AR089881A1 - PIRIMIDINE FUNGICIDE COMPOUNDS - Google Patents
PIRIMIDINE FUNGICIDE COMPOUNDSInfo
- Publication number
- AR089881A1 AR089881A1 ARP130100325A AR089881A1 AR 089881 A1 AR089881 A1 AR 089881A1 AR P130100325 A ARP130100325 A AR P130100325A AR 089881 A1 AR089881 A1 AR 089881A1
- Authority
- AR
- Argentina
- Prior art keywords
- alkyl
- alkoxy
- haloalkoxy
- haloalkyl
- alkynyl
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/32—One oxygen, sulfur or nitrogen atom
- C07D239/42—One nitrogen atom
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Compuestos fungicidas de pirimidina de fórmula (1) como se define en la presente, su uso y métodos para combatir hongos fitopatogénicos. Reivindicación 1: Compuestos de fórmula (1) en donde: Rᵃ⁵ es metilo o halometilo; Rᵃ², Rᵃ⁶ independientemente uno de otro son hidrógeno, halógeno, CN, NO₂, OH, SH, alquilo C₁₋₄, haloalquilo C₁₋₄, alcoxi C₁₋₄, haloalcoxi C₁₋₄, alquiltio C₁₋₄, haloalquiltio C₁₋₄, alquilsulfinilo C₁₋₄, haloalquilsulfinilo C₁₋₄, alquilsulfonilo C₁₋₄, haloalquilsulfonilo C₁₋₄, alcoxi C₁₋₄-alquilo C₁₋₄, alcoxi C₁₋₄-alcoxi C₁₋₄-, alquenilo C₂₋₄-, alquinilo C₂₋₄, haloalquenilo C₂₋₄-, haloalquinilo C₂₋₄-, cicloalquilo C₃₋₈, cicloalquiloxi C₃₋₈, cicloalquil C₃₋₈-alquilo C₁₋₄, NRARB, C(=O)R, C(=NOR)R o C(=NH)-O-R; RA, RB independientemente uno de otro son hidrógeno, alquilo C₁₋₄, alquenilo C₂₋₄, alquinilo C₂₋₄, fenilo, bencilo, cicloalquilo C₃₋₈, cicloalquenilo C₃₋₈ o C(=O)-R; R es hidrógeno, OH, NH₂, alquilo C₁₋₄-, haloalquilo C₁₋₄-, alquenilo C₂₋₄-, alquinilo C₂₋₄-, alcoxi C₁₋₄-, haloalcoxi C₁₋₄-, alquilamino C₁₋₄- o di(alquil C₁₋₄-)amino; R es hidrógeno, alquilo C₁₋₄-, haloalquilo C₁₋₄, alquenilo C₂₋₄-, alquinilo C₂₋₄- o alcoxi C₁₋₄-alquilo C₁₋₄; R es hidrógeno o alquilo C₁₋₄; R es hidrógeno, alquilo C₁₋₄, haloalquilo C₁₋₄, alcoxi C₁₋₄, haloalcoxi C₁₋₄, alcoxi C₁₋₄-alquilo C₁₋₄, haloalcoxi C₁₋₄-alquilo C₁₋₄, alquenilo C₂₋₄, haloalquenilo C₂₋₄, alquinilo C₂₋₄, haloalquinilo C₂₋₄, CN, CH₂CN, NRARB o CH₂-O-C(=O)R; R¹, R² independientemente uno de otro son hidrógeno, halógeno, OH, CN, alquilo C₁₋₄, haloalquilo C₁₋₄, alcoxi C₁₋₄, haloalcoxi C₁₋₄, alcoxi C₁₋₄-alquilo C₁₋₄, haloalcoxi C₁₋₄-alquilo C₁₋₄, alquenilo C₂₋₄, haloalquenilo C₂₋₄, alquinilo C₂₋₄, haloalquinilo C₂₋₄, cicloalquilo C₃₋₈-, cicloalcoxi C₃₋₈, cicloalquil C₃₋₈-alquilo-C₁₋₄, NRARB, C(=O)R, C(=NOR)R, C(=NH)-O-R o bencilo, en donde el resto fenilo de bencilo está no sustituido o transporta 1, 2, 3, 4, ó 5 sustituyentes seleccionados del grupo que consiste en CN, halógeno, alquilo C₁₋₄, haloalquilo C₁₋₄, alcoxi C₁₋₄, haloalcoxi C₁₋₄, (alcoxi C₁₋₄-)carbonilo y di(alquil C₁₋₄)aminocarbonilo, o dos radicales R¹ y R² que están unidos al mismo átomos de carbono forman juntos con dicho átomo de carbono un carbociclo saturado o parcialmente insaturado de 3, 4, 5, 6 ó 7-miembros o un heterociclo saturado o parcialmente insaturado de 3, 4, 5, 6 ó 7-miembros, en donde los átomos del miembro del anillo del heterociclo antes mencionado incluyen además de los átomos de carbono 1, 2, 3 ó 4 heteroátomos seleccionados del grupo de N, O y S, y en donde el ciclo antes mencionado está no sustituido o transporta 1, 2, 3 ó 4 sustituyentes seleccionados de halógeno, CN, OH, SH, alquilo C₁₋₄-, alcoxi C₁₋₄ o alquiltio C₁₋₄; y uno o dos grupos CH₂ de los ciclos antes mencionados pueden ser reemplazados por uno o dos grupos C(=O) o C(=S) respectivamente; n indica el número de sustituyentes Rᵇ en el anillo fenilo y n es 0, 1, 2, 3 ó 4; Rᵇ es halógeno, CN, NO₂, alquilo C₁₋₄-, haloalquilo C₁₋₄-, alcoxi C₁₋₄-, haloalcoxi C₁₋₄-, alquenilo C₂₋₄-, haloalquenilo C₂₋₄-, alquinilo C₂₋₄-, haloalquinilo C₂₋₄-, NRARB, C(=NOR)R o C(=NH)-O-R, siendo posible para n = 2, 3, ó 4 que Rᵇ sean idénticos o diferentes; Het es un heteroarilo de 5 ó 6 miembros, en donde los átomos del miembro del anillo del heteroarilo incluyen además de átomos de carbono 1, 2, 3, o 4 heteroátomos seleccionados del grupo de N, O y S y en donde el heteroarilo está no sustituido o transporta 1, 2, 3 ó 4 grupos Rᶜ idénticos o diferentes: Rᶜ es halógeno, CN, NO₂, alquilo C₁₋₆-, haloalquilo C₁₋₆-, alcoxi C₁₋₆-, haloalcoxi C₁₋₆-, alquiltio C₁₋₆-, haloalquiltio C₁₋₆-, alquilsulfinilo C₁₋₆-, haloalquilsulfinilo C₁₋₆-, alquilsulfonilo C₁₋₆-, haloalquilsulfinilo C₁₋₆-, alcoxi C₁₋₆-alquilo C₁₋₄-, haloalcoxi C₁₋₆-alquilo C₁₋₄-, alquenilo C₂₋₆-, alquinilo C₂₋₆-, NRARB, C(=O)R, C(=NOR)R, C(=NH)-O-R, cicloalquilo C₃₋₈-, cicloalquilo C₃₋₈-alquilo C₁₋₄-, fenilo, fenilalquilo C₁₋₄-, fenoxi, fenoxi-alquilo C₁₋₄ o un heteroarilo de 5 ó 6 miembros, en donde los átomos del miembro del anillo del heteroarilo incluyen además de átomos de carbono 1, 2, 3 ó 4 heteroátomos seleccionados del grupo de N, O y S, y en donde los radicales cíclicos antes mencionados están no sustituidos o transportan 1, 2, 3 ó 4 sustituyentes Rᵈ idénticos o diferentes: Rᵈ es halógeno, CN, alquilo C₁₋₄-, haloalquilo C₁₋₄-, alcoxi C₁₋₄- o haloalcoxi C₁₋₄-; o dos radicales Rᶜ que están unidos a los átomos del miembro del anillo adyacente del grupo Het forman junto con dichos átomos del miembro del anillo un carbociclo o heterociclo fusionado de 5, 6, ó 7 miembros saturado, parcialmente insaturado o aromático, donde los átomos del miembro del anillo del heterociclo fusionado incluyen además de los átomos de carbono 1, 2, 3 ó 4 heteroátomos seleccionados del grupo de N, O y S, y en donde el carbociclo o heterociclo fusionado está no sustituido o trasporta 1, 2, 3 ó 4 grupos radicales Rᵉ idénticos o diferentes: Rᵉ es halógeno, CN, alquilo C₁₋₄-, haloalquilo C₁₋₄-, alcoxi C₁₋₄- o haloalcoxi C₁₋₄-; y sus N-óxidos y sus sales aceptables para uso agrícola.Pyrimidine fungicidal compounds of formula (1) as defined herein, their use and methods to combat phytopathogenic fungi. Claim 1: Compounds of formula (1) wherein: Rᵃ⁵ is methyl or halomethyl; Rᵃ², Rᵃ⁶ independently of one another are hydrogen, halogen, CN, NO₂, OH, SH, C₁₋₄ alkyl, C₁₋₄ haloalkyl, C₁₋₄ alkoxy, C₁₋₄ haloalkoxy, C₁₋₄ alkylthio, C₁₋₄ haloalkylthio, C₁₋₄ alkylsulfinyl, C₁₋₄ haloalkylsulfinyl, C₁₋₄ alkylsulfonyl, C₁₋₄ haloalkylsulfonyl, C₁₋₄ alkoxy-C₁₋₄ alkyl, C₁₋₄ alkoxy-C₁₋₄- alkoxy, C₂₋₄- alkenyl, C₂₋ alkynyl ₄, C₂₋₄- haloalkenyl, C₂₋₄- haloalkynyl, C₃₋₈ cycloalkyl, C₃₋₈ cycloalkyloxy, C₃₋₈ cycloalkyl-C alquilo alkyl, NRARB, C (= O) R, C (= NOR) R or C (= NH) -OR; RA, RB independently of each other are hydrogen, C₁₋₄ alkyl, C₂₋₄ alkenyl, C₂₋₄ alkynyl, phenyl, benzyl, C₃₋₈ cycloalkyl, C₃₋₈ or C (= O) -R cycloalkenyl; R is hydrogen, OH, NH₂, C₁₋₄- alkyl, C₁₋₄- haloalkyl, C₂₋₄- alkenyl, C₂₋₄- alkynyl, C₁₋₄- alkoxy, C₁₋₄- haloalkoxy, C₁₋₄- alkylamino di (C₁₋₄-) alkyl; R is hydrogen, C₁₋₄- alkyl, C₁₋₄ haloalkyl, C₂₋₄- alkenyl, C₂₋₄- alkynyl or C₁₋₄ alkoxy-C₁₋₄ alkyl; R is hydrogen or C₁₋₄ alkyl; R is hydrogen, C₁₋₄ alkyl, C₁₋₄ haloalkyl, C₁₋₄ alkoxy, C₁₋₄ haloalkoxy, C₁₋₄ alkoxy-C₁₋₄ alkyl, C₁₋₄ haloalkoxy-C₁₋₄ alkyl, C₂₋₄ alkenyl, haloalkenyl C₂₋₄, C₂₋₄ alkynyl, C₂₋₄ haloalkynyl, CN, CH₂CN, NRARB or CH₂-OC (= O) R; R¹, R² independently of each other are hydrogen, halogen, OH, CN, C₁₋₄ alkyl, C₁₋₄ haloalkyl, C₁₋₄ alkoxy, C₁₋₄ haloalkoxy, C₁₋₄ alkoxy-C₁₋₄ alkyl, C₁₋₄ haloalkoxy -C₁₋₄ alkyl, C₂₋₄ alkenyl, C₂₋₄ haloalkenyl, C₂₋₄ alkynyl, C₂₋₄ haloalkynyl, C₃₋₈ cycloalkyl, C₃₋₈ cycloalkoxy, C₃₋₈-C-alkylcycloalkyl, NRARB, C (= O) R, C (= NOR) R, C (= NH) -OR or benzyl, wherein the phenyl benzyl moiety is unsubstituted or transports 1, 2, 3, 4, or 5 substituents selected from the group consisting of CN, halogen, C₁₋₄ alkyl, C₁₋₄ haloalkyl, C₁₋₄ alkoxy, C₁₋₄ haloalkoxy, (C₁₋₄- alkoxy) carbonyl and di (C₁₋₄ alkyl) aminocarbonyl, or two radicals R¹ and R² which are attached to the same carbon atoms together form with said carbon atom a saturated or partially unsaturated carbocycle of 3, 4, 5, 6 or 7-members or a satur heterocycle ado or partially unsaturated of 3, 4, 5, 6 or 7-members, wherein the atoms of the heterocycle ring member mentioned above include in addition to carbon atoms 1, 2, 3 or 4 heteroatoms selected from the group of N, O and S, and wherein the above-mentioned cycle is unsubstituted or transports 1, 2, 3 or 4 substituents selected from halogen, CN, OH, SH, C₁₋₄- alkyl, C₁₋₄ alkoxy or C₁₋₄ alkylthio; and one or two CH₂ groups of the aforementioned cycles may be replaced by one or two groups C (= O) or C (= S) respectively; n indicates the number of substituents Rᵇ in the phenyl ring and n is 0, 1, 2, 3 or 4; Rᵇ is halogen, CN, NO₂, C₁₋₄- alkyl, C₁₋₄- haloalkyl, C₁₋₄- alkoxy, C₁₋₄- haloalkoxy, C₂₋₄- alkenyl, C₂₋₄- haloalkenyl, C₂₋₄- alkynyl, haloalkynyl C₂₋₄-, NRARB, C (= NOR) R or C (= NH) -OR, it being possible for n = 2, 3, or 4 that Rᵇ be identical or different; Het is a 5- or 6-membered heteroaryl, wherein the atoms of the heteroaryl ring member include in addition to carbon atoms 1, 2, 3, or 4 heteroatoms selected from the group of N, O and S and wherein the heteroaryl is unsubstituted or transports 1, 2, 3 or 4 identical or different Rᶜ groups: Rᶜ is halogen, CN, NO₂, C₁₋₆- alkyl, C₁₋₆- haloalkyl, C₁₋₆- alkoxy, C₁₋₆- haloalkoxy, alkylthio C₁₋₆-, haloalkylthio C₁₋₆-, alkylsulfinyl C₁₋₆-, haloalkylsulfinyl C₁₋₆-, alkylsulfonyl C₁₋₆-, haloalkylsulfinyl C₁₋₆-, alkoxy C₁₋₆-alkyl C₁₋₄-, haloalkoxy C₁₋₆ -C₁₋₄- alkyl, C₂₋₆- alkenyl, C₂₋₆- alkynyl, NRARB, C (= O) R, C (= NOR) R, C (= NH) -OR, C₃₋₈- cycloalkyl, cycloalkyl C₃₋₈-C₁₋₄- alkyl, phenyl, C₁₋₄- phenylalkyl, phenoxy, phenoxy-C₁₋₄ alkyl or a 5- or 6-membered heteroaryl, wherein the atoms of the hete ring member roaryl also include carbon atoms 1, 2, 3 or 4 heteroatoms selected from the group of N, O and S, and wherein the aforementioned cyclic radicals are unsubstituted or carry 1, 2, 3 or 4 identical or different Rᵈ substituents : Rᵈ is halogen, CN, C₁₋₄- alkyl, C₁₋₄- haloalkyl, C₁₋₄- alkoxy or C₁₋₄- haloalkoxy; or two radicals Rᶜ which are attached to the atoms of the adjacent ring member of the Het group together with said atoms of the ring member a fused carbocycle or heterocycle of 5, 6, or 7 members saturated, partially unsaturated or aromatic, where the atoms of the fused heterocycle ring member include in addition to carbon atoms 1, 2, 3 or 4 heteroatoms selected from the group of N, O and S, and wherein the fused carbocycle or heterocycle is unsubstituted or transports 1, 2, 3 or 4 identical or different Rᵉ radical groups: Rᵉ is halogen, CN, C₁₋₄- alkyl, C₁₋₄- haloalkyl, C₁₋₄- alkoxy or C₁₋₄- haloalkoxy; and its N-oxides and salts acceptable for agricultural use.
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EP12153758 | 2012-02-03 | ||
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AR089881A1 true AR089881A1 (en) | 2014-09-24 |
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ARP130100325 AR089881A1 (en) | 2012-02-03 | 2013-02-01 | PIRIMIDINE FUNGICIDE COMPOUNDS |
ARP130100326 AR089882A1 (en) | 2012-02-03 | 2013-02-01 | PIRIMIDINE FUNGICIDE COMPOUNDS |
ARP130100327 AR089883A1 (en) | 2012-02-03 | 2013-02-01 | PIRIMIDINE FUNGICIDES COMPOUND |
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Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN104684900B (en) * | 2012-10-25 | 2017-04-12 | 沈阳中化农药化工研发有限公司 | Substituted pyrimidine compound and uses thereof |
CA2923101A1 (en) * | 2013-09-16 | 2015-03-19 | Basf Se | Fungicidal pyrimidine compounds |
CN105753791B (en) * | 2014-12-19 | 2019-09-13 | 沈阳中化农药化工研发有限公司 | Substituted uracil compound and application thereof |
CN111789120B (en) * | 2020-07-29 | 2022-04-01 | 湖南省植物保护研究所 | Bactericide imazalil ionic liquid, and preparation method and application thereof |
Family Cites Families (112)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3325503A (en) | 1965-02-18 | 1967-06-13 | Diamond Alkali Co | Polychloro derivatives of mono- and dicyano pyridines and a method for their preparation |
US3296272A (en) | 1965-04-01 | 1967-01-03 | Dow Chemical Co | Sulfinyl- and sulfonylpyridines |
JPS54115388A (en) | 1978-03-01 | 1979-09-07 | Nippon Chemiphar Co Ltd | Acetic acid derivative and its preparation |
GB2059955A (en) | 1979-09-13 | 1981-04-29 | Merck & Co Inc | Process for preparing methylvanillyl ketone |
DE3338292A1 (en) | 1983-10-21 | 1985-05-02 | Basf Ag, 6700 Ludwigshafen | 7-AMINO-AZOLO (1,5-A) -PYRIMIDINE AND FUNGICIDES CONTAINING THEM |
CA1249832A (en) | 1984-02-03 | 1989-02-07 | Shionogi & Co., Ltd. | Azolyl cycloalkanol derivatives and agricultural fungicides |
BR8600161A (en) | 1985-01-18 | 1986-09-23 | Plant Genetic Systems Nv | CHEMICAL GENE, HYBRID, INTERMEDIATE PLASMIDIO VECTORS, PROCESS TO CONTROL INSECTS IN AGRICULTURE OR HORTICULTURE, INSECTICIDE COMPOSITION, PROCESS TO TRANSFORM PLANT CELLS TO EXPRESS A PLANTINIDE TOXIN, PRODUCED BY CULTURES, UNITED BY BACILLA |
DE3545319A1 (en) | 1985-12-20 | 1987-06-25 | Basf Ag | ACRYLIC ACID ESTERS AND FUNGICIDES THAT CONTAIN THESE COMPOUNDS |
MY100846A (en) | 1986-05-02 | 1991-03-15 | Stauffer Chemical Co | Fungicidal pyridyl imidates |
DE3782883T2 (en) | 1986-08-12 | 1993-06-09 | Mitsubishi Chem Ind | PYRIDINE CARBOXAMIDE DERIVATIVES AND THEIR USE AS A FUNGICIDAL AGENT. |
US4895849A (en) | 1986-10-08 | 1990-01-23 | Ube Industries, Ltd. | Aralkylaminopyrimidine compounds which are useful as for producing thereof and insecticides |
DE3642452A1 (en) * | 1986-12-12 | 1988-06-23 | Bayer Ag | SUBSTITUTED 4-AMINO-PYRIMIDINE |
EP0374753A3 (en) | 1988-12-19 | 1991-05-29 | American Cyanamid Company | Insecticidal toxines, genes coding therefor, antibodies binding them, transgenic plant cells and plants expressing these toxines |
DE69034081T2 (en) | 1989-03-24 | 2004-02-12 | Syngenta Participations Ag | Disease resistant transgenic plant |
DE69018772T2 (en) | 1989-11-07 | 1996-03-14 | Pioneer Hi Bred Int | Larvae kill lectins and plant resistance to insects based on them. |
AU628229B2 (en) | 1989-11-10 | 1992-09-10 | Agro-Kanesho Co. Ltd. | Hexahydrotriazine compounds and insecticides |
EP0519211A1 (en) * | 1991-05-17 | 1992-12-23 | Hoechst Schering AgrEvo GmbH | Substituted 4-aminopyrimidine, process for their preparation and their use as parasiticide |
JP2828186B2 (en) | 1991-09-13 | 1998-11-25 | 宇部興産株式会社 | Acrylate-based compounds, their preparation and fungicides |
UA48104C2 (en) | 1991-10-04 | 2002-08-15 | Новартіс Аг | Dna fragment including sequence that codes an insecticide protein with optimization for corn, dna fragment providing directed preferable for the stem core expression of the structural gene of the plant related to it, dna fragment providing specific for the pollen expression of related to it structural gene in the plant, recombinant dna molecule, method for obtaining a coding sequence of the insecticide protein optimized for corn, method of corn plants protection at least against one pest insect |
US5439911A (en) | 1992-12-28 | 1995-08-08 | Shionogi & Co., Ltd. | Aminopyrimidine derivatives and their production and use |
AU677502B2 (en) | 1994-01-07 | 1997-04-24 | Dowelanco | N-(4-pyrimidinyl)amide pesticides |
EP0665225B1 (en) | 1994-02-01 | 1996-11-27 | Ube Industries, Ltd. | 4-Phenethylamino pyrimidine derivative, process for preparing the same and agricultural and horticultural chemical for controlling noxious organisms containing the same |
US5530195A (en) | 1994-06-10 | 1996-06-25 | Ciba-Geigy Corporation | Bacillus thuringiensis gene encoding a toxin active against insects |
DE19518073A1 (en) | 1995-05-17 | 1996-11-21 | Hoechst Ag | Substituted benzyloxycarbonylguanidines, process for their preparation, their use as a medicament or diagnostic agent and medicament containing them |
DE19603576A1 (en) | 1996-02-01 | 1997-08-07 | Bayer Ag | Acylated 4-amino and 4-hydrazinopyrimidines |
JPH1036355A (en) | 1996-07-19 | 1998-02-10 | Ube Ind Ltd | Production of 4-amino-5-chloro-6-(1-fluoroehyl)pyrimidine derivative |
DE19650197A1 (en) | 1996-12-04 | 1998-06-10 | Bayer Ag | 3-thiocarbamoylpyrazole derivatives |
TW460476B (en) | 1997-04-14 | 2001-10-21 | American Cyanamid Co | Fungicidal trifluoromethylalkylamino-triazolopyrimidines |
CN1117074C (en) | 1997-09-18 | 2003-08-06 | 巴斯福股份公司 | Benzamidoxim derivatives, intermediate products and methods for preparing and using them as fungicides |
DE19750012A1 (en) | 1997-11-12 | 1999-05-20 | Bayer Ag | Isothiazole carboxamides |
WO1999027783A1 (en) | 1997-12-04 | 1999-06-10 | Dow Agrosciences Llc | Fungicidal compositions and methods, and compounds and methods for the preparation thereof |
AU2006201959B2 (en) | 1997-12-22 | 2008-09-04 | Bayer Healthcare Llc | Inhibition of Raf Kinase using Substituted Heterocyclic Ureas |
ATE305465T1 (en) | 1998-11-17 | 2005-10-15 | Kumiai Chemical Industry Co | PYRIMIDINYLBENZIMIDAZOLE AND TRIAZINYLBENZIMIDAZOLE DERIVATIVES AND AGRICULT/HORTICULT FUNGICIDES |
IT1303800B1 (en) | 1998-11-30 | 2001-02-23 | Isagro Ricerca Srl | DIPEPTID COMPOUNDS HAVING HIGH FUNGICIDE AND AGRICULTURAL USE. |
JP3417862B2 (en) | 1999-02-02 | 2003-06-16 | 新東工業株式会社 | Silica gel highly loaded with titanium oxide photocatalyst and method for producing the same |
AU770077B2 (en) | 1999-03-11 | 2004-02-12 | Dow Agrosciences Llc | Heterocyclic substituted isoxazolidines and their use as fungicides |
US6586617B1 (en) | 1999-04-28 | 2003-07-01 | Sumitomo Chemical Takeda Agro Company, Limited | Sulfonamide derivatives |
UA73307C2 (en) | 1999-08-05 | 2005-07-15 | Куміаі Кемікал Індастрі Ко., Лтд. | Carbamate derivative and fungicide of agricultural/horticultural destination |
DE10021412A1 (en) | 1999-12-13 | 2001-06-21 | Bayer Ag | Fungicidal active ingredient combinations |
PL202070B1 (en) | 2000-01-25 | 2009-05-29 | Syngenta Participations Ag | Herbicidal composition |
US6376548B1 (en) | 2000-01-28 | 2002-04-23 | Rohm And Haas Company | Enhanced propertied pesticides |
IL167956A (en) | 2000-02-04 | 2009-02-11 | Sumitomo Chemical Co | Isocyanate compound |
KR100581163B1 (en) | 2000-08-25 | 2006-05-22 | 신젠타 파티서페이션즈 아게 | A hybrid Bacillus thuringiensis toxin, a nucleic acid encoding the same and a method for controlling an insect with the same |
BR0114122A (en) | 2000-09-18 | 2003-07-01 | Du Pont | Compound, fungicidal compositions and method of controlling plant diseases caused by fungal plant pathogens |
PT1341534E (en) | 2000-11-17 | 2010-04-14 | Dow Agrosciences | Compounds having fungicidal activity and processes to make and use same |
JP5034142B2 (en) | 2001-04-20 | 2012-09-26 | 住友化学株式会社 | Plant disease control composition |
DE10136065A1 (en) | 2001-07-25 | 2003-02-13 | Bayer Cropscience Ag | pyrazolylcarboxanilides |
AR037228A1 (en) | 2001-07-30 | 2004-11-03 | Dow Agrosciences Llc | ACID COMPOUNDS 6- (ARIL OR HETEROARIL) -4-AMYNOPYCOLINIC, HERBICIDE COMPOSITION THAT UNDERSTANDS AND METHOD TO CONTROL UNWANTED VEGETATION |
FR2828196A1 (en) | 2001-08-03 | 2003-02-07 | Aventis Cropscience Sa | New iodochromone derivatives, useful for the prevention or cure of plant fungal disorders, especially in cereals, vines, fruits, legumes or ornamental plants |
AU2002327096B2 (en) | 2001-08-17 | 2007-11-22 | Sankyo Agro Company, Limited | 3-phenoxy-4-pyridazinol derivative and herbicide composition containing the same |
US7230167B2 (en) | 2001-08-31 | 2007-06-12 | Syngenta Participations Ag | Modified Cry3A toxins and nucleic acid sequences coding therefor |
AU2002361696A1 (en) | 2001-12-17 | 2003-06-30 | Syngenta Participations Ag | Novel corn event |
AU2002354251A1 (en) | 2001-12-21 | 2003-07-09 | Nissan Chemical Industries, Ltd. | Bactericidal composition |
TWI327462B (en) | 2002-01-18 | 2010-07-21 | Sumitomo Chemical Co | Condensed heterocyclic sulfonyl urea compound, a herbicide containing the same, and a method for weed control using the same |
US20030166476A1 (en) | 2002-01-31 | 2003-09-04 | Winemiller Mark D. | Lubricating oil compositions with improved friction properties |
DE10204390A1 (en) | 2002-02-04 | 2003-08-14 | Bayer Cropscience Ag | Disubstituted thiazolylcarboxanilides |
RU2323931C2 (en) | 2002-03-05 | 2008-05-10 | Синджента Партисипейшнс Аг | O-cyclopropylcarboxanilides and application thereof as fungicides |
CN1305852C (en) | 2002-09-19 | 2007-03-21 | 伊莱利利公司 | Diaryl ethers as opioid receptor antagonist |
GB0227966D0 (en) | 2002-11-29 | 2003-01-08 | Syngenta Participations Ag | Organic Compounds |
WO2004083193A1 (en) | 2003-03-17 | 2004-09-30 | Sumitomo Chemical Company, Limited | Amide compound and bactericide composition containing the same |
NZ544367A (en) | 2003-06-25 | 2009-12-24 | Elan Pharm Inc | Combination therapy involving methotrexate for treating rheumatoid arthritis |
MXPA06001320A (en) | 2003-08-01 | 2006-05-04 | Pfizer Prod Inc | 6-menbered heteroaryl compounds for the treatment of neurodegenerative disorders. |
WO2005014534A1 (en) | 2003-08-08 | 2005-02-17 | Transtech Pharma, Inc. | Aryl and heteroaryl compounds, compositions, and methods of use |
TWI355894B (en) | 2003-12-19 | 2012-01-11 | Du Pont | Herbicidal pyrimidines |
US9487519B2 (en) | 2004-03-10 | 2016-11-08 | Basf Se | 5,6-Dialkyl-7-aminotriazolopyrimidines, their preparation and their use for controlling harmful fungi, and compositions comprising these compounds |
AU2005221807A1 (en) | 2004-03-10 | 2005-09-22 | Basf Aktiengesellschaft | 5,6-dialkyl-7-amino-triazolopyrimidines, method for their production, their use for controlling pathogenic fungi and agents containing said compounds |
CN101693695A (en) | 2004-03-30 | 2010-04-14 | 大正制药株式会社 | Pyrimidine derivatives and methods of treatment related to the use thereof |
US7459562B2 (en) | 2004-04-23 | 2008-12-02 | Bristol-Myers Squibb Company | Monocyclic heterocycles as kinase inhibitors |
BRPI0510887A (en) | 2004-06-03 | 2007-12-26 | Du Pont | fungicidal mixture, fungicidal composition and method for controlling plant diseases |
JP2008502636A (en) | 2004-06-18 | 2008-01-31 | ビーエーエスエフ アクチェンゲゼルシャフト | N- (Ortho-phenyl) -1-methyl-3-difluoromethylpyrazole-4-carboxyanilide and their use as fungicides |
DE502005009089D1 (en) | 2004-06-18 | 2010-04-08 | Basf Se | 1-METHYL-3-TRIFLUOROMETHYL-PYRAZOLE-4-CARBOXYLIC ACID (ORTHO-PHENYL) -ANILIDES AND THEIR USE AS FUNGICIDES |
GB0418048D0 (en) | 2004-08-12 | 2004-09-15 | Syngenta Participations Ag | Method for protecting useful plants or plant propagation material |
EP1838718B1 (en) | 2005-01-10 | 2011-06-15 | Pfizer Inc. | Pyrrolopyrazoles, potent kinase inhibitors |
MX2007008410A (en) | 2005-01-14 | 2007-08-21 | Hoffmann La Roche | Thiazole-4-carboxamide derivatives as mglur5 antagonists. |
DE102005007160A1 (en) | 2005-02-16 | 2006-08-24 | Basf Ag | Pyrazolecarboxylic acid anilides, process for their preparation and compositions containing them for controlling harmful fungi |
ATE400576T1 (en) | 2005-02-16 | 2008-07-15 | Basf Se | 5-ALKOXYALKYL-6-ALKYL-7-AMINO-AZOLOPYRIMIDINES, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE FOR CONTROLLING HARMFUL FUNGALS AND AGENTS CONTAINING SAME |
DE102005009458A1 (en) | 2005-03-02 | 2006-09-07 | Bayer Cropscience Ag | pyrazolylcarboxanilides |
JP2008533018A (en) | 2005-03-09 | 2008-08-21 | シェーリング コーポレイション | Condensed thieno [2,3-b] pyridine compounds and condensed thiazolo [5,4-b] pyridine compounds for inhibiting KSP kinesin activity |
US20070021435A1 (en) | 2005-06-10 | 2007-01-25 | Gaul Michael D | Aminopyrimidines as kinase modulators |
GB0513841D0 (en) | 2005-07-07 | 2005-08-10 | Medivir Ab | Cysteine protease inhibitors |
CA2619402C (en) | 2005-08-15 | 2015-02-03 | Boehringer Ingelheim International Gmbh | Method for producing betamimetics |
GB0516705D0 (en) | 2005-08-15 | 2005-09-21 | Syngenta Participations Ag | Process |
JP5243960B2 (en) | 2005-10-21 | 2013-07-24 | ダウ アグロサイエンシィズ エルエルシー | Thieno-pyrimidine compounds having bactericidal activity |
EP1971583B1 (en) | 2005-12-20 | 2015-03-25 | Incyte Corporation | N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase |
CN102731381B (en) | 2006-01-13 | 2016-08-17 | 美国陶氏益农公司 | The polysubstituted aryl of 6-()-4-aminopyridine formic acid esters and the purposes as herbicide thereof |
EP1983832A2 (en) | 2006-02-09 | 2008-10-29 | Syngeta Participations AG | A method of protecting a plant propagation material, a plant, and/or plant organs |
WO2007096647A2 (en) | 2006-02-27 | 2007-08-30 | Sterix Limited | Diaryl compounds as non-steroidal inhibitors of 17-beta hydroxysteroid dehydrogenase and/or steroid sulphatase for the treatment of oestrogen-related diseases such as hormone dependent breast cancer |
US7989500B2 (en) | 2006-09-15 | 2011-08-02 | Reviva Pharmaceuticals, Inc. | Synthesis, methods of using, and compositions of cycloalkylmethylamines |
US8779154B2 (en) | 2006-09-26 | 2014-07-15 | Qinglin Che | Fused ring compounds for inflammation and immune-related uses |
WO2008039882A1 (en) | 2006-09-30 | 2008-04-03 | Sanofi-Aventis U.S. Llc | A combination of niacin and a prostaglandin d2 receptor antagonist |
ES2302447B1 (en) | 2006-10-20 | 2009-06-12 | Laboratorios Almirall S.A. | DERIVATIVES OF 4- (2-AMINO-1-HYDROXYETHYL) Phenol as agonists of the BETA2 ADRENERGIC RECEIVER. |
TW200831488A (en) | 2006-11-29 | 2008-08-01 | Astrazeneca Ab | Novel compounds |
PE20081559A1 (en) | 2007-01-12 | 2008-11-20 | Merck & Co Inc | SPIROCHROMANONE DERIVATIVES SUBSTITUTED AS ACETYL COA CARBOXYLASE INHIBITORS |
WO2008124757A1 (en) | 2007-04-10 | 2008-10-16 | Bristol-Myers Squibb Company | Thiazolyl compounds useful as kinase inhibitors |
JP5478488B2 (en) | 2007-06-20 | 2014-04-23 | メルク・シャープ・アンド・ドーム・コーポレーション | JANUS kinase inhibitors |
JP5749017B2 (en) | 2008-01-22 | 2015-07-15 | ダウ アグロサイエンシィズ エルエルシー | 5-Fluoropyrimidine derivatives |
SI2303846T1 (en) | 2008-06-24 | 2015-08-31 | Sanofi | Substituted isoquinolines and isoquinolinones as rho kinase inhibitors |
DE102008040168A1 (en) | 2008-07-04 | 2010-01-07 | Robert Bosch Gmbh | Solenoid valve for a fuel injector and fuel injector |
US20100068197A1 (en) | 2008-07-11 | 2010-03-18 | Myriad Pharmaceuticals, Inc. | Pharmaceutical compounds as inhibitors of cell proliferation and the use thereof |
US8268843B2 (en) | 2008-08-29 | 2012-09-18 | Dow Agrosciences, Llc. | 5,8-difluoro-4-(2-(4-(heteroaryloxy)-phenyl)ethylamino)quinazolines and their use as agrochemicals |
EP2344458A1 (en) | 2008-09-11 | 2011-07-20 | Pfizer Inc. | Heteroaryls amide derivatives and their use as glucokinase activators |
TW201024281A (en) | 2008-11-24 | 2010-07-01 | Boehringer Ingelheim Int | New compounds |
EP2210890A1 (en) | 2009-01-19 | 2010-07-28 | Almirall, S.A. | Oxadiazole derivatives as S1P1 receptor agonists |
BRPI1011657A2 (en) | 2009-05-28 | 2019-04-16 | Novartis Ag | substituted aminopropionic derivatives as neprilysin inhibitors |
US8461164B2 (en) | 2009-08-31 | 2013-06-11 | Dow Agrosciences, Llc. | Pteridines and their use as agrochemicals |
NZ597911A (en) | 2009-08-31 | 2014-06-27 | Dow Agrosciences Llc | Pteridines and their use as agrochemicals |
NZ598809A (en) | 2009-09-01 | 2014-02-28 | Dow Agrosciences Llc | Synergistic fungicidal compositions containing a 5-fluoropyrimidine derivative for fungal control in cereals |
WO2011032277A1 (en) | 2009-09-18 | 2011-03-24 | Boehringer Ingelheim International Gmbh | Quinazolinone derivatives as viral polymerase inhibitors |
WO2011053835A1 (en) | 2009-10-30 | 2011-05-05 | Aton Pharma, Inc. | Stereoselective synthesis of metyrosine |
AU2011205283B2 (en) | 2010-01-13 | 2014-07-10 | Tempero Pharmaceuticals, Inc. | Compounds and methods |
JP2013519673A (en) | 2010-02-10 | 2013-05-30 | レクシコン ファーマシューティカルズ インコーポレイテッド | Tryptophan hydroxylase inhibitors for the treatment of metastatic bone disease |
CN102260263A (en) | 2010-05-26 | 2011-11-30 | 四川大学 | Diphenylamine purine derivatives, and preparation method and medicinal application thereof |
-
2013
- 2013-01-31 WO PCT/EP2013/051855 patent/WO2013113788A1/en active Application Filing
- 2013-01-31 WO PCT/EP2013/051854 patent/WO2013113787A1/en active Application Filing
- 2013-01-31 WO PCT/EP2013/051859 patent/WO2013113791A1/en active Application Filing
- 2013-02-01 AR ARP130100325 patent/AR089881A1/en unknown
- 2013-02-01 AR ARP130100326 patent/AR089882A1/en unknown
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WO2013113791A1 (en) | 2013-08-08 |
WO2013113787A1 (en) | 2013-08-08 |
AR089882A1 (en) | 2014-09-24 |
WO2013113788A1 (en) | 2013-08-08 |
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