AT372951B - METHOD FOR PRODUCING NEW BENZIMIDAZOLES OR BENZIMIDAZOLIDINES AND THEIR SALTS - Google Patents

METHOD FOR PRODUCING NEW BENZIMIDAZOLES OR BENZIMIDAZOLIDINES AND THEIR SALTS

Info

Publication number
AT372951B
AT372951B AT0263379A AT263379A AT372951B AT 372951 B AT372951 B AT 372951B AT 0263379 A AT0263379 A AT 0263379A AT 263379 A AT263379 A AT 263379A AT 372951 B AT372951 B AT 372951B
Authority
AT
Austria
Prior art keywords
benzimidazolidines
salts
producing new
new benzimidazoles
benzimidazoles
Prior art date
Application number
AT0263379A
Other languages
German (de)
Other versions
ATA263379A (en
Original Assignee
Mundipharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mundipharma Ag filed Critical Mundipharma Ag
Publication of ATA263379A publication Critical patent/ATA263379A/en
Application granted granted Critical
Publication of AT372951B publication Critical patent/AT372951B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10Antioedematous agents; Diuretics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D235/08Radicals containing only hydrogen and carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/18Benzimidazoles; Hydrogenated benzimidazoles with aryl radicals directly attached in position 2
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/30Nitrogen atoms not forming part of a nitro radical

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
AT0263379A 1978-04-10 1979-04-09 METHOD FOR PRODUCING NEW BENZIMIDAZOLES OR BENZIMIDAZOLIDINES AND THEIR SALTS AT372951B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US89504878A 1978-04-10 1978-04-10

Publications (2)

Publication Number Publication Date
ATA263379A ATA263379A (en) 1983-04-15
AT372951B true AT372951B (en) 1983-12-12

Family

ID=25403870

Family Applications (1)

Application Number Title Priority Date Filing Date
AT0263379A AT372951B (en) 1978-04-10 1979-04-09 METHOD FOR PRODUCING NEW BENZIMIDAZOLES OR BENZIMIDAZOLIDINES AND THEIR SALTS

Country Status (19)

Country Link
JP (1) JPS54138561A (en)
AT (1) AT372951B (en)
AU (1) AU531086B2 (en)
BE (1) BE875425A (en)
CA (1) CA1126280A (en)
DE (1) DE2914084A1 (en)
DK (1) DK139079A (en)
ES (1) ES479446A1 (en)
FI (1) FI74461C (en)
FR (1) FR2422644A1 (en)
GB (1) GB2018766B (en)
GR (1) GR68483B (en)
IL (1) IL57105A (en)
IT (1) IT1193755B (en)
NL (1) NL7902802A (en)
NZ (1) NZ190136A (en)
PT (1) PT69458A (en)
SE (1) SE446532B (en)
ZA (1) ZA791726B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102070466A (en) * 2010-12-28 2011-05-25 天津市筠凯化工科技有限公司 Preparation method of 5-chiorine-2-nitroaniline
CN108558712A (en) * 2018-06-20 2018-09-21 新乡市锦源化工有限公司 It is a kind of using antifebrin as the method and P-aminobenzene-sulfonamide of Material synthesis high-purity P-aminobenzene-sulfonamide
CN110305018B (en) * 2019-06-06 2022-07-15 浙江普洛家园药业有限公司 Preparation method of 3-bromo-2-fluoronitrobenzene

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH404675A (en) * 1961-06-29 1965-12-31 Siegfried Ag Process for the preparation of new heterocyclic sulfonamido compounds
FR1469504A (en) * 1964-10-22 1967-02-17 Fisons Pest Control Ltd Insecticidal compounds
FR1477792A (en) * 1965-03-24 1967-04-21 Fisons Pest Control Ltd New benzimidazoles
GB1163262A (en) * 1966-01-13 1969-09-04 Fisons Pest Control Ltd Substituted Benzimidazoles and Biocidally Active Compositions
GB1356244A (en) * 1970-07-29 1974-06-12 Fisons Ltd Substituted benzimidazole parasiticides

Also Published As

Publication number Publication date
NZ190136A (en) 1982-11-23
AU531086B2 (en) 1983-08-11
NL7902802A (en) 1979-10-12
DE2914084A1 (en) 1979-10-25
CA1126280A (en) 1982-06-22
GB2018766A (en) 1979-10-24
ATA263379A (en) 1983-04-15
PT69458A (en) 1979-05-01
FR2422644B1 (en) 1982-12-17
IL57105A0 (en) 1979-07-25
FI74461B (en) 1987-10-30
IT7948686A0 (en) 1979-04-10
FR2422644A1 (en) 1979-11-09
AU4567579A (en) 1979-10-18
SE7902911L (en) 1979-10-11
GB2018766B (en) 1982-09-22
ZA791726B (en) 1980-05-28
IL57105A (en) 1983-10-31
JPS54138561A (en) 1979-10-27
GR68483B (en) 1982-01-04
IT1193755B (en) 1988-08-24
FI74461C (en) 1988-02-08
DK139079A (en) 1979-10-11
BE875425A (en) 1979-07-31
ES479446A1 (en) 1979-08-01
FI791083A (en) 1979-10-11
SE446532B (en) 1986-09-22
JPH0250904B2 (en) 1990-11-05

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Legal Events

Date Code Title Description
ELJ Ceased due to non-payment of the annual fee