AR082560A1 - Forma de dosificacion farmaceutica que comprende 6’-fluoro-(n-metil- o n,n-dimetil)-4-fenil-4’,9’-dihidro-3’h-espiro[ciclohexan-1,1’-pirano[3,4,b]indol]-4-amina - Google Patents

Forma de dosificacion farmaceutica que comprende 6’-fluoro-(n-metil- o n,n-dimetil)-4-fenil-4’,9’-dihidro-3’h-espiro[ciclohexan-1,1’-pirano[3,4,b]indol]-4-amina

Info

Publication number
AR082560A1
AR082560A1 ARP110102820A ARP110102820A AR082560A1 AR 082560 A1 AR082560 A1 AR 082560A1 AR P110102820 A ARP110102820 A AR P110102820A AR P110102820 A ARP110102820 A AR P110102820A AR 082560 A1 AR082560 A1 AR 082560A1
Authority
AR
Argentina
Prior art keywords
fluoro
phenyl
methyl
dosage form
pharmaceutical dosage
Prior art date
Application number
ARP110102820A
Other languages
English (en)
Inventor
Grning Nadja Dr
Schiller Marc Dr
Friedrich Ingo Dr
Kirby Chris Dr
Original Assignee
Gruenenthal Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43481034&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR082560(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gruenenthal Gmbh filed Critical Gruenenthal Gmbh
Publication of AR082560A1 publication Critical patent/AR082560A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/145—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/146—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Indole Compounds (AREA)

Abstract

Forma de dosificación farmacéutica para administración dos veces al día, una vez al día o con menor frecuencia, la cual contiene 6’-fluoro-(N-metil- o N,N-dimetil)-4-fenil-4’,9’-dihidro-3’H-espiro[ciclohexan-1,1’-pirano[3,4,b]indol]-4-amina o una sal fisiológicamente aceptable de la misma.
ARP110102820A 2010-08-04 2011-08-04 Forma de dosificacion farmaceutica que comprende 6’-fluoro-(n-metil- o n,n-dimetil)-4-fenil-4’,9’-dihidro-3’h-espiro[ciclohexan-1,1’-pirano[3,4,b]indol]-4-amina AR082560A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP10008116 2010-08-04

Publications (1)

Publication Number Publication Date
AR082560A1 true AR082560A1 (es) 2012-12-19

Family

ID=43481034

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP110102820A AR082560A1 (es) 2010-08-04 2011-08-04 Forma de dosificacion farmaceutica que comprende 6’-fluoro-(n-metil- o n,n-dimetil)-4-fenil-4’,9’-dihidro-3’h-espiro[ciclohexan-1,1’-pirano[3,4,b]indol]-4-amina

Country Status (28)

Country Link
EP (1) EP2600839B1 (es)
JP (1) JP5792300B2 (es)
KR (1) KR101828768B1 (es)
CN (1) CN103179953A (es)
AR (1) AR082560A1 (es)
AU (1) AU2011287956B2 (es)
BR (1) BR112013002714A2 (es)
CA (1) CA2804878C (es)
CL (1) CL2012003582A1 (es)
CO (1) CO6640315A2 (es)
CY (1) CY1119887T1 (es)
DK (1) DK2600839T3 (es)
EC (1) ECSP13012419A (es)
ES (1) ES2665344T3 (es)
HR (1) HRP20180143T1 (es)
HU (1) HUE035543T2 (es)
IL (1) IL223880A (es)
LT (1) LT2600839T (es)
MX (1) MX345068B (es)
NZ (1) NZ604735A (es)
PE (1) PE20131107A1 (es)
PL (1) PL2600839T3 (es)
PT (1) PT2600839T (es)
RS (1) RS57027B1 (es)
RU (1) RU2582390C2 (es)
SI (1) SI2600839T1 (es)
WO (1) WO2012016699A2 (es)
ZA (1) ZA201300038B (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK3247352T3 (da) * 2015-01-23 2020-09-07 Gruenenthal Gmbh Cebranopadol til behandling af smerter hos individer med forringet lever- og/eller forringet nyrefunktion
BR112018017167A2 (pt) 2016-02-29 2019-01-02 Gruenenthal Gmbh titulação de cebranopadol
WO2024129782A1 (en) 2022-12-12 2024-06-20 Park Therapeutics, Inc. Regimens and compositions useful for alleviating pain

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR038681A1 (es) * 2002-02-14 2005-01-26 Solvay Pharm Bv Formulacion oral de solucion solida de una sustancia activa pobremente soluble en agua
DE10252667A1 (de) * 2002-11-11 2004-05-27 Grünenthal GmbH Spirocyclische Cyclohexan-Derivate
DE102005005446A1 (de) * 2005-02-04 2006-08-10 Grünenthal GmbH Bruchfeste Darreichungsformen mit retardierter Freisetzung
US20070048228A1 (en) * 2003-08-06 2007-03-01 Elisabeth Arkenau-Maric Abuse-proofed dosage form
DE102006046745A1 (de) * 2006-09-29 2008-04-03 Grünenthal GmbH Gemischte ORL1/µ-Agonisten zur Behandlung von Schmerz
DE102007009235A1 (de) * 2007-02-22 2008-09-18 Grünenthal GmbH Spirocyclische Cyclohexan-Derivate

Also Published As

Publication number Publication date
CL2012003582A1 (es) 2013-06-07
RU2582390C2 (ru) 2016-04-27
ZA201300038B (en) 2013-09-25
WO2012016699A8 (en) 2013-02-07
KR101828768B1 (ko) 2018-02-13
AU2011287956B2 (en) 2015-01-22
AU2011287956A8 (en) 2014-09-25
SI2600839T1 (en) 2018-04-30
PE20131107A1 (es) 2013-10-17
EP2600839B1 (en) 2018-01-10
DK2600839T3 (da) 2018-01-29
LT2600839T (lt) 2018-03-26
ES2665344T3 (es) 2018-04-25
CA2804878A1 (en) 2012-02-09
NZ604735A (en) 2014-08-29
CA2804878C (en) 2019-01-08
JP2013532698A (ja) 2013-08-19
IL223880A (en) 2017-01-31
HUE035543T2 (en) 2018-05-28
CN103179953A (zh) 2013-06-26
CY1119887T1 (el) 2018-06-27
MX2013001114A (es) 2013-03-12
BR112013002714A2 (pt) 2017-05-30
AU2011287956A1 (en) 2013-01-10
KR20130135238A (ko) 2013-12-10
PT2600839T (pt) 2018-04-17
ECSP13012419A (es) 2013-03-28
RU2013109134A (ru) 2014-09-10
WO2012016699A2 (en) 2012-02-09
CO6640315A2 (es) 2013-03-22
PL2600839T3 (pl) 2018-07-31
WO2012016699A3 (en) 2012-08-16
HRP20180143T1 (hr) 2018-02-23
RS57027B1 (sr) 2018-05-31
MX345068B (es) 2017-01-16
JP5792300B2 (ja) 2015-10-07
EP2600839A2 (en) 2013-06-12

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