AR047922A1 - Nuevos derivados de pentafluorsulfanilo, su obtencion y su utilizacion como agentes farmaceuticos - Google Patents
Nuevos derivados de pentafluorsulfanilo, su obtencion y su utilizacion como agentes farmaceuticosInfo
- Publication number
- AR047922A1 AR047922A1 ARP050100812A ARP050100812A AR047922A1 AR 047922 A1 AR047922 A1 AR 047922A1 AR P050100812 A ARP050100812 A AR P050100812A AR P050100812 A ARP050100812 A AR P050100812A AR 047922 A1 AR047922 A1 AR 047922A1
- Authority
- AR
- Argentina
- Prior art keywords
- obtaining
- pentafluorsulfanilo
- pharmaceutical agents
- new derivatives
- compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Son objetos de la presente los compuestos de la formula (1), sus sales farmacéuticamente aceptables, formas enantioméricas, diastereoisomeros y racematos, la obtencion de los compuestos recién mencionados, los medicamentos que los contienen y su fabricacion, así como el uso de los compuestos recién mencionados para el control o prevencion de enfermedades, tales como el cáncer.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP04005275 | 2004-03-05 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR047922A1 true AR047922A1 (es) | 2006-03-01 |
Family
ID=34895965
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP050100812A AR047922A1 (es) | 2004-03-05 | 2005-03-03 | Nuevos derivados de pentafluorsulfanilo, su obtencion y su utilizacion como agentes farmaceuticos |
Country Status (12)
Country | Link |
---|---|
US (1) | US7235574B2 (es) |
EP (1) | EP1725549A1 (es) |
JP (1) | JP2007526275A (es) |
KR (1) | KR20060124746A (es) |
CN (1) | CN1930153A (es) |
AR (1) | AR047922A1 (es) |
AU (1) | AU2005229352A1 (es) |
BR (1) | BRPI0508485A (es) |
CA (1) | CA2557402A1 (es) |
RU (1) | RU2006135084A (es) |
TW (1) | TW200531688A (es) |
WO (1) | WO2005095388A1 (es) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7317124B2 (en) * | 2003-11-13 | 2008-01-08 | Sanofi-Aventis Deutschland Gmbh | Ortho-substituted pentafluorosulfanylbenzenes, process for their preparation and their use as valuable synthetic intermediates |
TW200533657A (en) | 2004-02-17 | 2005-10-16 | Esteve Labor Dr | Substituted pyrazoline compounds, their preparation and use as medicaments |
TW200612914A (en) * | 2004-03-05 | 2006-05-01 | Hoffmann La Roche | Novel oxidized thioether derivatives, their manufacture and use as pharmaceutical agents |
TW200533346A (en) * | 2004-03-18 | 2005-10-16 | Hoffmann La Roche | Novel ether derivatives, their manufacture and use as pharmaceutical agents |
US20060069095A1 (en) * | 2004-09-24 | 2006-03-30 | Thomas Hofmeister | Azole derivatives |
WO2008101212A2 (en) * | 2007-02-16 | 2008-08-21 | State University Of New York At Albany | Pentafluorosulfanyl containing amino acids |
WO2009028514A1 (ja) * | 2007-08-28 | 2009-03-05 | Ube Industries, Ltd. | ペンタフルオロスルファニルベンゼン化合物の製造方法、及び新規なペンタフルオロスルファニルベンゼン化合物 |
CN101981034B (zh) * | 2008-02-05 | 2013-08-14 | 赛诺菲-安万特 | 作为par1抑制剂的三唑并哒嗪、其制备及其制备药物的用途 |
RU2494100C2 (ru) * | 2008-02-05 | 2013-09-27 | Санофи-Авентис | Соли триазолия в качестве ингибиторов par1, их получение и применение в качестве лекарственного средства |
WO2009097972A1 (de) * | 2008-02-05 | 2009-08-13 | Sanofi-Aventis | Sf5-derivate als par1-inhibitoren, ihre herstellung und verwendung als arzneimittel |
WO2012094451A1 (en) * | 2011-01-06 | 2012-07-12 | Beta Pharma Canada Inc. | Novel ureas for the treatment and prevention of cancer |
CN103380110A (zh) | 2011-02-15 | 2013-10-30 | 宇部兴产株式会社 | 生产芳基硫五氟化物的工业方法 |
CN106414402A (zh) * | 2013-11-01 | 2017-02-15 | 宇部兴产株式会社 | 丙烯酰(氧基或氨基)五氟硫烷基苯化合物、其药学可接受的盐及其前药 |
CN112920133B (zh) * | 2021-01-29 | 2022-09-16 | 中国医科大学 | (e)-4-甲基-2-(4-(三氟甲基)苯乙烯基)噁唑类化合物及其制备方法与用途 |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0912562A1 (en) | 1996-07-19 | 1999-05-06 | Takeda Chemical Industries, Ltd. | Heterocyclic compounds, their production and use |
PE20011178A1 (es) | 2000-04-07 | 2001-11-19 | Takeda Chemical Industries Ltd | Compuestos heterociclicos y su produccion |
US6984653B2 (en) * | 2001-10-05 | 2006-01-10 | Takeda Pharmaceutical Company Limited | Heterocyclic compounds, oxazole derivatives, process for preparation of the same and use thereof |
JP2003277379A (ja) * | 2002-01-17 | 2003-10-02 | Takeda Chem Ind Ltd | 含窒素複素環化合物、その製造法および用途 |
JP2004059452A (ja) | 2002-07-25 | 2004-02-26 | Asahi Glass Co Ltd | ペンタフルオロサルファー置換ベンズイミダゾール化合物およびその製造方法 |
US7596415B2 (en) * | 2002-12-06 | 2009-09-29 | Medtronic, Inc. | Medical devices incorporating carbon nanotube material and methods of fabricating same |
US7259262B2 (en) * | 2003-10-24 | 2007-08-21 | Hoffmann-La Roche Inc. | Arylazole derivatives, their manufacture and use as pharmaceutical agents |
TW200612914A (en) * | 2004-03-05 | 2006-05-01 | Hoffmann La Roche | Novel oxidized thioether derivatives, their manufacture and use as pharmaceutical agents |
US7288557B2 (en) * | 2004-09-21 | 2007-10-30 | Hoffmann-La Roche Inc. | Triazole derivatives |
US20060069095A1 (en) * | 2004-09-24 | 2006-03-30 | Thomas Hofmeister | Azole derivatives |
US20060116407A1 (en) * | 2004-11-22 | 2006-06-01 | Birgit Bossenmaier | Amide derivatives |
-
2005
- 2005-03-01 TW TW094106110A patent/TW200531688A/zh unknown
- 2005-03-03 AR ARP050100812A patent/AR047922A1/es unknown
- 2005-03-04 KR KR1020067018040A patent/KR20060124746A/ko not_active Application Discontinuation
- 2005-03-04 BR BRPI0508485-7A patent/BRPI0508485A/pt not_active IP Right Cessation
- 2005-03-04 CA CA002557402A patent/CA2557402A1/en not_active Abandoned
- 2005-03-04 EP EP05715739A patent/EP1725549A1/en not_active Withdrawn
- 2005-03-04 RU RU2006135084/04A patent/RU2006135084A/ru not_active Application Discontinuation
- 2005-03-04 JP JP2007501230A patent/JP2007526275A/ja active Pending
- 2005-03-04 CN CNA200580007086XA patent/CN1930153A/zh active Pending
- 2005-03-04 WO PCT/EP2005/002310 patent/WO2005095388A1/en active Application Filing
- 2005-03-04 US US11/073,227 patent/US7235574B2/en not_active Expired - Fee Related
- 2005-03-04 AU AU2005229352A patent/AU2005229352A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
CN1930153A (zh) | 2007-03-14 |
CA2557402A1 (en) | 2005-10-13 |
RU2006135084A (ru) | 2008-04-10 |
AU2005229352A1 (en) | 2005-10-13 |
EP1725549A1 (en) | 2006-11-29 |
KR20060124746A (ko) | 2006-12-05 |
TW200531688A (en) | 2005-10-01 |
JP2007526275A (ja) | 2007-09-13 |
US7235574B2 (en) | 2007-06-26 |
BRPI0508485A (pt) | 2007-07-31 |
WO2005095388A1 (en) | 2005-10-13 |
US20050197370A1 (en) | 2005-09-08 |
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FB | Suspension of granting procedure |