AR027897A1 - FORM OF CELECOXIB IN SOLID STATE THAT EXHIBIT INCREASED BIODISPONIBILITY - Google Patents

FORM OF CELECOXIB IN SOLID STATE THAT EXHIBIT INCREASED BIODISPONIBILITY

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Publication number
AR027897A1
AR027897A1 ARP000106473A ARP000106473A AR027897A1 AR 027897 A1 AR027897 A1 AR 027897A1 AR P000106473 A ARP000106473 A AR P000106473A AR P000106473 A ARP000106473 A AR P000106473A AR 027897 A1 AR027897 A1 AR 027897A1
Authority
AR
Argentina
Prior art keywords
biodisponibility
celecoxib
solid state
exhibit increased
exhibit
Prior art date
Application number
ARP000106473A
Other languages
Spanish (es)
Original Assignee
Pharmacia Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia Corp filed Critical Pharmacia Corp
Publication of AR027897A1 publication Critical patent/AR027897A1/en

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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ARP000106473A 1999-12-08 2000-12-05 FORM OF CELECOXIB IN SOLID STATE THAT EXHIBIT INCREASED BIODISPONIBILITY AR027897A1 (en)

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ARP000106473A AR027897A1 (en) 1999-12-08 2000-12-05 FORM OF CELECOXIB IN SOLID STATE THAT EXHIBIT INCREASED BIODISPONIBILITY
ARP000106475A AR030039A1 (en) 1999-12-08 2000-12-06 PHARMACEUTICAL COMPOSITION THAT INCLUDES A SELECTIVE INHIBITOR DRUG OF CYCLOOXYGENASA-2, ITS USE IN THE MANUFACTURE OF A MEDICINAL PRODUCT TO TREAT OR PREVENT AFFECTIONS THROUGH CYCLOOXYGENASE-2 AND METHOD TO MAKE SUCH MEDICINAL PRODUCT

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US7927613B2 (en) 2002-02-15 2011-04-19 University Of South Florida Pharmaceutical co-crystal compositions
EP1494998A2 (en) 2002-03-01 2005-01-12 University Of South Florida Multiple-component solid phases containing at least one active pharmaceutical ingredient
BR0309913A (en) * 2002-05-13 2005-06-07 Pharmacia Corp Stable amorphous celecoxib composite and manufacturing process
AU2003243354A1 (en) 2002-05-31 2003-12-19 Transform Pharmaceuticals, Inc. Novel conazole crystalline forms and related processes, pharmaceutical compositions and methods
CA2489984A1 (en) * 2002-06-21 2003-12-31 Transform Pharmaceuticals, Inc. Pharmaceutical compositions with improved dissolution
AU2003267231A1 (en) * 2002-09-20 2004-04-08 Transform Pharmaceuticals, Inc. Pharmaceutical compositions with improved dissolution
JP5021934B2 (en) * 2002-12-30 2012-09-12 トランスフォーム・ファーマシューティカルズ・インコーポレイテッド Pharmaceutical composition having improved solubility
US8183290B2 (en) 2002-12-30 2012-05-22 Mcneil-Ppc, Inc. Pharmaceutically acceptable propylene glycol solvate of naproxen
PL1916994T3 (en) * 2004-06-29 2014-05-30 Takeda Pharma As Manufacturing of quick release pharmaceutical composition of water insoluble drugs and pharmaceutical compositions obtained by the process of the invention
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US20080171746A1 (en) * 2005-03-14 2008-07-17 Thomas Klein Method for Preventing Cardiovascular Diseases
CN103462920A (en) * 2012-06-06 2013-12-25 南京亿华药业有限公司 Oral cyclo-oxygenase-2 inhibitor Celecoxib composition
CN103524416B (en) * 2013-10-29 2016-08-17 湖北华世通生物医药科技有限公司 A kind of Novel celecoxib crystal form A and preparation method thereof
CN103539739B (en) * 2013-10-30 2016-02-10 中美华世通生物医药科技（武汉）有限公司 A kind of Novel celecoxib crystal form B and preparation method thereof
CN103508958A (en) * 2013-10-30 2014-01-15 中美华世通生物医药科技（武汉）有限公司 Novel celecoxib crystal form C and preparation method thereof
KR101476096B1 (en) * 2014-03-28 2014-12-24 대원제약주식회사 Pharmaceutical composition comprising celecoxib with improved solubility

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MY128366A (en) 2007-01-31
OA11831A (en) 2005-08-23
ECSP003807A (en) 2005-07-06
HUP0200580A2 (en) 2002-11-28
CN1411447A (en) 2003-04-16
CN1216869C (en) 2005-08-31
PT1150959E (en) 2008-04-21
CZ20012875A3 (en) 2002-02-13
PT1150960E (en) 2005-06-30
BG65239B1 (en) 2007-09-28
AR030039A1 (en) 2003-08-13
YU57801A (en) 2005-07-19
CO5251445A1 (en) 2003-02-28
ZA200107149B (en) 2003-02-28
PE20010911A1 (en) 2001-09-10
MY128971A (en) 2007-03-30
TWI276435B (en) 2007-03-21
EA200401397A1 (en) 2005-08-25
ES2236011T3 (en) 2005-07-16
HUP0200580A3 (en) 2002-12-28
KR100717570B1 (en) 2007-05-15
WO2001041536A2 (en) 2001-06-14
SV2002000235A (en) 2002-06-13
ZA200107146B (en) 2002-08-29
KR20020002386A (en) 2002-01-09
AU2041201A (en) 2001-06-18
NZ529933A (en) 2005-06-24

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