AR056013A1 - Hemifumarato de derivado de piperidina - Google Patents
Hemifumarato de derivado de piperidinaInfo
- Publication number
- AR056013A1 AR056013A1 ARP060103359A ARP060103359A AR056013A1 AR 056013 A1 AR056013 A1 AR 056013A1 AR P060103359 A ARP060103359 A AR P060103359A AR P060103359 A ARP060103359 A AR P060103359A AR 056013 A1 AR056013 A1 AR 056013A1
- Authority
- AR
- Argentina
- Prior art keywords
- hemifumarate
- solvate
- piperidine derivative
- salt
- chlorobenzyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/56—Nitrogen atoms
- C07D211/58—Nitrogen atoms attached in position 4
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4468—Non condensed piperidines, e.g. piperocaine having a nitrogen directly attached in position 4, e.g. clebopride, fentanyl
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/007—Pulmonary tract; Aromatherapy
- A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
- A61K9/0075—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Otolaryngology (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Medicinal Preparation (AREA)
Abstract
Hemifumarato de N-{2-[((2S)-3-{[1-(4-clorobencil)piperidin-4-il]amino}-2-hidroxi-2-metilpropil)oxi]-4-hidroxifenil}acetamida, o un solvato del mismo, composiciones farmacéuticas que contienen la sal o el solvato y uso de la sal o el solvato en terapias. Reivindicacion 3: El compuesto de acuerdo con la cláusula 2, caracterizado porque exhibe al menos los siguientes picos característicos de difraccion por rayos X de polvo (expresados en grados 2(Theta): a) 6,2, 10,7 y 12,5; o 6,2, 10,7 y 18,8; o c) 6,2, 10,7 y 18,0; o d) 6,2, 10,7, 12,5, 18,0 y 18,8; o e) 6,2, 10,7, 12,5, 18,0, 18,8, 19,7 y 19,8.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE0501769 | 2005-08-02 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR056013A1 true AR056013A1 (es) | 2007-09-12 |
Family
ID=37708913
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP060103359A AR056013A1 (es) | 2005-08-02 | 2006-08-02 | Hemifumarato de derivado de piperidina |
Country Status (16)
Country | Link |
---|---|
US (1) | US20080176902A1 (es) |
EP (1) | EP1912944A1 (es) |
JP (1) | JP2009503066A (es) |
KR (1) | KR20080031370A (es) |
CN (1) | CN101238104A (es) |
AR (1) | AR056013A1 (es) |
AU (1) | AU2006276346A1 (es) |
BR (1) | BRPI0614535A2 (es) |
CA (1) | CA2617406A1 (es) |
IL (1) | IL188484A0 (es) |
MX (1) | MX2008001114A (es) |
NO (1) | NO20081079L (es) |
TW (1) | TW200734305A (es) |
UY (1) | UY29713A1 (es) |
WO (1) | WO2007015668A1 (es) |
ZA (1) | ZA200800488B (es) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AR028948A1 (es) * | 2000-06-20 | 2003-05-28 | Astrazeneca Ab | Compuestos novedosos |
TW200738634A (en) * | 2005-08-02 | 2007-10-16 | Astrazeneca Ab | New salt |
GB0814729D0 (en) * | 2008-08-12 | 2008-09-17 | Argenta Discovery Ltd | New combination |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE69938193D1 (de) * | 1998-11-20 | 2008-04-03 | Hoffmann La Roche | Piperidin ccr-3 rezeptor-hemmer |
CO5300399A1 (es) * | 2000-02-25 | 2003-07-31 | Astrazeneca Ab | Heterocicliocs que contienen nitrogeno, proceso para su preparacion y composiciones farmaceuticas que los contienen |
GB0012260D0 (en) * | 2000-05-19 | 2000-07-12 | Astrazeneca Ab | Novel composition |
AR028948A1 (es) * | 2000-06-20 | 2003-05-28 | Astrazeneca Ab | Compuestos novedosos |
AR028947A1 (es) * | 2000-06-20 | 2003-05-28 | Astrazeneca Ab | Compuestos novedosos |
GB0021670D0 (en) * | 2000-09-04 | 2000-10-18 | Astrazeneca Ab | Chemical compounds |
SE0104251D0 (sv) * | 2001-12-14 | 2001-12-14 | Astrazeneca Ab | Novel compounds |
TW200303304A (en) * | 2002-02-18 | 2003-09-01 | Astrazeneca Ab | Chemical compounds |
-
2006
- 2006-07-25 TW TW095127080A patent/TW200734305A/zh unknown
- 2006-07-31 AU AU2006276346A patent/AU2006276346A1/en not_active Abandoned
- 2006-07-31 CN CNA2006800286267A patent/CN101238104A/zh active Pending
- 2006-07-31 KR KR1020087002810A patent/KR20080031370A/ko not_active Application Discontinuation
- 2006-07-31 MX MX2008001114A patent/MX2008001114A/es not_active Application Discontinuation
- 2006-07-31 BR BRPI0614535-3A patent/BRPI0614535A2/pt not_active IP Right Cessation
- 2006-07-31 US US11/997,489 patent/US20080176902A1/en not_active Abandoned
- 2006-07-31 EP EP06769591A patent/EP1912944A1/en not_active Withdrawn
- 2006-07-31 UY UY29713A patent/UY29713A1/es not_active Application Discontinuation
- 2006-07-31 WO PCT/SE2006/000922 patent/WO2007015668A1/en active Application Filing
- 2006-07-31 JP JP2008524934A patent/JP2009503066A/ja active Pending
- 2006-07-31 CA CA002617406A patent/CA2617406A1/en not_active Abandoned
- 2006-08-02 AR ARP060103359A patent/AR056013A1/es not_active Application Discontinuation
-
2007
- 2007-12-27 IL IL188484A patent/IL188484A0/en unknown
-
2008
- 2008-01-16 ZA ZA200800488A patent/ZA200800488B/xx unknown
- 2008-02-29 NO NO20081079A patent/NO20081079L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
TW200734305A (en) | 2007-09-16 |
AU2006276346A1 (en) | 2007-02-08 |
US20080176902A1 (en) | 2008-07-24 |
NO20081079L (no) | 2008-02-29 |
JP2009503066A (ja) | 2009-01-29 |
ZA200800488B (en) | 2008-12-31 |
IL188484A0 (en) | 2008-04-13 |
CA2617406A1 (en) | 2007-02-08 |
KR20080031370A (ko) | 2008-04-08 |
MX2008001114A (es) | 2008-03-11 |
BRPI0614535A2 (pt) | 2011-04-05 |
EP1912944A1 (en) | 2008-04-23 |
CN101238104A (zh) | 2008-08-06 |
UY29713A1 (es) | 2007-02-28 |
WO2007015668A1 (en) | 2007-02-08 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FA | Abandonment or withdrawal |