AR074770A1 - Producto que contiene nicotina - Google Patents

Producto que contiene nicotina

Info

Publication number
AR074770A1
AR074770A1 ARP090104938A ARP090104938A AR074770A1 AR 074770 A1 AR074770 A1 AR 074770A1 AR P090104938 A ARP090104938 A AR P090104938A AR P090104938 A ARP090104938 A AR P090104938A AR 074770 A1 AR074770 A1 AR 074770A1
Authority
AR
Argentina
Prior art keywords
nicotine
product
pharmaceutically acceptable
preparation
weight
Prior art date
Application number
ARP090104938A
Other languages
English (en)
Original Assignee
Siegfried Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Siegfried Ltd filed Critical Siegfried Ltd
Publication of AR074770A1 publication Critical patent/AR074770A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/56Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule
    • A61K47/58Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. poly[meth]acrylate, polyacrylamide, polystyrene, polyvinylpyrrolidone, polyvinylalcohol or polystyrene sulfonic acid resin
    • A61K47/585Ion exchange resins, e.g. polystyrene sulfonic acid resin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/34Tobacco-abuse
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • A61K9/0058Chewing gums
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/70Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023Transdermal patches and similar drug-containing composite devices, e.g. cataplasms

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

La presente se refiere a un producto que contiene nicotina que comprende un sustrato polimérico farmacéuticamente aceptable, el cual es capaz de unirse a cationes, nicotina o un derivado de nicotina farmacéuticamente aceptable, y cationes inorgánicos farmacéuticamente aceptables. También se refiere a un método para la preparación de dicho producto que contiene nicotina y a su uso para la preparación de un producto farmacéutico. Reivindicación 2: Producto que contiene nicotina de acuerdo con la reivindicación 1, caracterizado en que el sustrato polimérico farmacéuticamente aceptable se selecciona del grupo que consiste en resinas de intercambio catiónico y polisacáridos. Reivindicación 6: Producto que contiene nicotina de acuerdo con una de las reivindicaciones 1 a 5, caracterizado en que comprende menos de 20% en peso de nicotina o el derivado de nicotina farmacéuticamente aceptable, preferentemente 8-18% en peso, más preferentemente 10-15% en peso. Reivindicación 8: Producto que contiene nicotina de acuerdo con una de las reivindicaciones 1 a 7, caracterizado en que el catión inorgánico farmacéuticamente aceptable se selecciona del grupo que consiste en Li+, K+, Na+, Mg2+, Ca2+, Fe2+, Zn2+ y mezclas de los mismos. Reivindicación 14: Uso de un producto que contiene nicotina de acuerdo con una de las reivindicaciones 1 a 9 para la preparación de un producto farmacéutico que contiene nicotina destinado para la administración oral. Reivindicación 15: Uso de un producto que contiene nicotina de acuerdo con una de las reivindicaciones 1 a 9 para la preparación de un producto farmacéutico que contiene nicotina destinado para la administración transdérmica.
ARP090104938A 2008-12-19 2009-12-17 Producto que contiene nicotina AR074770A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP08022123A EP2198865B1 (en) 2008-12-19 2008-12-19 Nicotine-containing product

Publications (1)

Publication Number Publication Date
AR074770A1 true AR074770A1 (es) 2011-02-09

Family

ID=40602533

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP090104938A AR074770A1 (es) 2008-12-19 2009-12-17 Producto que contiene nicotina

Country Status (17)

Country Link
US (1) US9585967B2 (es)
EP (2) EP2392331A1 (es)
AR (1) AR074770A1 (es)
AT (1) ATE533487T1 (es)
AU (1) AU2009328589B2 (es)
CA (1) CA2734403C (es)
DK (1) DK2198865T3 (es)
ES (1) ES2377673T3 (es)
HR (1) HRP20110954T1 (es)
MX (1) MX2011003942A (es)
NZ (1) NZ591209A (es)
PL (1) PL2198865T3 (es)
PT (1) PT2198865E (es)
SI (1) SI2198865T1 (es)
UY (1) UY32337A (es)
WO (1) WO2010069507A1 (es)
ZA (1) ZA201101124B (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11911375B2 (en) * 2020-11-16 2024-02-27 Fertin Pharma A/S Solid oral nicotine formulation

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3901248A (en) 1970-07-22 1975-08-26 Leo Ab Chewable smoking substitute composition
GB1332503A (en) * 1970-10-15 1973-10-03 British American Tobacco Co Smoking compositions
US3845217A (en) * 1972-11-16 1974-10-29 Helsingborg L Ab Buffered smoking substitute compositions
IT1104351B (it) * 1978-06-14 1985-10-21 Muzzarelli Riccardo Il complesso glucano chitosano il metodo della sua produzione a partire da muffe funghi e lieviti e i suoi usi
GB9310412D0 (en) 1993-05-20 1993-07-07 Danbiosyst Uk Nasal nicotine system
GB2385288A (en) 2002-01-18 2003-08-20 Advanced Phytonics Ltd Preparing a resinate.
US6586449B1 (en) 2002-05-28 2003-07-01 Cambrex Charles City, Inc. Nicotine-containing, controlled release composition and method
US20050123502A1 (en) * 2003-10-07 2005-06-09 Chan Shing Y. Nicotine containing oral compositions
ATE439839T1 (de) 2003-12-02 2009-09-15 Fertin Pharma As Nikotin-abgabeprodukt und herstellungsverfahren
US20070269386A1 (en) * 2006-05-16 2007-11-22 Per Steen New product and use and manufacture thereof
US20070269492A1 (en) * 2006-05-16 2007-11-22 Per Steen New product and use and manufacture thereof
ES2401912T3 (es) * 2008-09-17 2013-04-25 Siegfried Ltd. Granulado que contiene nicotina

Also Published As

Publication number Publication date
DK2198865T3 (da) 2012-01-16
ATE533487T1 (de) 2011-12-15
ES2377673T3 (es) 2012-03-29
CA2734403A1 (en) 2010-06-24
PL2198865T3 (pl) 2012-04-30
CA2734403C (en) 2013-05-14
AU2009328589A1 (en) 2010-06-24
EP2198865B1 (en) 2011-11-16
AU2009328589B2 (en) 2012-12-06
US20110207782A1 (en) 2011-08-25
EP2198865A1 (en) 2010-06-23
SI2198865T1 (sl) 2012-02-29
NZ591209A (en) 2012-11-30
EP2392331A1 (en) 2011-12-07
MX2011003942A (es) 2011-05-19
HRP20110954T1 (hr) 2012-01-31
PT2198865E (pt) 2012-02-07
ZA201101124B (en) 2012-05-30
UY32337A (es) 2010-07-30
WO2010069507A1 (en) 2010-06-24
US9585967B2 (en) 2017-03-07

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