AR115991A1 - EL USO DE AGONISTAS DE LOS RECEPTORES a2 ADRENÉRGICOS PARA MEJORAR LA VISIÓN - Google Patents

EL USO DE AGONISTAS DE LOS RECEPTORES a2 ADRENÉRGICOS PARA MEJORAR LA VISIÓN

Info

Publication number
AR115991A1
AR115991A1 ARP190102374A ARP190102374A AR115991A1 AR 115991 A1 AR115991 A1 AR 115991A1 AR P190102374 A ARP190102374 A AR P190102374A AR P190102374 A ARP190102374 A AR P190102374A AR 115991 A1 AR115991 A1 AR 115991A1
Authority
AR
Argentina
Prior art keywords
visual
individual
compound
formula
pharmaceutically acceptable
Prior art date
Application number
ARP190102374A
Other languages
English (en)
Inventor
Miguel Alcantara
Wayne Chen
Daniel W Gil
Mohammed Dibas
Original Assignee
Allergan Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Allergan Inc filed Critical Allergan Inc
Publication of AR115991A1 publication Critical patent/AR115991A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41841,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41781,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0048Eye, e.g. artificial tears
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0048Eye, e.g. artificial tears
    • A61K9/0051Ocular inserts, ocular implants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/10Ophthalmic agents for accommodation disorders, e.g. myopia

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Ophthalmology & Optometry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Reivindicación 1: Un método para tratar una condición ocular en un individuo que necesita ese tratamiento, el método comprende la administración al individuo de una cantidad terapéuticamente efectiva de un compuesto de la fórmula (1) o una sal suya farmacéuticamente aceptable, y en donde la condición ocular se selecciona de un grupo que consiste en presbicia, visión nocturna deficiente, deslumbramiento visual, destellos visuales, halos visuales y miopía nocturna. Reivindicación 41: Un compuesto de la fórmula (1) o una sal suya farmacéuticamente aceptable, en un método para tratar una condición ocular en un individuo que la necesita, el método comprende la administración al individuo de una cantidad terapéuticamente efectiva de el compuesto de la fórmula (1) o una sal suya farmacéuticamente aceptable, y en donde la condición ocular se selecciona de un grupo que consiste en presbicia, visión nocturna deficiente, deslumbramiento visual, destellos visuales, halos visuales y miopía nocturna.
ARP190102374A 2018-08-21 2019-08-21 EL USO DE AGONISTAS DE LOS RECEPTORES a2 ADRENÉRGICOS PARA MEJORAR LA VISIÓN AR115991A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201862720671P 2018-08-21 2018-08-21

Publications (1)

Publication Number Publication Date
AR115991A1 true AR115991A1 (es) 2021-03-17

Family

ID=67841225

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP190102374A AR115991A1 (es) 2018-08-21 2019-08-21 EL USO DE AGONISTAS DE LOS RECEPTORES a2 ADRENÉRGICOS PARA MEJORAR LA VISIÓN

Country Status (17)

Country Link
US (3) US20210205273A1 (es)
EP (1) EP3840750A1 (es)
JP (1) JP2021534217A (es)
KR (1) KR20210047323A (es)
CN (1) CN112823003A (es)
AR (1) AR115991A1 (es)
AU (1) AU2019325486A1 (es)
BR (1) BR112021003295A2 (es)
CA (1) CA3110318A1 (es)
CL (1) CL2021000440A1 (es)
CO (1) CO2021003460A2 (es)
IL (1) IL280990A (es)
MX (1) MX2021002112A (es)
PH (1) PH12021550372A1 (es)
SG (1) SG11202101730SA (es)
TW (1) TW202021584A (es)
WO (1) WO2020041340A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20210260041A1 (en) * 2020-02-20 2021-08-26 Allergan, Inc. Pharmaceutical compositions of alpha-2-adrenergic receptor agonists and their use for improving vision
JP2024508811A (ja) 2021-02-24 2024-02-28 オキュラ セラピューティクス,インコーポレイテッド 小管内デポーインサータ装置

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5478858A (en) * 1993-12-17 1995-12-26 The Procter & Gamble Company 5-(2-imidazolinylamino) benzimidazole compounds useful as alpha-2 adrenoceptor agonists
US6495583B1 (en) 1997-03-25 2002-12-17 Synaptic Pharmaceutical Corporation Benzimidazole derivatives
US20050244463A1 (en) * 2004-04-30 2005-11-03 Allergan, Inc. Sustained release intraocular implants and methods for treating ocular vasculopathies
US7931909B2 (en) * 2005-05-10 2011-04-26 Allergan, Inc. Ocular therapy using alpha-2 adrenergic receptor compounds having enhanced anterior clearance rates
KR20180117211A (ko) 2010-01-22 2018-10-26 알러간, 인코포레이티드 전방내 서방성 치료제 이식물
US10507245B2 (en) * 2012-07-19 2019-12-17 Luis Felipe Vejarano Restrepo Ophthalmic formulation and method for ameliorating presbyopia
TWI722298B (zh) 2013-03-15 2021-03-21 美商歐樂根公司 含有前列醯胺之眼內植入物
CA2907881A1 (en) 2013-03-27 2014-10-02 Forsight Vision5, Inc. Bimatoprost ocular silicone inserts and methods of use thereof
EP2981248B1 (en) 2013-04-01 2020-09-02 Allergan, Inc. Microsphere drug delivery system for sustained intraocular release
US9089562B2 (en) * 2013-08-28 2015-07-28 Presbyopia Therapies Llc Compositions and methods for the treatment of presbyopia
WO2016168141A1 (en) 2015-04-13 2016-10-20 Forsight Vision5, Inc. Ocular insert composition of semi-crystalline or crystalline pharmaceutically active agent
US11077053B2 (en) * 2018-08-21 2021-08-03 Allergan, Inc. Alpha-2-adrenergic receptor agonists for treatment of presbyopia, visual glare, visual starbursts, visual halos and night myopia

Also Published As

Publication number Publication date
CO2021003460A2 (es) 2021-04-08
US20220160623A1 (en) 2022-05-26
US20210205273A1 (en) 2021-07-08
PH12021550372A1 (en) 2021-11-29
KR20210047323A (ko) 2021-04-29
CN112823003A (zh) 2021-05-18
WO2020041340A1 (en) 2020-02-27
CL2021000440A1 (es) 2021-09-20
BR112021003295A2 (pt) 2021-05-18
JP2021534217A (ja) 2021-12-09
TW202021584A (zh) 2020-06-16
EP3840750A1 (en) 2021-06-30
AU2019325486A1 (en) 2021-03-25
US20220288031A1 (en) 2022-09-15
IL280990A (en) 2021-04-29
CA3110318A1 (en) 2020-02-27
SG11202101730SA (en) 2021-03-30
MX2021002112A (es) 2021-07-16

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