AR065670A1 - Combinacion de metformina r-(+) lipoato y agentes antihiperlipidemicos para el tratamiento de hiperglucemia diabetica y complicaciones diabeticas - Google Patents
Combinacion de metformina r-(+) lipoato y agentes antihiperlipidemicos para el tratamiento de hiperglucemia diabetica y complicaciones diabeticasInfo
- Publication number
- AR065670A1 AR065670A1 ARP080100977A ARP080100977A AR065670A1 AR 065670 A1 AR065670 A1 AR 065670A1 AR P080100977 A ARP080100977 A AR P080100977A AR P080100977 A ARP080100977 A AR P080100977A AR 065670 A1 AR065670 A1 AR 065670A1
- Authority
- AR
- Argentina
- Prior art keywords
- diabetic
- lipoate
- metformin
- treatment
- pharmaceutical composition
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
- A61K31/385—Heterocyclic compounds having sulfur as a ring hetero atom having two or more sulfur atoms in the same ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
- A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Diabetes (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Endocrinology (AREA)
- Emergency Medicine (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Composiciones farmacéuticas, métodos y kits, que comprenden metformina R-(+) lipoato y un agente antihiperlipidémico o una sal, hidrato, solvato y prodroga derivada de la misma farmacéuticamente aceptable para el tratamiento de hiperglucemiadiabética Tipo 2 y las complicaciones diabéticas. Reivindicacion 1: Una composicion farmacéutica caracterizada porque comprende metformina R-(+) lipoato [MR-(+)LA], y un inhibidor reductasa HMG-CoA o una sal aceptable en términos farmacéuticos,hidrato, solvato o un profármaco derivado de estos. Reivindicacion 7: La composicion farmacéutica de la reivindicacion 4 caracterizada porque el inhibidor reductasa HMG-CoA es atorvastatina cálcica. Reivindicacion 14: La composicion farmacéuticade la reivindicacion 3 caracterizada porque el inhibidor reductasa HMG-CoA es simvastatina, o una sal de esta aceptable en términos farmacéuticos. Reivindicacion 23: La composicion farmacéutica de la reivindicacion 22, caracterizada porque elinhibidor de absorcion de colesterol es ezetimibe, o una sal aceptable en términos farmacéuticos, hidrato, solvato y un profármaco derivado de éste.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US90599007P | 2007-03-09 | 2007-03-09 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR065670A1 true AR065670A1 (es) | 2009-06-24 |
Family
ID=39760278
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP080100977A AR065670A1 (es) | 2007-03-09 | 2008-03-07 | Combinacion de metformina r-(+) lipoato y agentes antihiperlipidemicos para el tratamiento de hiperglucemia diabetica y complicaciones diabeticas |
Country Status (5)
Country | Link |
---|---|
EP (1) | EP2134169A2 (es) |
AR (1) | AR065670A1 (es) |
CL (1) | CL2008000684A1 (es) |
TW (1) | TW200901959A (es) |
WO (1) | WO2008112166A2 (es) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2009085223A1 (en) * | 2007-12-20 | 2009-07-09 | Indigene Pharmaceuticals, Inc. | Combination of metformin r-(+)-lipoate and antihyperglycemic agents for the treatment of diabetic hyperglycemia and diabetic complications |
WO2012073256A1 (en) * | 2010-11-29 | 2012-06-07 | Cadila Healthcare Limited | Salts of rosuvastatin |
WO2015001568A2 (en) * | 2013-07-01 | 2015-01-08 | Laurus Labs Private Limited | Sitagliptin lipoate salt, process for the preparation and pharmaceutical composition thereof |
US10166246B2 (en) | 2014-05-27 | 2019-01-01 | City Of Hope | TGR5 agonist complexes for treating diabetes and cancer |
MX2021002090A (es) * | 2018-08-24 | 2021-04-28 | Esperion Therapeutics Inc | Metodos para reducir el riesgo de diabetes en pacientes que son tratados por enfermedades relacionadas con el colesterol alto. |
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-
2008
- 2008-03-07 TW TW097108037A patent/TW200901959A/zh unknown
- 2008-03-07 AR ARP080100977A patent/AR065670A1/es unknown
- 2008-03-07 WO PCT/US2008/003094 patent/WO2008112166A2/en active Application Filing
- 2008-03-07 EP EP08726603A patent/EP2134169A2/en not_active Withdrawn
- 2008-03-07 CL CL200800684A patent/CL2008000684A1/es unknown
Also Published As
Publication number | Publication date |
---|---|
EP2134169A2 (en) | 2009-12-23 |
WO2008112166A3 (en) | 2008-10-30 |
WO2008112166A2 (en) | 2008-09-18 |
CL2008000684A1 (es) | 2008-08-01 |
TW200901959A (en) | 2009-01-16 |
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