AR204813A1 - Proceso para la preparacion de derivados de ampilicina - Google Patents

Proceso para la preparacion de derivados de ampilicina

Info

Publication number
AR204813A1
AR204813A1 ARJA247904A AR24790473A AR204813A1 AR 204813 A1 AR204813 A1 AR 204813A1 AR JA247904 A ARJA247904 A AR JA247904A AR 24790473 A AR24790473 A AR 24790473A AR 204813 A1 AR204813 A1 AR 204813A1
Authority
AR
Argentina
Prior art keywords
ampylicin
derivatives
preparation
ampylicin derivatives
Prior art date
Application number
ARJA247904A
Other languages
English (en)
Spanish (es)
Original Assignee
Yamanouchi Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP4511872A external-priority patent/JPS5547036B2/ja
Priority claimed from JP8342472A external-priority patent/JPS4941396A/ja
Priority claimed from JP8510272A external-priority patent/JPS4942692A/ja
Priority claimed from JP8510372A external-priority patent/JPS4942693A/ja
Priority claimed from JP12595272A external-priority patent/JPS4981388A/ja
Application filed by Yamanouchi Pharma Co Ltd filed Critical Yamanouchi Pharma Co Ltd
Priority claimed from JP1991773A external-priority patent/JPS49108092A/ja
Priority claimed from JP3813273A external-priority patent/JPS49125386A/ja
Application granted granted Critical
Publication of AR204813A1 publication Critical patent/AR204813A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/44Compounds with an amino radical acylated by carboxylic acids, attached in position 6
    • C07D499/48Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical
    • C07D499/58Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical
    • C07D499/64Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms
    • C07D499/68Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms with aromatic rings as additional substituents on the carbon chain

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ARJA247904A 1972-05-08 1973-01-01 Proceso para la preparacion de derivados de ampilicina AR204813A1 (es)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
JP4511872A JPS5547036B2 (fi) 1972-05-08 1972-05-08
JP8342472A JPS4941396A (fi) 1972-08-21 1972-08-21
JP8510272A JPS4942692A (fi) 1972-08-25 1972-08-25
JP8510372A JPS4942693A (fi) 1972-08-25 1972-08-25
JP12595272A JPS4981388A (fi) 1972-12-15 1972-12-15
JP1991773A JPS49108092A (fi) 1973-02-18 1973-02-18
JP3813273A JPS49125386A (fi) 1973-04-04 1973-04-04

Publications (1)

Publication Number Publication Date
AR204813A1 true AR204813A1 (es) 1976-03-05

Family

ID=27563884

Family Applications (2)

Application Number Title Priority Date Filing Date
ARJA247904A AR204813A1 (es) 1972-05-08 1973-01-01 Proceso para la preparacion de derivados de ampilicina
AR251189A AR204162A1 (es) 1972-05-08 1973-01-01 Proceso para la preparacion de derivados de ampicilina

Family Applications After (1)

Application Number Title Priority Date Filing Date
AR251189A AR204162A1 (es) 1972-05-08 1973-01-01 Proceso para la preparacion de derivados de ampicilina

Country Status (10)

Country Link
US (1) US3953428A (fi)
AR (2) AR204813A1 (fi)
AT (1) AT331970B (fi)
BE (1) BE799202A (fi)
CA (1) CA1050971A (fi)
DE (1) DE2322750A1 (fi)
DK (1) DK139754B (fi)
FI (1) FI58131C (fi)
FR (1) FR2183895B1 (fi)
GB (1) GB1407566A (fi)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4202900A (en) * 1972-09-27 1980-05-13 Ciba-Geigy Corporation Derivatives of penam-3-carboxylic acid and a pharmaceutical composition containing the same
JPS5751837B2 (fi) * 1973-04-05 1982-11-04
US3994874A (en) * 1973-11-07 1976-11-30 Richardson-Merrell Inc. 6-[(2-Oxo-1-pyridinyl)acylamino]penicillin derivatives
US3954734A (en) * 1974-01-21 1976-05-04 Parke, Davis & Company Novel antibacterial amide compounds and process means for producing the same
IL47168A (en) * 1974-05-09 1979-07-25 Toyama Chemical Co Ltd Mono or dioxo piperazino(thio)carbonylamino derivatives ofpenicillins and cephalosporins and process for producing the same
US3989687A (en) * 1974-09-27 1976-11-02 Richardson-Merrell Inc. 4-Oxo-1-pyridinyl penicillin derivatives
GB1568962A (en) * 1975-10-31 1980-06-11 Beecham Group Ltd Reparation and compositions containing them (heterocyclic-carbonylamino)pencillins methods for their p
NZ184434A (en) * 1976-06-30 1979-03-28 Dainippon Pharmaceutical Co Penicillins with a substituted p-hydroxy-benzyl side-chain, and injectable pharmaceutical compositions
GB1579362A (en) * 1977-03-16 1980-11-19 Beecham Group Ltd 6-(a-heterocyclylcarbonyl amino-acetamido)-penicillins and compositions containing them
EP0001041A3 (en) * 1977-07-27 1979-06-27 Sandoz Ag Alpha(pyridonecarboxylamino)-alpha substituted acetamido penicillins and -cephalosporins, process for their preparation, their use in pharmaceuticals; pyridones used in the process
NL7811865A (nl) * 1977-12-06 1979-06-08 Nippon Chemiphar Co Nieuwe penicilline en cefalosporine derivaten en werk- wijze voor de bereiding daarvan.
US4231928A (en) * 1979-04-24 1980-11-04 Bristol-Myers Company Antibacterial agents
JPS5651488A (en) * 1979-10-02 1981-05-09 Meiji Seika Kaisha Ltd Penicillin derivative and its preparation
US5281612A (en) * 1982-09-09 1994-01-25 Warner-Lambert Company Naphthyridine antibacterial agents
IE55898B1 (en) * 1982-09-09 1991-02-14 Warner Lambert Co Antibacterial agents
IT1215277B (it) * 1985-05-27 1990-01-31 Pomezia Roma A Derivato chinolin-lattaminico ad attivita' antibatterica ed inibitrice delle b-lattamasi.
US5328908A (en) * 1988-10-24 1994-07-12 Procter & Gamble Pharmaceuticals, Inc. Antimicrobial quinolone thioureas
US5491139A (en) * 1988-10-24 1996-02-13 The Procter & Gamble Company Antimicrobial quinolonyl lactams
CA2001203C (en) * 1988-10-24 2001-02-13 Thomas P. Demuth, Jr. Novel antimicrobial dithiocarbamoyl quinolones
US5273973A (en) * 1988-10-24 1993-12-28 Norwich Eaton Pharmaceuticals, Inc. Antimicrobial quinolonyl esters
EP0366189A3 (en) * 1988-10-24 1992-01-02 Norwich Eaton Pharmaceuticals, Inc. Novel antimicrobial lactam-quinolones
US5180719A (en) * 1988-10-24 1993-01-19 Norwich Eaton Pharmaceuticals, Inc. Antimicrobial quinolonyl lactam esters
CA2078444A1 (en) * 1990-04-18 1991-10-19 Thomas P. Demuth, Jr. Antimicrobial quinolonyl lactams
FR2713637B1 (fr) * 1993-12-15 1996-01-05 Cird Galderma Nouveaux composés bi-aromatiques dérivés d'amide, compositions pharmaceutiques et cosmétiques les contenant et utilisations.
AU753800B2 (en) * 1997-08-25 2002-10-31 Neurogen Corporation Substituted 4-oxo-napthyridine-3-carboxamides as gaba brain receptor ligands
US6143760A (en) 1997-08-25 2000-11-07 Neurogen Corporation Substituted 4-oxo-napthyridine-3-carboxamides: GABA brain receptor ligands
AU2005251745A1 (en) * 2004-06-04 2005-12-22 The Regents Of The University Of California Compounds having activity in increasing ion transport by mutant-CFTR and uses thereof
US8669370B2 (en) * 2011-01-26 2014-03-11 Sanofi Substituted 3-heteroaroylamino-propionic acid derivatives and their use as pharmaceuticals

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1180745A (en) * 1966-10-04 1970-02-11 Beecham Group Ltd Penicillins
US3668198A (en) * 1970-06-01 1972-06-06 Squibb & Sons Inc {60 -ureido-2,4,6-cycloheptatrienylmethylpenicillins
US3711471A (en) * 1971-02-03 1973-01-16 Bristol Myers Co Purification of 6-{8 d-{60 -(3-guanyl-1-ureido)phenylacetamido{9 {0 penicillanic acid

Also Published As

Publication number Publication date
DK139754B (da) 1979-04-09
FI58131C (fi) 1980-12-10
ATA399573A (de) 1975-12-15
US3953428A (en) 1976-04-27
DE2322750A1 (de) 1973-11-29
GB1407566A (en) 1975-09-24
FI58131B (fi) 1980-08-29
FR2183895A1 (fi) 1973-12-21
AR204162A1 (es) 1975-11-28
AT331970B (de) 1975-12-15
AU5504573A (en) 1974-11-07
BE799202A (fr) 1973-08-31
FR2183895B1 (fi) 1976-07-02
CA1050971A (en) 1979-03-20
DK139754C (fi) 1979-09-24

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