AR230748A1 - Procedimiento para la preparacion de derivados de imidazo(1,2-a)tien(3,2-d)pirimidim-6,9-(5h,7h)-diona y compuestos para su exclusivo uso como intermediarios en dicho procedimiento - Google Patents

Procedimiento para la preparacion de derivados de imidazo(1,2-a)tien(3,2-d)pirimidim-6,9-(5h,7h)-diona y compuestos para su exclusivo uso como intermediarios en dicho procedimiento

Info

Publication number
AR230748A1
AR230748A1 AR285881A AR28588181A AR230748A1 AR 230748 A1 AR230748 A1 AR 230748A1 AR 285881 A AR285881 A AR 285881A AR 28588181 A AR28588181 A AR 28588181A AR 230748 A1 AR230748 A1 AR 230748A1
Authority
AR
Argentina
Prior art keywords
procedure
pirimidim
diona
intermediaries
compounds
Prior art date
Application number
AR285881A
Other languages
English (en)
Spanish (es)
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Application granted granted Critical
Publication of AR230748A1 publication Critical patent/AR230748A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D495/14—Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pulmonology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Immunology (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
AR285881A 1980-06-27 1981-06-26 Procedimiento para la preparacion de derivados de imidazo(1,2-a)tien(3,2-d)pirimidim-6,9-(5h,7h)-diona y compuestos para su exclusivo uso como intermediarios en dicho procedimiento AR230748A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH499580 1980-06-27

Publications (1)

Publication Number Publication Date
AR230748A1 true AR230748A1 (es) 1984-06-29

Family

ID=4286126

Family Applications (1)

Application Number Title Priority Date Filing Date
AR285881A AR230748A1 (es) 1980-06-27 1981-06-26 Procedimiento para la preparacion de derivados de imidazo(1,2-a)tien(3,2-d)pirimidim-6,9-(5h,7h)-diona y compuestos para su exclusivo uso como intermediarios en dicho procedimiento

Country Status (25)

Country Link
US (2) US4376121A (fr)
EP (1) EP0043054B1 (fr)
JP (1) JPS5762282A (fr)
KR (1) KR840000705B1 (fr)
AR (1) AR230748A1 (fr)
AT (1) ATE9698T1 (fr)
AU (1) AU7196781A (fr)
BR (1) BR8103967A (fr)
CA (1) CA1142924A (fr)
CS (1) CS217997B2 (fr)
CU (1) CU35489A (fr)
DE (1) DE3166449D1 (fr)
DK (1) DK252981A (fr)
ES (1) ES8207541A1 (fr)
FI (1) FI811600L (fr)
GR (1) GR74943B (fr)
HU (1) HU181608B (fr)
IL (1) IL63145A (fr)
MC (1) MC1395A1 (fr)
NO (1) NO812208L (fr)
NZ (1) NZ197476A (fr)
PH (1) PH16060A (fr)
PT (1) PT73270B (fr)
ZA (1) ZA814162B (fr)
ZW (1) ZW11781A1 (fr)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZW11781A1 (en) * 1980-06-27 1982-01-20 Hoffmann La Roche Pyrimidine derivatives
US4797486A (en) * 1986-09-08 1989-01-10 Pfizer Inc. Heterocyclic ring fused pyrimidine-4(3H)-ones as anticoccidial agents
US4725599A (en) * 1986-09-08 1988-02-16 Pfizer Inc. Heterocyclic ring fused pyrimidine-4 (3H)-ones as anticoccidial agents
DK522187D0 (da) * 1987-10-06 1987-10-06 Ferrosan As Imidozothienopyrimidiner, deres fremstilling og anvendelse
DK0888359T3 (da) 1996-03-11 2002-08-12 Syngenta Participations Ag Pyrimidin-4-on-derivat som pesticid
FR2872165B1 (fr) 2004-06-24 2006-09-22 Sod Conseils Rech Applic Nouveaux derives de pyrimido-benzimidazole
US8809346B2 (en) * 2008-05-30 2014-08-19 Universite De Versailles-Saint-Quentin-En-Yvelines ANT-ligands molecules and biological applications
CN104478851A (zh) * 2014-12-31 2015-04-01 济南诚汇双达化工有限公司 一种盐酸阿替卡因的制备方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE755404A (fr) * 1969-08-29 1971-03-01 Sandoz Sa Nouveau derives de la thiazolo-(3,2-a) pyrrolo (2,3-d) pyrimidine, leurpreparation et medicaments contenant ces derives
US3932407A (en) * 1973-11-19 1976-01-13 Bristol-Myers Company Optionally substituted 1,2,3,5-tetrahydroimidezo(2,1-b)-quinazolin-2-ones and 6(H)-1,2,3,4-tetrahydropyimido(2,1-b)quinazolin-2-ones
DE2411274A1 (de) * 1974-03-06 1975-09-18 Schering Ag Neue 2-nitrothieno eckige klammer auf 2,3-d eckige klammer zu pyrimidinon-derivate und verfahren zu ihrer herstellung
DE2411273A1 (de) * 1974-03-06 1975-09-18 Schering Ag Neue thieno eckige klammer auf 2,3-d eckige klammer zu pyrimidinone und verfahren zu ihrer herstellung
US4054656A (en) * 1975-09-10 1977-10-18 Mead Johnson & Company Thieno[2,3-d]pyrimidine antiallergic agents
JPS5527105A (en) * 1978-08-11 1980-02-27 Dai Ichi Seiyaku Co Ltd Imidazothienopyrimidinones compound
US4230707A (en) * 1979-08-27 1980-10-28 Warner-Lambert Company Oxo-pyrido[1,2-a]thienopyrimidine compounds and methods for their production
ZW11781A1 (en) * 1980-06-27 1982-01-20 Hoffmann La Roche Pyrimidine derivatives

Also Published As

Publication number Publication date
HU181608B (en) 1983-10-28
KR830006302A (ko) 1983-09-20
ZW11781A1 (en) 1982-01-20
PH16060A (en) 1983-06-09
ES503407A0 (es) 1982-10-01
US4442289A (en) 1984-04-10
CS217997B2 (en) 1983-02-25
ZA814162B (en) 1982-07-28
PT73270A (en) 1981-07-01
CU35489A (en) 1982-12-22
FI811600L (fi) 1981-12-28
JPS5762282A (en) 1982-04-15
NZ197476A (en) 1984-05-31
ES8207541A1 (es) 1982-10-01
ATE9698T1 (de) 1984-10-15
EP0043054B1 (fr) 1984-10-03
BR8103967A (pt) 1982-03-09
EP0043054A3 (en) 1982-03-17
CA1142924A (fr) 1983-03-15
EP0043054A2 (fr) 1982-01-06
PT73270B (en) 1983-05-11
DE3166449D1 (en) 1984-11-08
MC1395A1 (fr) 1982-04-27
KR840000705B1 (ko) 1984-05-21
AU7196781A (en) 1982-01-07
US4376121A (en) 1983-03-08
IL63145A0 (en) 1981-09-13
IL63145A (en) 1984-05-31
GR74943B (fr) 1984-07-12
NO812208L (no) 1981-12-28
DK252981A (da) 1981-12-28

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