AR096402A1 - Medicamento de metformina y dihidroquercetina - Google Patents

Medicamento de metformina y dihidroquercetina

Info

Publication number
AR096402A1
AR096402A1 ARP140102045A ARP140102045A AR096402A1 AR 096402 A1 AR096402 A1 AR 096402A1 AR P140102045 A ARP140102045 A AR P140102045A AR P140102045 A ARP140102045 A AR P140102045A AR 096402 A1 AR096402 A1 AR 096402A1
Authority
AR
Argentina
Prior art keywords
pharmaceutically acceptable
acceptable salt
metformin
methormin
dihydrochercetin
Prior art date
Application number
ARP140102045A
Other languages
English (en)
Inventor
Onishi Kenji
Nagahama Yasuharu
Watanabe Takashi
Kiyono Kunihiko
Original Assignee
Otsuka Pharmaceuticals Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Otsuka Pharmaceuticals Co Ltd filed Critical Otsuka Pharmaceuticals Co Ltd
Publication of AR096402A1 publication Critical patent/AR096402A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A61K31/3533,4-Dihydrobenzopyrans, e.g. chroman, catechin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/155Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/18Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Abstract

Medicamento para reducir los efectos colaterales de metformina o una de sus sales farmacéuticamente aceptables y de utilidad como un agente contra tumores malignos, en donde se combinan metformina o una de sus sales farmacéuticamente aceptables y dihidroquercetina. o una de sus sales farmacéuticamente aceptables. Reivindicación 11: Un potenciador de una acción contra tumores malignos de metformina o una de sus sales farmacéuticamente aceptables, caracterizado porque comprende dihidroquercetina o una de sus sales farmacéuticamente aceptables como un ingrediente activo. Reivindicación 14: Uso de dihidroquercetina o una de sus sales farmacéuticamente aceptables en combinación con metformina o una de sus sales farmacéuticamente aceptables en la producción de un, medicamento para la prevención o el tratamiento de un tumor maligno.
ARP140102045A 2013-05-24 2014-05-23 Medicamento de metformina y dihidroquercetina AR096402A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2013110278 2013-05-24

Publications (1)

Publication Number Publication Date
AR096402A1 true AR096402A1 (es) 2015-12-30

Family

ID=50980347

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP140102045A AR096402A1 (es) 2013-05-24 2014-05-23 Medicamento de metformina y dihidroquercetina

Country Status (14)

Country Link
US (4) US9808440B2 (es)
EP (1) EP3003296B1 (es)
JP (2) JP6440212B2 (es)
KR (1) KR102182946B1 (es)
CN (1) CN105263484B (es)
AR (1) AR096402A1 (es)
AU (1) AU2014269401A1 (es)
CA (1) CA2912881A1 (es)
HK (1) HK1223304A1 (es)
PH (1) PH12015502616A1 (es)
RU (2) RU2018135973A (es)
SG (1) SG11201509555UA (es)
TW (2) TWI667021B (es)
WO (1) WO2014189152A1 (es)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10468144B2 (en) 2014-08-19 2019-11-05 Nuscale Power, Llc Spent fuel storage rack
CN105330575A (zh) * 2015-10-14 2016-02-17 吉林海格力斯医药生物科技发展有限公司 一种用于治疗放疗、化疗引起的骨髓损伤的化合物
WO2018060959A1 (en) * 2016-09-30 2018-04-05 Laboratorios Silanes S.A. De C.V. Metformin glycinate, pharmaceutical compositions comprising the same, and methods of using the same
CN108078938A (zh) * 2018-01-15 2018-05-29 栾晓民 一种二氢槲皮素制剂的制备方法及应用
CN112888673B (zh) 2018-04-25 2022-07-29 查尔斯德鲁医药科学大学 新颖mct4抑制剂及其用途
KR102349477B1 (ko) * 2019-08-30 2022-01-10 (주)프론트바이오 바이구아나이드 계열 화합물 및 플라본, 하이드록시플라본, 플라바논, 플라본 유도체, 하이드록시플라본 유도체, 플라바논 유도체의 복합제를 유효성분으로 함유하는 암 예방 또는 치료용 약학적 조성물
CA3163122A1 (en) * 2020-02-25 2021-09-02 Aram Oganesian Combination decitabine and cedazuridine solid oral dosage forms
CN111467332B (zh) * 2020-03-31 2021-08-24 中国科学院苏州生物医学工程技术研究所 低温等离子体与二甲双胍联用的应用
RU2740946C1 (ru) * 2020-06-30 2021-01-21 Федеральное государственное бюджетное научное учреждение "Федеральный исследовательский центр фундаментальной и трансляционной медицины" (ФИЦ ФТМ) Средство для снижения патоморфологических изменений при гиперплазии предстательной железы
US20220409567A1 (en) * 2021-06-23 2022-12-29 Thomas Winston Adjuvant and complementary therapies for the treatment of cancer
CN115154458B (zh) * 2022-07-25 2023-11-10 天水师范学院 一种槲皮素-盐酸二甲双胍复合降糖药物的制备方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP3523287B2 (ja) * 1993-02-26 2004-04-26 丸善製薬株式会社 発癌プロモーション抑制剤
US8178123B2 (en) 2001-08-29 2012-05-15 Femina Pharma Incorporated Method for augmentation of intraepithelial and systemic exposure of therapeutic agents having substrate activity for cytochrome P450 enzymes and membrane efflux systems following vaginal and oral cavity administration
CN1320925C (zh) * 2005-03-30 2007-06-13 淮北市辉克药业有限公司 长期使用的治疗糖尿病的复方制剂
CA2606658A1 (en) 2006-10-13 2008-04-13 Mike Tyers Compositions and methods for treating neurological disorders or damage
DE102008029460A1 (de) 2008-06-20 2009-12-31 Otkrytoe Aktsionernoe Obschestvo Zavod Ekologicheskoy Tekhniki I Ekopitaniya 'diod' Taxifolinderivate zur Prophylaxe und Behandlung von neurologischen und psychiatrischen Störungen des zentralen Nervensystems
JP2012505251A (ja) 2008-10-10 2012-03-01 リメリック バイオファーマ, インコーポレイテッド 代謝性疾患の処置のためのピロン
CA2772120A1 (en) * 2009-08-25 2011-03-17 President And Fellows Of Harvard College Use of metformin in cancer treatment and prevention
WO2012122295A2 (en) * 2011-03-07 2012-09-13 Ned Biosystems, Inc. Treatment for pancreatic adenocarcinoma and other cancers of epithelial origin
RU2451506C1 (ru) * 2011-06-02 2012-05-27 Сергей Юрьевич Лешков Комбинация для лечения сахарного диабета и его осложнений
JP5645796B2 (ja) 2011-11-21 2014-12-24 東京エレクトロン株式会社 液処理装置及び液処理方法

Also Published As

Publication number Publication date
CN105263484A (zh) 2016-01-20
KR102182946B1 (ko) 2020-11-25
WO2014189152A1 (en) 2014-11-27
EP3003296B1 (en) 2018-10-10
JP2019048850A (ja) 2019-03-28
TW201536275A (zh) 2015-10-01
US9808440B2 (en) 2017-11-07
TWI667021B (zh) 2019-08-01
HK1223304A1 (zh) 2017-07-28
US10292962B2 (en) 2019-05-21
PH12015502616A1 (en) 2016-02-29
RU2018135973A3 (es) 2022-03-04
AU2014269401A1 (en) 2016-01-21
JP6440212B2 (ja) 2018-12-19
US20160101082A1 (en) 2016-04-14
RU2015155283A (ru) 2017-06-29
TWI688387B (zh) 2020-03-21
US20180036280A1 (en) 2018-02-08
SG11201509555UA (en) 2015-12-30
US20180050014A1 (en) 2018-02-22
CA2912881A1 (en) 2014-11-27
TW201906603A (zh) 2019-02-16
CN105263484B (zh) 2018-08-03
JP6754071B2 (ja) 2020-09-09
JP2016522202A (ja) 2016-07-28
US20180353466A1 (en) 2018-12-13
KR20160013164A (ko) 2016-02-03
EP3003296A1 (en) 2016-04-13
RU2671488C2 (ru) 2018-11-01
RU2018135973A (ru) 2018-11-14

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