AR224392A1 - Procedimiento para preparar compuestos de 2-(2-guanidin-4-tiazolilmetiltio)-etil o propilamino 5-metil-4-pirimidona y sus sales utiles como antagonistas de la histamina - Google Patents
Procedimiento para preparar compuestos de 2-(2-guanidin-4-tiazolilmetiltio)-etil o propilamino 5-metil-4-pirimidona y sus sales utiles como antagonistas de la histaminaInfo
- Publication number
- AR224392A1 AR224392A1 AR280058A AR28005880A AR224392A1 AR 224392 A1 AR224392 A1 AR 224392A1 AR 280058 A AR280058 A AR 280058A AR 28005880 A AR28005880 A AR 28005880A AR 224392 A1 AR224392 A1 AR 224392A1
- Authority
- AR
- Argentina
- Prior art keywords
- thiazolylmethyll
- guanidin
- pyrimidone
- propylamine
- ethyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/55—Acids; Esters
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB7906070 | 1979-02-21 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR224392A1 true AR224392A1 (es) | 1981-11-30 |
Family
ID=10503327
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AR280058A AR224392A1 (es) | 1979-02-21 | 1980-02-21 | Procedimiento para preparar compuestos de 2-(2-guanidin-4-tiazolilmetiltio)-etil o propilamino 5-metil-4-pirimidona y sus sales utiles como antagonistas de la histamina |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US4521418A (es) |
| EP (1) | EP0015138B1 (es) |
| JP (1) | JPS55115883A (es) |
| AR (1) | AR224392A1 (es) |
| AT (1) | AT377260B (es) |
| AU (1) | AU536194B2 (es) |
| DD (1) | DD149217A5 (es) |
| DE (1) | DE3062310D1 (es) |
| DK (1) | DK74680A (es) |
| ES (1) | ES488772A0 (es) |
| FI (1) | FI800515A (es) |
| GR (1) | GR74009B (es) |
| IE (1) | IE49270B1 (es) |
| NO (1) | NO800463L (es) |
| PL (1) | PL222115A1 (es) |
| PT (1) | PT70850A (es) |
| RO (1) | RO79711A (es) |
| ZA (1) | ZA801002B (es) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4383343A (en) * | 1979-08-09 | 1983-05-17 | Kulka Thomas S | Foot supporting strap for hospital bed |
| US4227271A (en) * | 1979-08-09 | 1980-10-14 | Kulka Thomas S | Foot supporting strap for hospital bed |
| NZ202797A (en) * | 1981-12-28 | 1985-08-30 | Lilly Co Eli | Pyrimidine derivatives and pharmaceutical compositions |
| CA1211111A (en) * | 1982-02-15 | 1986-09-09 | Isao Yanagisawa | Process for preparing novel pyrimidone compounds |
| US4808589A (en) * | 1982-02-20 | 1989-02-28 | Smith Kline & French Laboratories Limited | Pyrimidone derivatives |
| US4444381A (en) * | 1982-05-11 | 1984-04-24 | Wayne Sherwyn J | Operating table accessory, particularly for lumbar laminectomies |
| DE3220118A1 (de) * | 1982-05-28 | 1983-12-01 | Bayer Ag, 5090 Leverkusen | Alkylenverbrueckte guanidinothiazolderivate, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel |
| DE3306102C1 (de) * | 1983-02-22 | 1984-08-02 | Ludwig Heumann & Co GmbH, 8500 Nürnberg | Pyridin-Pyrimidinon-Derivate,Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel |
| GB8320505D0 (en) * | 1983-07-29 | 1983-09-01 | Smith Kline French Lab | Chemical compounds |
| US4772704A (en) * | 1983-09-21 | 1988-09-20 | Bristol-Myers Company | 2,5-disubstituted-4(3H)-pyrimidones having histamine H2 -receptor antagonist activity |
| GB8421427D0 (en) * | 1984-08-23 | 1984-09-26 | Smith Kline French Lab | Chemical compounds |
| IT1178026B (it) * | 1984-10-05 | 1987-09-03 | Medosan Ind Biochimi | Derivati del 2-amino-tiazolo |
| JO1410B1 (en) * | 1984-11-03 | 1986-11-30 | سميث كلاين اند فرينش لابوراتوريز ليمتد | Vehicles |
| JP2807577B2 (ja) * | 1990-06-15 | 1998-10-08 | エーザイ株式会社 | 環状アミド誘導体 |
| US5611097A (en) * | 1995-08-17 | 1997-03-18 | Dumke; Dan | Foot stop for beds |
| WO2022034121A1 (en) | 2020-08-11 | 2022-02-17 | Université De Strasbourg | H2 blockers targeting liver macrophages for the prevention and treatment of liver disease and cancer |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1223686A (en) * | 1967-02-24 | 1971-03-03 | Ici Ltd | Salts of pyrimidine derivatives and the use thereof as fungicides |
| US3980781A (en) * | 1966-03-31 | 1976-09-14 | Imperial Chemical Industries Limited | Fungicidal composition and method containing 2-amino-pyrimidines |
| GB1419994A (en) * | 1973-05-03 | 1976-01-07 | Smith Kline French Lab | Heterocyclicalkylaminotheterocyclic compounds methods for their preparation and compositions comprising them |
| IN146736B (es) * | 1975-10-02 | 1979-08-25 | Smith Kline French Lab | |
| US4145546A (en) * | 1975-10-02 | 1979-03-20 | Smith Kline & French Laboratories Limited | 4-Pyrimidone compounds |
| US4154834A (en) * | 1975-12-29 | 1979-05-15 | Smith Kline & French Laboratories Limited | Substituted isocytosines having histamine H2 -antagonist activity |
| MW5076A1 (en) * | 1975-12-29 | 1978-02-08 | Smith Kline French Lab | Pharmacologicalle active compounds |
| US4216318A (en) * | 1975-12-29 | 1980-08-05 | Smith Kline & French Laboratories Limited | Heterocyclic alkyl 4-pyrimidones |
| US4165378A (en) * | 1977-04-20 | 1979-08-21 | Ici Americas Inc. | Guanidine derivatives of imidazoles and thiazoles |
| NO781300L (no) * | 1977-04-20 | 1978-10-23 | Ici Ltd | Fremgangsmaate for fremstilling av fysiologisk aktive guanidinderivater |
| DE2817078C2 (de) * | 1977-04-20 | 1995-06-14 | Zeneca Ltd | Guanidinderivate |
| DE2961923D1 (en) * | 1978-01-18 | 1982-03-11 | Ici Plc | Antisecretory guanidine derivatives, processes for their manufacture and pharmaceutical compositions containing them |
| US4374836A (en) * | 1978-10-16 | 1983-02-22 | Imperial Chemical Industries Ltd. | Antisecretory heterocyclic derivatives, process for their manufacture and pharmaceutical compositions containing them |
-
1980
- 1980-02-12 US US06/120,807 patent/US4521418A/en not_active Expired - Lifetime
- 1980-02-19 GR GR61235A patent/GR74009B/el unknown
- 1980-02-20 JP JP2106580A patent/JPS55115883A/ja active Pending
- 1980-02-20 PL PL22211580A patent/PL222115A1/xx unknown
- 1980-02-20 DE DE8080300478T patent/DE3062310D1/de not_active Expired
- 1980-02-20 ES ES488772A patent/ES488772A0/es active Granted
- 1980-02-20 EP EP80300478A patent/EP0015138B1/en not_active Expired
- 1980-02-20 IE IE337/80A patent/IE49270B1/en unknown
- 1980-02-20 PT PT70850A patent/PT70850A/pt unknown
- 1980-02-20 NO NO800463A patent/NO800463L/no unknown
- 1980-02-21 AR AR280058A patent/AR224392A1/es active
- 1980-02-21 DK DK74680A patent/DK74680A/da not_active Application Discontinuation
- 1980-02-21 ZA ZA00801002A patent/ZA801002B/xx unknown
- 1980-02-21 AU AU55791/80A patent/AU536194B2/en not_active Ceased
- 1980-02-21 RO RO80100261A patent/RO79711A/ro unknown
- 1980-02-21 FI FI800515A patent/FI800515A/fi not_active Application Discontinuation
- 1980-02-21 DD DD80219202A patent/DD149217A5/de unknown
- 1980-02-21 AT AT0098280A patent/AT377260B/de not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| DE3062310D1 (en) | 1983-04-21 |
| IE800337L (en) | 1980-08-21 |
| US4521418A (en) | 1985-06-04 |
| DK74680A (da) | 1980-08-22 |
| ES8103078A1 (es) | 1981-02-16 |
| ATA98280A (de) | 1984-07-15 |
| AU536194B2 (en) | 1984-04-19 |
| ES488772A0 (es) | 1981-02-16 |
| ZA801002B (en) | 1981-03-25 |
| FI800515A (fi) | 1980-08-22 |
| IE49270B1 (en) | 1985-09-04 |
| JPS55115883A (en) | 1980-09-06 |
| RO79711A (ro) | 1982-08-17 |
| GR74009B (es) | 1984-06-06 |
| NO800463L (no) | 1980-08-22 |
| DD149217A5 (de) | 1981-07-01 |
| PL222115A1 (es) | 1980-12-01 |
| AT377260B (de) | 1985-02-25 |
| EP0015138A1 (en) | 1980-09-03 |
| EP0015138B1 (en) | 1983-03-16 |
| AU5579180A (en) | 1980-08-28 |
| PT70850A (en) | 1980-03-01 |
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