AR098311A1 - Compuestos para el control de artrópodos - Google Patents

Compuestos para el control de artrópodos

Info

Publication number
AR098311A1
AR098311A1 ARP140104156A ARP140104156A AR098311A1 AR 098311 A1 AR098311 A1 AR 098311A1 AR P140104156 A ARP140104156 A AR P140104156A AR P140104156 A ARP140104156 A AR P140104156A AR 098311 A1 AR098311 A1 AR 098311A1
Authority
AR
Argentina
Prior art keywords
alkyl
cycloalkyl
substituted
alkylamino
alkoxy
Prior art date
Application number
ARP140104156A
Other languages
English (en)
Inventor
Dr Horstmann Sebastian
Dr Hallenbach Werner
Grgens Ulrich
Dr Turberg Andreas
Dr Ilg Kerstin
Dr Kbberling Johannes
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of AR098311A1 publication Critical patent/AR098311A1/es

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/041,2,3-Triazoles; Hydrogenated 1,2,3-triazoles
    • C07D249/061,2,3-Triazoles; Hydrogenated 1,2,3-triazoles with aryl radicals directly attached to ring atoms
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01CPLANTING; SOWING; FERTILISING
    • A01C1/00Apparatus, or methods of use thereof, for testing or treating seed, roots, or the like, prior to sowing or planting
    • A01C1/06Coating or dressing seed
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N25/00Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
    • A01N25/30Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests characterised by the surfactants
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647Triazoles; Hydrogenated triazoles
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/713Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with four or more nitrogen atoms as the only ring hetero atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Public Health (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Soil Sciences (AREA)
  • Toxicology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Se describen procedimientos para la preparación de compuestos adecuados para combatir insectos, arácnidos y nematodos en la agricultura así como para combatir ectoparásitos en la medicina veterinaria. Reivindicación 1: Compuestos de la fórmula (1) en la que R¹ representa H, alquilo C₁₋₆, alquenilo C₂₋₆, alquinilo C₂₋₆, cicloalquilo C₃₋₇, alquilcarbonilo C₁₋₆, alcoxicarbonilo C₁₋₆, aril-alquilo C₁₋₃, heteroaril-alquilo C₁₋₃ sustituidos respectivamente dado el caso, los grupos A¹ representa CR² o N; A² representa CR³ o N; A³ representa CR⁴ o N; A⁴ representa CR⁵ o N; B¹ representa CR⁶ o N; B² representa CR⁷ o N; B³ representa CR⁸ o N; B⁴ representa CR⁹ o N; y B⁵ representa CR¹⁰ o N, pero en donde no más que tres de los grupos A¹ a A⁴ representan N y no más que tres de los grupos B¹ a B⁵ representan N; R², R³, R⁴, R⁵, R⁶, R⁷, R⁹ y R¹⁰ independientemente entre sí representa H, halógeno, ciano, nitro, o alquilo C₁₋₆, cicloalquilo C₃₋₆, alcoxi C₁₋₆, N-alcoxi C₁₋₆-imino-alquilo C₁₋₃, alquilsulfanilo C₁₋₆, alquilsulfinilo C₁₋₆, alquilsulfonilo C₁₋₆, N-alquilamino C₁₋₆ o N,N-di-alquilamino C₁₋₆ sustituidos respectivamente dado el caso; si ninguno de los grupos A² y A³ representan N, R³ y R⁴ junto con el átomo de carbono al que están unidos, pueden formar un anillo de 5 ó 6 miembros, que contiene 0, 1 ó 2 átomos-N y/o 0 ó 1 átomo-O y/o 0 ó 1 átomo-S, o si ninguno de los grupos A¹ y A² representan N, R² y R³ junto con el átomo de carbono al que están unidos, pueden formar un anillo de 6 miembros, que contiene 0, 1 ó 2 átomos-N; R⁸ representa halógeno, ciano, nitro, o alquilo C₁₋₆, cicloalquilo C₃₋₆, alcoxi C₁₋₆, N-alcoxi C₁₋₆-imino-alquilo C₁₋₃, alquilsulfanilo C₁₋₆, alquilsulfinilo C₁₋₆, alquilsulfonilo C₁₋₆, N-alquilamino C₁₋₆ o N,N-di-alquilamino C₁₋₆, sustituidos respectivamente dado el caso; W representa O ó S; Q representa H, formilo, hidroxi, amino o alquilo C₁₋₆, alquenilo C₂₋₆, alquinilo C₂₋₆, cicloalquilo C₃₋₆, heterocicloalquilo C₁₋₅, alcoxi C₁₋₄, alquilo C₁₋₆-cicloalquilo C₃₋₆, cicloalquilo C₃₋₆-alquilo C₁₋₆, arilo C₆,C₁₀,C₁₄, heteroarilo C₁₋₅, aril C₆,C₁₀,C₁₄-alquilo C₁₋₃, heteroarilo C₁₋₅-alquilo C₁₋₃, N-alquilamino C₁₋₄, N-alquilcarbonilamino C₁₋₄, o N,N-di-alquilamino C₁₋₄ sustituidos respectivamente dado el caso; o representa un carbociclo de 6 miembros insaturado dado el caso polisustituido con V; o representa un anillo heterocíclico de 5 ó 6 miembros insaturado, dado el caso polisustituido con V, donde V independientemente entre si representa halógeno, ciano, nitro, o alquilo C₁₋₆, alquenilo C₁₋₄, alquinilo C₁₋₄, cicloalquilo C₃₋₆, alcoxi C₁₋₆, N-alcoxi C₁₋₆-imino-alquilo C₁₋₃, alquilsulfanilo C₁₋₆, alquilsulfinilo C₁₋₆, alquilsulfonilo C₁₋₆, o N,N-di-(alquilo C₁₋₆)amino sustituidos respectivamente dado el caso; T representa un heteroaromático de 5 miembros dado el caso sustituido respectivamente que contiene tres heteroaromáticos, seleccionados preferentemente de un grupo que se compone de N, O y S; con la condición que T no represente un resto de fórmula (2), donde R¹³ representa H, halógeno, alquilo C₁₋₄, alquilo C₁₋₆ sustituido con halógeno o ciano; así como sales, N-óxidos y formas tautoméricas de los compuestos de la fórmula (1).
ARP140104156A 2013-11-05 2014-11-05 Compuestos para el control de artrópodos AR098311A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP13191612 2013-11-05

Publications (1)

Publication Number Publication Date
AR098311A1 true AR098311A1 (es) 2016-05-26

Family

ID=49518815

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP140104156A AR098311A1 (es) 2013-11-05 2014-11-05 Compuestos para el control de artrópodos

Country Status (17)

Country Link
US (1) US10836732B2 (es)
EP (1) EP3066083B1 (es)
JP (1) JP2016536365A (es)
KR (1) KR20160078974A (es)
CN (1) CN105873908A (es)
AR (1) AR098311A1 (es)
AU (1) AU2014345595B2 (es)
BR (1) BR112016010164A2 (es)
CA (1) CA2929401A1 (es)
CL (1) CL2016001077A1 (es)
ES (1) ES2759902T3 (es)
IL (1) IL245377A0 (es)
MX (1) MX2016005857A (es)
RU (1) RU2016122104A (es)
TW (1) TW201609674A (es)
WO (1) WO2015067648A1 (es)
ZA (1) ZA201603793B (es)

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CN108368064B (zh) * 2015-11-30 2022-04-26 北兴化学工业株式会社 1,2,3-三唑衍生物和包含这种衍生物作为活性成分的杀虫剂和杀螨剂
MX2018007527A (es) 2015-12-22 2018-09-07 Syngenta Participations Ag Derivados de pirazol activos como pesticidas.
JP6850300B2 (ja) 2016-02-18 2021-03-31 シンジェンタ パーティシペーションズ アーゲー 殺有害生物活性ピラゾール誘導体
US11472797B2 (en) 2017-04-05 2022-10-18 Syngenta Participations Ag Pesticidally active pyrazole derivatives
WO2018185191A1 (en) 2017-04-05 2018-10-11 Syngenta Participations Ag Pesticidally active pyrazole derivatives
EP3606917A1 (en) 2017-04-05 2020-02-12 Syngenta Participations AG Pesticidally active pyrazole derivatives
JP7202371B2 (ja) 2017-06-19 2023-01-11 シンジェンタ パーティシペーションズ アーゲー 殺有害生物的に活性なピラゾール誘導体
AR112673A1 (es) 2017-08-11 2019-11-27 Syngenta Participations Ag Derivados de pirazol activos como plaguicidas
AR112672A1 (es) 2017-08-11 2019-11-27 Syngenta Participations Ag Derivados de tiofeno activos como plaguicidas
US11252963B2 (en) 2017-08-11 2022-02-22 Syngenta Participations Ag Pesticidally active pyrazole derivatives
US20200288713A1 (en) 2017-08-11 2020-09-17 Syngenta Participations Ag Pesticidally active pyrazole derivatives
WO2019068819A1 (en) 2017-10-06 2019-04-11 Syngenta Participations Ag PYRROLE DERIVATIVES ACTIVE ON THE PESTICIDE PLAN
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WO2019089631A1 (en) * 2017-10-30 2019-05-09 University Of North Texas Health Science Center At Fort Worth Deterrents for arthropods and marine organisms
CN109761918B (zh) * 2018-12-14 2021-10-26 华南理工大学 一种n1-(2,2,2-三氟-1-芳基乙基)-三氮唑衍生物及其合成方法
WO2020127345A1 (en) 2018-12-21 2020-06-25 Syngenta Participations Ag Pesticidally active pyrazole derivatives
WO2020164994A1 (en) 2019-02-13 2020-08-20 Syngenta Crop Protection Ag Pesticidally active pyrazole derivatives
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JPWO2020251013A1 (es) 2019-06-13 2020-12-17
CN111920791A (zh) * 2020-09-16 2020-11-13 新疆医科大学第一附属医院 枯茗醛在制备治疗细粒棘球蚴病药物中的应用
CR20230492A (es) 2021-04-01 2023-11-23 Sterilex LLC Desinfectante/sanitizante en polvo sin quats
CN117736196A (zh) * 2022-09-15 2024-03-22 顺毅股份有限公司 一种吡啶酰胺衍生物及其用途

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Also Published As

Publication number Publication date
RU2016122104A3 (es) 2018-06-07
EP3066083B1 (de) 2019-10-30
WO2015067648A1 (de) 2015-05-14
US20160280668A1 (en) 2016-09-29
US10836732B2 (en) 2020-11-17
ZA201603793B (en) 2019-04-24
BR112016010164A2 (pt) 2017-08-08
MX2016005857A (es) 2016-08-11
CN105873908A (zh) 2016-08-17
KR20160078974A (ko) 2016-07-05
RU2016122104A (ru) 2017-12-11
AU2014345595A1 (en) 2016-05-19
ES2759902T3 (es) 2020-05-12
JP2016536365A (ja) 2016-11-24
CL2016001077A1 (es) 2017-01-27
EP3066083A1 (de) 2016-09-14
AU2014345595B2 (en) 2019-01-24
TW201609674A (zh) 2016-03-16
IL245377A0 (en) 2016-06-30
CA2929401A1 (en) 2015-05-14

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