AR057123A1 - Composicion farmaceutica estable que contiene una pirimidina-sulfamida - Google Patents

Composicion farmaceutica estable que contiene una pirimidina-sulfamida

Info

Publication number
AR057123A1
AR057123A1 ARP060103943A ARP060103943A AR057123A1 AR 057123 A1 AR057123 A1 AR 057123A1 AR P060103943 A ARP060103943 A AR P060103943A AR P060103943 A ARP060103943 A AR P060103943A AR 057123 A1 AR057123 A1 AR 057123A1
Authority
AR
Argentina
Prior art keywords
pharmaceutical composition
sulfamide
pyrimidine
composition containing
stable pharmaceutical
Prior art date
Application number
ARP060103943A
Other languages
English (en)
Original Assignee
Actelion Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26070369&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR057123(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Actelion Pharmaceuticals Ltd filed Critical Actelion Pharmaceuticals Ltd
Publication of AR057123A1 publication Critical patent/AR057123A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner

Abstract

Reivindicacion 1: Una composicion farmacéutica que comprende: a) un compuesto de la formula (1), o una sal, solvato, hidrato o forma morfologica farmacéuticamente aceptable de éste, b) relleno, c) un desintegrante, d) un agente tensoactivo, y e) un lubricante. Reivindicacion 16: El uso de un compuesto de la formula (1) como se define en la reivindicacion 1, o una sal, un solvato, un hidrato o una forma morfologica de éste, para la preparacion de un medicamento, para ser utilizado en el tratamiento de hipertension arterial pulmonar.
ARP060103943A 1999-05-22 2006-09-11 Composicion farmaceutica estable que contiene una pirimidina-sulfamida AR057123A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP9903532 1999-05-22
US09/573,504 US6316453B1 (en) 1999-05-22 2000-05-18 Aqueous pharmaceutical composition

Publications (1)

Publication Number Publication Date
AR057123A1 true AR057123A1 (es) 2007-11-14

Family

ID=26070369

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP060103943A AR057123A1 (es) 1999-05-22 2006-09-11 Composicion farmaceutica estable que contiene una pirimidina-sulfamida

Country Status (12)

Country Link
US (1) US6316453B1 (es)
EP (1) EP1060749B1 (es)
JP (1) JP4632385B2 (es)
AR (1) AR057123A1 (es)
AT (1) ATE235255T1 (es)
CA (1) CA2308660C (es)
DE (1) DE60001768T2 (es)
DK (1) DK1060749T3 (es)
ES (1) ES2195818T3 (es)
NZ (1) NZ504671A (es)
PT (1) PT1060749E (es)
ZA (1) ZA200002318B (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7528065B2 (en) * 2006-01-17 2009-05-05 International Business Machines Corporation Structure and method for MOSFET gate electrode landing pad

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW313568B (es) * 1994-12-20 1997-08-21 Hoffmann La Roche
EP0897914B1 (en) * 1997-08-19 2004-05-26 F. Hoffmann-La Roche Ag Process for the preparation of 2,5-disubstitued pyridines

Also Published As

Publication number Publication date
EP1060749A1 (en) 2000-12-20
PT1060749E (pt) 2003-08-29
JP4632385B2 (ja) 2011-02-16
ES2195818T3 (es) 2003-12-16
DE60001768T2 (de) 2003-10-16
ZA200002318B (en) 2000-11-16
US6316453B1 (en) 2001-11-13
NZ504671A (en) 2001-11-30
JP2001002564A (ja) 2001-01-09
CA2308660A1 (en) 2000-11-22
CA2308660C (en) 2008-08-12
DE60001768D1 (de) 2003-04-30
DK1060749T3 (da) 2003-06-23
ATE235255T1 (de) 2003-04-15
EP1060749B1 (en) 2003-03-26

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Legal Events

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