AR038924A1 - Utilizacion del acido 6-[3-(1-adamantil)-4-metoxifenil)-2-naftoico para el tratamiento de desordenes dermatologicos - Google Patents
Utilizacion del acido 6-[3-(1-adamantil)-4-metoxifenil)-2-naftoico para el tratamiento de desordenes dermatologicosInfo
- Publication number
- AR038924A1 AR038924A1 ARP030100823A ARP030100823A AR038924A1 AR 038924 A1 AR038924 A1 AR 038924A1 AR P030100823 A ARP030100823 A AR P030100823A AR P030100823 A ARP030100823 A AR P030100823A AR 038924 A1 AR038924 A1 AR 038924A1
- Authority
- AR
- Argentina
- Prior art keywords
- adapalene
- treatment
- inflammatory
- pharmaceutical composition
- weight
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0014—Skin, i.e. galenical aspects of topical compositions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/192—Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/06—Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/10—Anti-acne agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/12—Keratolytics, e.g. wart or anti-corn preparations
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/16—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
- A61K47/18—Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
- A61K47/183—Amino acids, e.g. glycine, EDTA or aspartame
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/32—Macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. carbomers, poly(meth)acrylates, or polyvinyl pyrrolidone
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Dermatology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cosmetics (AREA)
Abstract
Utilización del ácido 6-[3-(1-adamantil)-4-metoxifenil]-2-naftanoico (adapaleno) o de sus sales para la fabricación de una composición farmacéutica destinada al tratamiento de las afecciones dermatológicas de componente inflamatorio o proliferativo que comprende 0,3% de peso de adapaleno con respecto al peso total de la composición. Reivindicación 1: Utilización del ácido 6-[3-(1-adamantil)-4-metoxifenil]-2-naftanoico (adapaleno) o de sus sales para la fabricación de una composición farmacéutica destinada al tratamiento de las afecciones dermatológicas de componente inflamatorio o proliferativo elegidas entre los acnés vulgares, comedonianos, polimorfos, los acnés noduloquísticos, conglobata, los acnés secundarios tales como el acné solar, medicamentoso o profesional, las formas extendidas y/o severas de psoriasis, las ictiosis y los estados ictiosiformes, la enfermedad de Darier, las queratodermias palmoplantares y la queratosis pilar, y las pigmentaciones postinflamatorias, caracterizada porque la composición farmacéutica comprende 0,3% de peso de adapaleno con respecto al peso total de la composición. Reivindicación 7: Composición farmacéutica que comprende, en un medio fisiológicamente aceptable, ácido 6-[3-(1-adamantil)-4-metoxifenil]-2-naftanoico (adapaleno) o de sus sales destinada al tratamiento de las afecciones dermatológicas de componente inflamatorio proliferativo caracterizada porque comprende 0,3% de peso de adapaleno con respecto al peso total de la composición.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0203070A FR2837101B1 (fr) | 2002-03-12 | 2002-03-12 | Utilisation de l'acide 6-[1-adamantyl)-4-methoxyphenyl]-2- naphthoique pour le traitement de desordres dermatologiques |
Publications (1)
Publication Number | Publication Date |
---|---|
AR038924A1 true AR038924A1 (es) | 2005-02-02 |
Family
ID=27772059
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP030100823A AR038924A1 (es) | 2002-03-12 | 2003-03-11 | Utilizacion del acido 6-[3-(1-adamantil)-4-metoxifenil)-2-naftoico para el tratamiento de desordenes dermatologicos |
Country Status (4)
Country | Link |
---|---|
KR (1) | KR101007161B1 (es) |
AR (1) | AR038924A1 (es) |
FR (1) | FR2837101B1 (es) |
ZA (1) | ZA200405853B (es) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR100798853B1 (ko) * | 2005-02-15 | 2008-01-28 | (주)한국스티펠 | 레티노이드를 유효성분으로 하는 백반증 예방 및 치료용 약학적 조성물 |
FR2901701B1 (fr) * | 2006-05-31 | 2010-10-29 | Galderma Res & Dev | Compostions comprenant au moins un derive de l'acide naphtoique et au moins un agent filmogene, leurs procedes de preparation, et leurs utilisations |
FR2903603B1 (fr) | 2006-07-13 | 2009-03-20 | Galderma Res & Dev S N C Snc | Combinaison d'adapalene et de peroxyde de benzole dans le traitement de l'acne |
EP2097075A1 (fr) * | 2006-11-20 | 2009-09-09 | Galderma Research & Development, S.N.C. | Utilisation d'adapalène pour moduler l'expression de cd1d ou il-10. |
EP2097076A1 (fr) * | 2006-11-20 | 2009-09-09 | Galderma Research & Development, S.N.C. | Utilisation d'adapalène pour moduler l'expression de l'il-1ra. |
JP2013518920A (ja) | 2010-02-09 | 2013-05-23 | ガルデルマ・リサーチ・アンド・デヴェロップメント | 非白人系人種における炎症後色素沈着の減少と共にざ瘡の処置を目的とする、アダパレンと過酸化ベンゾイルとの組合せを含む皮膚科学的組成物 |
JP2013527161A (ja) | 2010-04-29 | 2013-06-27 | ガルデルマ・リサーチ・アンド・デヴェロップメント | アダパレン0.3%による瘢痕の処置方法 |
EP2854791A1 (en) | 2012-05-25 | 2015-04-08 | Galderma Research & Development | Treatment of preadolescent moderate acne vulgaris |
EP3220903A1 (fr) * | 2014-11-20 | 2017-09-27 | Galderma S.A. | Compositions comprenant un compose de la famille des avermectines et un compose agoniste d'au moins un des recepteurs de l'acide retinoique pour le traitement de l'acne |
KR102486502B1 (ko) * | 2015-09-15 | 2023-01-09 | 주식회사 엘지생활건강 | 여드름 치료제 전달을 위한 용해성 미세바늘 패치 |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
LU85849A1 (fr) * | 1985-04-11 | 1986-11-05 | Cird | Derives benzonaphtaleniques,leur procede de preparation et leur application dans les domaines pharmaceutiques et cosmetiques |
FR2730930B1 (fr) * | 1995-02-27 | 1997-04-04 | Oreal | Utilisation d'inhibiteurs de no-synthase pour diminuer l'effet irritant cutane de produits utilises dans le domaine cosmetique ou pharmaceutique |
-
2002
- 2002-03-12 FR FR0203070A patent/FR2837101B1/fr not_active Expired - Fee Related
-
2003
- 2003-03-11 AR ARP030100823A patent/AR038924A1/es not_active Application Discontinuation
- 2003-03-12 KR KR1020047014228A patent/KR101007161B1/ko active IP Right Grant
-
2004
- 2004-07-22 ZA ZA200405853A patent/ZA200405853B/xx unknown
Also Published As
Publication number | Publication date |
---|---|
ZA200405853B (en) | 2008-10-29 |
FR2837101A1 (fr) | 2003-09-19 |
KR20040111394A (ko) | 2004-12-31 |
FR2837101B1 (fr) | 2004-07-02 |
KR101007161B1 (ko) | 2011-01-12 |
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