AR046205A1 - Formulacion farmaceutica de licofelona - Google Patents

Formulacion farmaceutica de licofelona

Info

Publication number
AR046205A1
AR046205A1 ARP040103905A ARP040103905A AR046205A1 AR 046205 A1 AR046205 A1 AR 046205A1 AR P040103905 A ARP040103905 A AR P040103905A AR P040103905 A ARP040103905 A AR P040103905A AR 046205 A1 AR046205 A1 AR 046205A1
Authority
AR
Argentina
Prior art keywords
water soluble
pharmaceutical formulation
copolymers
soluble polymer
licofelona
Prior art date
Application number
ARP040103905A
Other languages
English (en)
Inventor
F Sievert
Original Assignee
Merckle Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merckle Gmbh filed Critical Merckle Gmbh
Publication of AR046205A1 publication Critical patent/AR046205A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Neurosurgery (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Formulación farmacéutica sólida que comprende licofelona o una sal farmacéuticamente aceptable de la misma y por lo menos un polímero soluble en agua seleccionado entre hidroxialquil celulosa, metil celulosa, polivinil pirrolidonas y copolímeros de los mismos, alcoholes polivinílicos, copolímeros hidrolizados o parcialmente hidrolizados de N-vinilpirrolidona y ésteres vinílicos, y/o por lo menos un poliol soluble en agua seleccionado entre polietilen glicoles con un peso molecular que oscila entre 8000 y 20000 y alcoholes de azúcares. La formulación libera con rapidez el ingrediente activo. Uso de un polímero soluble en agua y/o un poliol soluble en agua para producir dicha formulación farmacéutica.
ARP040103905A 2003-10-31 2004-10-27 Formulacion farmaceutica de licofelona AR046205A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10351035A DE10351035A1 (de) 2003-10-31 2003-10-31 Pharmazeutische Licofelone-Formulierung

Publications (1)

Publication Number Publication Date
AR046205A1 true AR046205A1 (es) 2005-11-30

Family

ID=34485181

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP040103905A AR046205A1 (es) 2003-10-31 2004-10-27 Formulacion farmaceutica de licofelona

Country Status (4)

Country Link
AR (1) AR046205A1 (es)
DE (1) DE10351035A1 (es)
TW (1) TW200524592A (es)
WO (1) WO2005041920A2 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN109718220A (zh) * 2017-10-27 2019-05-07 天津药物研究院有限公司 Ml-4000包合物胶囊的制备方法
EP3593792A1 (de) 2018-07-11 2020-01-15 Welding GmbH & Co. KG Pharmazeutische zusammensetzung umfassend 6-(4-chlorphenyl)-2,2-dimethyl-7-phenyl-2,3-dihydro-1h-pyrrolizin-5-yl-essigsäurecholinsalz
WO2023089636A1 (en) * 2021-11-21 2023-05-25 Aizant Drug Research Solutions Private Limited Pharmaceutical compositions of licofelone

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6136839A (en) * 1995-06-12 2000-10-24 G. D. Searle & Co. Treatment of inflammation and inflammation-related disorders with a combination of a cyclooxygenase-2 inhibitor and a 5-lipoxygenase inhibitor
DE69709069T2 (de) * 1996-02-13 2002-07-04 Searle & Co Zusammensetzungen mit immunosuppressiven wirkungen, welche 5-lipoxygenase-inhibitoren und cyclooxygenase-2-inhibitoren enthalten
DE10121252A1 (de) * 2001-04-30 2002-11-07 Christos C Zouboulis Behandlung der Akne
EP1505964B1 (en) * 2002-05-17 2007-11-21 Merckle Gmbh Annelated pyrrole compounds as proton pump inhibitors for treating ulcer

Also Published As

Publication number Publication date
DE10351035A1 (de) 2005-05-25
WO2005041920A2 (de) 2005-05-12
WO2005041920A3 (de) 2005-07-14
TW200524592A (en) 2005-08-01

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