25 | 2009-04-21 | Wyeth | Inhibitors of protein tyrosine phosphatase 1B |
| WO2005081960A2 (en) * | 2004-02-25 | 2005-09-09 | Wyeth | Inhibitors of protein tyrosine phosphatase 1b |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL281394A (de) * | 1961-07-25 | |||
| US3342826A (en) * | 1964-01-13 | 1967-09-19 | Ile De France | Heterocyclic aminoalkyl benzamides |
| US3932503A (en) * | 1966-05-28 | 1976-01-13 | Hoechst Aktiengesellschaft | Benzenesulfonyl ureas |
| GB1166364A (en) * | 1966-11-25 | 1969-10-08 | American Cyanamid Co | N-(Tert-Aminoalkyl) Amide Derivatives and Process for Preparing the Same |
| DE1937759A1 (de) * | 1967-08-12 | 1970-09-24 | Hoechst Ag | Benzolsulfonylsemicarbazide und Verfahren zu ihrer Herstellung |
| DE2500157C2 (de) * | 1975-01-03 | 1983-09-15 | Hoechst Ag, 6230 Frankfurt | N-Acyl-4-(2-aminoäthyl)-benzoesäuren, deren Salze und Ester, Verfahren zu deren Herstellung und deren Verwendung |
| US4123550A (en) * | 1977-10-31 | 1978-10-31 | Syntex (U.S.A.) Inc. | Bicyclo[3.1.0]hexylethylaminocarbonyl-substituted heteroaryl cardiovascular agents |
| US4321378A (en) * | 1979-01-16 | 1982-03-23 | Delalande S.A. | 8-(5-Pyrimidinecarboxamide)nor-tropane derivatives |
| SE8101536L (sv) * | 1981-03-11 | 1982-09-12 | Astra Laekemedel Ab | Bensamid-derivat |
| DE3119796A1 (de) * | 1981-05-19 | 1982-12-23 | Hoechst Ag, 6000 Frankfurt | Substituierte tryptaminderivate von thienyloxpropanolaminen, verfahren zu ihrer herstellung, pharmazeutische praeparate auf basis dieser verbindungen sowie ihre verwendung |
| DE3227329A1 (de) * | 1982-07-22 | 1984-01-26 | Basf Ag, 6700 Ludwigshafen | Verfahren zur herstellung von 2-n,n-disubstituierten aminothiazolen |
| DE3602889A1 (de) * | 1985-06-29 | 1987-01-08 | Bayer Ag | Alkoxycarbonyl-substituierte hydroxythiophen-carbonamide |
| DE3610711A1 (de) * | 1986-03-29 | 1987-10-15 | Bayer Ag | Acyloxythiophen-carbonamide |
| DE3613792A1 (de) * | 1986-04-24 | 1987-10-29 | Bayer Ag | Carbamoyloxythiophen-derivate |
| GB8708833D0 (en) * | 1987-04-13 | 1987-05-20 | Lilly S A E | Organic compounds |
-
1988
- 1988-09-30 GB GB888823040A patent/GB8823040D0/en active Pending
-
1989
- 1989-09-25 CA CA000612931A patent/CA1338845C/en not_active Expired - Fee Related
- 1989-09-26 US US07/412,685 patent/US5021449A/en not_active Expired - Fee Related
- 1989-09-29 AT AT89309970T patent/ATE101150T1/de not_active IP Right Cessation
- 1989-09-29 EP EP89309970A patent/EP0368464B1/de not_active Expired - Lifetime
- 1989-09-29 JP JP1255119A patent/JP2740296B2/ja not_active Expired - Lifetime
- 1989-09-29 DE DE68912887T patent/DE68912887T2/de not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| EP0368464A1 (de) | 1990-05-16 |
| DE68912887T2 (de) | 1994-05-26 |
| US5021449A (en) | 1991-06-04 |
| JP2740296B2 (ja) | 1998-04-15 |
| GB8823040D0 (en) | 1988-11-09 |
| DE68912887D1 (de) | 1994-03-17 |
| EP0368464B1 (de) | 1994-02-02 |
| JPH02160780A (ja) | 1990-06-20 |
| CA1338845C (en) | 1997-01-14 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification | ||
| REN | Ceased due to non-payment of the annual fee |